Members of CRF family and their receptors: from past to future
Liapakis, G, Venihaki, M, Margioris, A, Grigoriadis, D, Gkountelias, K
Published in Current medicinal chemistry (01.06.2011)
Published in Current medicinal chemistry (01.06.2011)
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Urocortin III, A Brain Neuropeptide of the Corticotropin-Releasing Hormone Family: Modulation by Stress and Attenuation of Some Anxiety-Like Behaviours
Venihaki, M., Sakihara, S., Subramanian, S., Dikkes, P., Weninger, S. C., Liapakis, G., Graf, T., Majzoub, J. A.
Published in Journal of neuroendocrinology (01.05.2004)
Published in Journal of neuroendocrinology (01.05.2004)
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Development of a selective agonist at the somatostatin receptor subtype sstr1
Liapakis, G, Hoeger, C, Rivier, J, Reisine, T
Published in The Journal of pharmacology and experimental therapeutics (01.03.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1996)
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Alanine Scanning Mutagenesis of the Second Extracellular Loop of Type 1 Corticotropin-Releasing Factor Receptor Revealed Residues Critical for Peptide Binding
Gkountelias, Kostas, Tselios, Theodoros, Venihaki, Maria, Deraos, George, Lazaridis, Iakovos, Rassouli, Olga, Gravanis, Achille, Liapakis, George
Published in Molecular pharmacology (01.04.2009)
Published in Molecular pharmacology (01.04.2009)
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A novel role of peripheral corticotropin-releasing hormone (CRH) on dermal fibroblasts
Rassouli, Olga, Liapakis, George, Lazaridis, Iakovos, Sakellaris, George, Gkountelias, Kostas, Gravanis, Achille, Margioris, Andrew N, Karalis, Katia P, Venihaki, Maria
Published in PloS one (13.07.2011)
Published in PloS one (13.07.2011)
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Novel long-acting somatostatin analog with endocrine selectivity: potent suppression of growth hormone but not of insulin
Afargan, M, Janson, E T, Gelerman, G, Rosenfeld, R, Ziv, O, Karpov, O, Wolf, A, Bracha, M, Shohat, D, Liapakis, G, Gilon, C, Hoffman, A, Stephensky, D, Oberg, K
Published in Endocrinology (Philadelphia) (01.01.2001)
Published in Endocrinology (Philadelphia) (01.01.2001)
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Lanthionine−Somatostatin Analogs: Synthesis, Characterization, Biological Activity, and Enzymatic Stability Studies
Ösapay, George, Prokai, Laszlo, Kim, Ho-Seung, Medzihradszky, Katalin F, Coy, David H, Liapakis, George, Reisine, Terry, Melacini, Giuseppe, Zhu, Qin, Wang, Susan H.-H, Mattern, Ralph-Heiko, Goodman, Murray
Published in Journal of medicinal chemistry (04.07.1997)
Published in Journal of medicinal chemistry (04.07.1997)
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Template-constrained cyclic peptide analogues of somatostatin: subtype-selective binding to somatostatin receptors and antiangiogenic activity
Suich, Daniel J, Mousa, Shaker A, Singh, Gurke, Liapakis, George, Reisine, Terry, DeGrado, William F
Published in Bioorganic & medicinal chemistry (01.09.2000)
Published in Bioorganic & medicinal chemistry (01.09.2000)
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Structural and Compositional Determinants of Cortistatin Activity
Criado, J R, Li, Haitao, Jiang, Xiaohui, Spina, M, Huitron-Resendiz, S, Liapakis, G, Calbet, M, Siehler, S, Henriksen, S J, Koob, G, Hoyer, D, Sutcliffe, J G, Goodman, M, De Lecea, L
Published in Journal of neuroscience research (15.06.1999)
Published in Journal of neuroscience research (15.06.1999)
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Activation of the beta 2-adrenergic receptor involves disruption of an ionic lock between the cytoplasmic ends of transmembrane segments 3 and 6
Ballesteros, J A, Jensen, A D, Liapakis, G, Rasmussen, S G, Shi, L, Gether, U, Javitch, J A
Published in The Journal of biological chemistry (03.08.2001)
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Published in The Journal of biological chemistry (03.08.2001)
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Structural and compositional determinants of cortistatin activity
Criado, José R., Li, Haitao, Jiang, Xiaohui, Spina, Mariarosa, Huitrón-Reséndiz, Salvador, Liapakis, George, Calbet, Marta, Siehler, Sandra, Henriksen, Steven J., Koob, George, Hoyer, Daniel, Sutcliffe, J. Gregor, Goodman, Murray, de Lecea, Luis
Published in Journal of neuroscience research (15.06.1999)
Published in Journal of neuroscience research (15.06.1999)
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