Cellular Oxygen Sensing: Crystal Structure of Hypoxia-Inducible Factor Prolyl Hydroxylase (PHD2)
McDonough, Michael A., Li, Vivian, Flashman, Emily, Chowdhury, Rasheduzzaman, Mohr, Christopher, Liénard, Benoît M. R., Zondlo, James, Oldham, Neil J., Clifton, Ian J., Lewis, Jeffrey, McNeill, Luke A., Kurzeja, Robert J. M., Hewitson, Kirsty S., Yang, Evelyn, Jordan, Steven, Syed, Rashid S., Schofield, Christopher J.
Published in Proceedings of the National Academy of Sciences - PNAS (27.06.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (27.06.2006)
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Structural basis for the broad-spectrum inhibition of metallo-beta-lactamases by thiols
Lienard, Benoit M. R., Garau, Gianpiero, Horsfall, Louise, Karsisiotis, Andreas I., Damblon, Christian, Lassaux, Patricia, Papamicael, Cyril, Roberts, Gordon C. K., Galleni, Moreno, Dideberg, Otto, Frere, Jean-Marie, Schofield, Christopher J.
Published in Organic & biomolecular chemistry (01.01.2008)
Published in Organic & biomolecular chemistry (01.01.2008)
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Dynamic Combinatorial Mass Spectrometry Leads to Metallo-β-lactamase Inhibitors
Liénard, Benoît M. R, Hüting, Rebekka, Lassaux, Patricia, Galleni, Moreno, Frère, Jean-Marie, Schofield, Christopher J
Published in Journal of medicinal chemistry (14.02.2008)
Published in Journal of medicinal chemistry (14.02.2008)
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Crystal structures of histone demethylase JMJD2A reveal basis for substrate specificity
NG, Stanley S, KAVANAGH, Kathryn L, ROSE, Nathan R, OFFER, John, SCHEINOST, Johanna C, BOROWSKI, Tomasz, SUNDSTROM, Michael, SCHOFIELD, Christopher J, OPPERMANN, Udo, MCDONOUGH, Michael A, BUTLER, Danica, PILKA, Ewa S, LIENARD, Benoit M. R, BRAY, James E, SAVITSKY, Pavel, GILEADI, Opher, VON DELFT, Frank
Published in Nature (05.07.2007)
Published in Nature (05.07.2007)
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Broad antibiotic resistance profile of the subclass B3 metallo‐β‐lactamase GOB‐1, a di‐zinc enzyme
Horsfall, Louise E., Izougarhane, Youssef, Lassaux, Patricia, Selevsek, Nathalie, Liénard, Benoit M. R., Poirel, Laurent, Kupper, Michael B., Hoffmann, Kurt M., Frère, Jean‐Marie, Galleni, Moreno, Bebrone, Carine
Published in The FEBS journal (01.04.2011)
Published in The FEBS journal (01.04.2011)
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Combined Mass Spectrometry and Dynamic Chemistry Approach to Identify Metalloenzyme Inhibitors
Liénard, Benoît M. R., Selevsek, Nathalie, Oldham, Neil J., Schofield, Christopher J.
Published in ChemMedChem (12.02.2007)
Published in ChemMedChem (12.02.2007)
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Inhibitor Scaffolds for 2-Oxoglutarate-Dependent Histone Lysine Demethylases
Rose, Nathan R, Ng, Stanley S, Mecinović, Jasmin, Liénard, Benoît M.R, Bello, Simon H, Sun, Zhe, McDonough, Michael A, Oppermann, Udo, Schofield, Christopher J
Published in Journal of medicinal chemistry (27.11.2008)
Published in Journal of medicinal chemistry (27.11.2008)
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Inhibitors of the FEZ-1 metallo-β-lactamase
Liénard, Benoît M.R., Horsfall, Louise E., Galleni, Moreno, Frère, Jean-Marie, Schofield, Christopher J.
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
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Studies on ternary metallo-β lactamase-inhibitor complexes using electrospray ionization mass spectrometry
SELEVSEK, Nathalie, THOLEY, Andreas, HEINZLE, Elmar, LIENARD, Benoit M. R, OLDHAM, Neil J, SCHOFIELD, Christopher J, HEINZ, Uwe, ADOLPH, Hans-Werner, FREEE, Jean-Marie
Published in Journal of the American Society for Mass Spectrometry (01.07.2006)
Published in Journal of the American Society for Mass Spectrometry (01.07.2006)
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Structural and Mechanistic Studies on the Inhibition of the Hypoxia-inducible Transcription Factor Hydroxylases by Tricarboxylic Acid Cycle Intermediates
Hewitson, Kirsty S., Liénard, Benoit M.R., McDonough, Michael A., Clifton, Ian J., Butler, Danica, Soares, Alexie S., Oldham, Neil J., McNeill, Luke A., Schofield, Christopher J.
Published in The Journal of biological chemistry (02.02.2007)
Published in The Journal of biological chemistry (02.02.2007)
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Studies on ternary metallo-β lactamase-inhibitor complexes using electrospray ionization mass spectrometry
Selevsek, Nathalie, Tholey, Andreas, Heinzle, Elmar, Liénard, Benoit M R, Oldham, Neil J, Schofield, Christopher J, Heinz, Uwe, Adolph, Hans-Werner, Frère, Jean-Marie
Published in Journal of the American Society for Mass Spectrometry (01.07.2006)
Published in Journal of the American Society for Mass Spectrometry (01.07.2006)
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Cover Picture: ESI-MS Studies on Prolyl Hydroxylase Domain 2 Reveal a New Metal Binding Site (ChemMedChem 4/2008)
Mecinović, Jasmin, Chowdhury, Rasheduzzaman, Liénard, Benoît M. R., Flashman, Emily, Buck, Matthew R. G., Oldham, Neil J., Schofield, Christopher J.
Published in ChemMedChem (14.04.2008)
Published in ChemMedChem (14.04.2008)
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Broad antibiotic resistance profile of the subclass B3 metallo-[beta]-lactamase GOB-1, a di-zinc enzyme
Horsfall, Louise E, Izougarhane, Youssef, Lassaux, Patricia, Selevsek, Nathalie, Liénard, Benoit M. R, Poirel, Laurent, Kupper, Michael B, Hoffmann, Kurt M, Frère, Jean-Marie, Galleni, Moreno, Bebrone, Carine
Published in The FEBS journal (01.04.2011)
Published in The FEBS journal (01.04.2011)
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