In-Depth Study of Tripeptide-Based α-Ketoheterocycles as Inhibitors of Thrombin. Effective Utilization of the S1‘ Subsite and Its Implications to Structure-Based Drug Design
Costanzo, Michael J, Almond, Harold R, Hecker, Leonard R, Schott, Mary R, Yabut, Stephen C, Zhang, Han-Cheng, Andrade-Gordon, Patricia, Corcoran, Thomas W, Giardino, Edward C, Kauffman, Jack A, Lewis, Joan M, de Garavilla, Lawrence, Haertlein, Barbara J, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Journal Article
In-Depth Study of Tripeptide-Based α-Ketoheterocycles as Inhibitors of Thrombin. Effective Utilization of the S1‘ Subsite and Its Implications to Structure-Based Drug Design
Costanzo, Michael J, Almond, Harold R, Hecker, Leonard R, Schott, Mary R, Yabut, Stephen C, Zhang, Han-Cheng, Andrade-Gordon, Patricia, Corcoran, Thomas W, Giardino, Edward C, Kauffman, Jack A, Lewis, Joan M, de Garavilla, Lawrence, Haertlein, Barbara J, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (15.11.2007)
Published in Journal of medicinal chemistry (15.11.2007)
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Journal Article
Potent Thrombin Inhibitors That Probe the S1‘ Subsite: Tripeptide Transition State Analogues Based on a Heterocycle-Activated Carbonyl Group
Costanzo, Michael J, Maryanoff, Bruce E, Hecker, Leonard R, Schott, Mary R, Yabut, Stephen C, Zhang, Han-Cheng, Andrade-Gordon, Patricia, Kauffman, Jack A, Lewis, Joan M, Krishnan, Raman, Tulinsky, Alexander
Published in Journal of medicinal chemistry (02.08.1996)
Published in Journal of medicinal chemistry (02.08.1996)
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Journal Article
1,2,3,4-Tetrahydroquinoline-containing αvβ3 integrin antagonists with enhanced oral bioavailability
GHOSH, Shyamali, SANTULLI, Rosemary J, THOMPSON, Andrew S, CHEN, Ian, KAWAHAMA, Reiko, TUMAN, Robert W, GALEMMO, Robert A, JOHNSON, Dana L, DAMIANO, Bruce P, MARYANOFF, Bruce E, KINNEY, William A, DECORTE, Bart L, LIU, Li, LEWIS, Joan M, PROOST, Jef C, LEO, Gregory C, MASUCCI, John, HAGEMAN, William E
Published in Bioorganic & medicinal chemistry letters (01.12.2004)
Published in Bioorganic & medicinal chemistry letters (01.12.2004)
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Journal Article
In-depth study of tripeptide-based alpha-ketoheterocycles as inhibitors of thrombin. Effective utilization of the S-1 ' subsite and its implications to structure-based drug design
Costanzo, MJ, Almond, HR, Hecker, LR, Schott, MR, Yabut, SC, Zhang, HC, Andrade-Gordon, P, Corcoran, TW, Giardino, EC, Kauffman, JA, Lewis, JM, de Garavilla, L, Haertlein, BJ, Maryanoff, BE
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
Get full text
Journal Article
In-Depth Study of Tripeptide-Based α-Ketoheterocycles as Inhibitors of Thrombin. Effective Utilization of the S 1 ‘ Subsite and Its Implications to Structure-Based Drug Design
Costanzo, Michael J., Almond, Harold R., Hecker, Leonard R., Schott, Mary R., Yabut, Stephen C., Zhang, Han-Cheng, Andrade-Gordon, Patricia, Corcoran, Thomas W., Giardino, Edward C., Kauffman, Jack A., Lewis, Joan M., de Garavilla, Lawrence, Haertlein, Barbara J., Maryanoff, Bruce E.
Published in Journal of medicinal chemistry (15.11.2007)
Published in Journal of medicinal chemistry (15.11.2007)
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Journal Article
1,2,3,4-Tetrahydroquinoline-containing α Vβ 3 integrin antagonists with enhanced oral bioavailability
Ghosh, Shyamali, Santulli, Rosemary J., Kinney, William A., DeCorte, Bart L., Liu, Li, Lewis, Joan M., Proost, Jef C., Leo, Gregory C., Masucci, John, Hageman, William E., Thompson, Andrew S., Chen, Ian, Kawahama, Reiko, Tuman, Robert W., Galemmo, Robert A., Johnson, Dana L., Damiano, Bruce P., Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (06.12.2004)
Published in Bioorganic & medicinal chemistry letters (06.12.2004)
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Journal Article
In-depth study of tripeptide-based α-ketoheterocycles as inhibitors of thrombin. Effective utilization of the S1' subsite and its implications to structure-based drug designs
COSTANZO, Michael J, ALMOND, Harold R, LEWIS, Joan M, DE GARAVILLA, Lawrence, HAERTLEIN, Barbara J, MARYANOFF, Bruce E, HECKER, Leonard R, SCHOTT, Mary R, YABUT, Stephen C, ZHANG, Han-Cheng, ANDRADE-GORDON, Patricia, CORCORAN, Thomas W, GIARDINO, Edward C, KAUFFMAN, Jack A
Published in Journal of medicinal chemistry (2005)
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Published in Journal of medicinal chemistry (2005)
Journal Article
Potent thrombin inhibitors that probe the S-1' subsite: Tripeptide transition state analogues based on a heterocycle-activated carbonyl group
Costanzo, MJ, Maryanoff, BE, Hecker, LR, Schott, MR, Yabut, SC, Zhang, HC, AndradeGordon, P, Kauffman, JA, Lewis, JM, Krishnan, R, Tulinsky, A
Published in Journal of medicinal chemistry (02.08.1996)
Published in Journal of medicinal chemistry (02.08.1996)
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Journal Article
1,2,3,4-Tetrahydroquinoline-containing alphaVbeta3 integrin antagonists with enhanced oral bioavailability
Ghosh, Shyamali, Santulli, Rosemary J, Kinney, William A, Decorte, Bart L, Liu, Li, Lewis, Joan M, Proost, Jef C, Leo, Gregory C, Masucci, John, Hageman, William E, Thompson, Andrew S, Chen, Ian, Kawahama, Reiko, Tuman, Robert W, Galemmo, Jr, Robert A, Johnson, Dana L, Damiano, Bruce P, Maryanoff, Bruce E
Published in Bioorganic & medicinal chemistry letters (06.12.2004)
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Published in Bioorganic & medicinal chemistry letters (06.12.2004)
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Novel thrombin inhibitors that are based on a macrocyclic tripeptide motif
Greco, Michael N., Powell, Eugene T., Hecker, Leonard R., Andrade-Gordon, Patricia, Kauffman, Jack A., Lewis, Joan M., Ganesh, Venkatapathy, Tulinsky, Alexander, Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
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N.J. BRIEFS: All Editions
Teresa M. McAleavy, Joan Verdon, Lewis Krauskopf, Prashant Gopal and Martha McKay
Published in The Record (Hackensack, N.J.) (16.03.2005)
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Published in The Record (Hackensack, N.J.) (16.03.2005)
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