Antitrypanosomal Activity of Sterol 14α-Demethylase (CYP51) Inhibitors VNI and VFV in the Swiss Mouse Models of Chagas Disease Induced by the Trypanosoma cruzi Y Strain
Guedes-da-Silva, F H, Batista, D G J, Da Silva, C F, De Araújo, J S, Pavão, B P, Simões-Silva, M R, Batista, M M, Demarque, K C, Moreira, O C, Britto, C, Lepesheva, G I, Soeiro, M N C
Published in Antimicrobial agents and chemotherapy (01.04.2017)
Published in Antimicrobial agents and chemotherapy (01.04.2017)
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Different Therapeutic Outcomes of Benznidazole and VNI Treatments in Different Genders in Mouse Experimental Models of Trypanosoma cruzi Infection
Guedes-da-Silva, F H, Batista, D G J, da Silva, C F, Meuser, M B, Simões-Silva, M R, de Araújo, J S, Ferreira, C G, Moreira, O C, Britto, C, Lepesheva, G I, Soeiro, Maria de Nazaré C
Published in Antimicrobial agents and chemotherapy (01.12.2015)
Published in Antimicrobial agents and chemotherapy (01.12.2015)
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Role of C-terminal sequence of cytochrome P450scc in folding and functional activity
Strushkevich, N V, Harnastai, I N, Lepesheva, G I, Usanov, S A
Published in Biochemistry (Moscow) (01.09.2006)
Published in Biochemistry (Moscow) (01.09.2006)
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Biodiversity of CYP51 in trypanosomes
Lepesheva, G I, Hargrove, T Y, Ott, R D, Nes, W D, Waterman, M R
Published in Biochemical Society transactions (01.12.2006)
Published in Biochemical Society transactions (01.12.2006)
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Site-directed mutagenesis of cytochrome P450scc. II. Effect of replacement of the Arg425 and Arg426 residues on the structural and functional properties of the cytochrome P450scc
Azeva, T N, Gilep, A A, Lepesheva, G I, Strushkevich, N V, Usanov, S A
Published in Biochemistry (Moscow) (01.05.2001)
Published in Biochemistry (Moscow) (01.05.2001)
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CYP51 from Trypanosoma cruzi: A Phyla-Specific Residue in the B' Helix Defines Substrate Preferences of Sterol 14 alpha -Demethylase
Lepesheva, Galina I, Zaitseva, Natalia G, Nes, WDavid, Zhou, Wenxu, Arase, Miharu, Liu, Jialin, Hill, George C, Waterman, Michael R
Published in The Journal of biological chemistry (10.02.2006)
Published in The Journal of biological chemistry (10.02.2006)
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Sterol 14α-demethylase, an abundant and essential mixed-function oxidase
Waterman, Michael R., Lepesheva, Galina I.
Published in Biochemical and biophysical research communications (09.12.2005)
Published in Biochemical and biophysical research communications (09.12.2005)
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CYP51—the omnipotent P450
Lepesheva, Galina I, Waterman, Michael R
Published in Molecular and cellular endocrinology (27.02.2004)
Published in Molecular and cellular endocrinology (27.02.2004)
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CYP51 from Trypanosoma brucei Is Obtusifoliol-Specific
Lepesheva, Galina I, Nes, W. David, Zhou, Wenxu, Hill, George C, Waterman, Michael R
Published in Biochemistry (Easton) (24.08.2004)
Published in Biochemistry (Easton) (24.08.2004)
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Conservation in the CYP51 Family. Role of the B‘ Helix/BC Loop and Helices F and G in Enzymatic Function
Lepesheva, Galina I, Virus, Cornelia, Waterman, Michael R
Published in Biochemistry (Easton) (05.08.2003)
Published in Biochemistry (Easton) (05.08.2003)
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