Picomolar Inhibitors as Transition-State Probes of 5′-Methylthioadenosine Nucleosidases
Gutierrez, Jemy A, Luo, Minkui, Singh, Vipender, Li, Lei, Brown, Rosemary L, Norris, Gillian E, Evans, Gary B, Furneaux, Richard H, Tyler, Peter C, Painter, Gavin F, Lenz, Dirk H, Schramm, Vern L
Published in ACS chemical biology (01.11.2007)
Published in ACS chemical biology (01.11.2007)
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Energetic Mapping of Transition State Analogue Interactions with Human and Plasmodium falciparum Purine Nucleoside Phosphorylases
Lewandowicz, Andrzej, Ringia, Erika A. Taylor, Ting, Li-Min, Kim, Kami, Tyler, Peter C., Evans, Gary B., Zubkova, Olga V., Mee, Simon, Painter, Gavin F., Lenz, Dirk H., Furneaux, Richard H., Schramm, Vern L.
Published in The Journal of biological chemistry (26.08.2005)
Published in The Journal of biological chemistry (26.08.2005)
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Femtomolar Transition State Analogue Inhibitors of 5′-Methylthioadenosine/S-Adenosylhomocysteine Nucleosidase from Escherichia coli
Singh, Vipender, Evans, Gary B., Lenz, Dirk H., Mason, Jennifer M., Clinch, Keith, Mee, Simon, Painter, Gavin F., Tyler, Peter C., Furneaux, Richard H., Lee, Jeffrey E., Howell, P. Lynne, Schramm, Vern L.
Published in The Journal of biological chemistry (06.05.2005)
Published in The Journal of biological chemistry (06.05.2005)
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Synthesis, Formulation, and Adjuvanticity of Monodesmosidic Saponins with Olenanolic Acid, Hederagenin and Gypsogenin Aglycones, and some C‐28 Ester Derivatives
Greatrex, Ben W., Daines, Alison M., Hook, Sarah, Lenz, Dirk H., McBurney, Warren, Rades, Thomas, Rendle, Phillip M.
Published in ChemistryOpen (Weinheim) (01.12.2015)
Published in ChemistryOpen (Weinheim) (01.12.2015)
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Structure and Inhibition of a Quorum Sensing Target from Streptococcus pneumoniae
Singh, Vipender, Shi, Wuxian, Almo, Steven C, Evans, Gary B, Furneaux, Richard H, Tyler, Peter C, Painter, Gavin F, Lenz, Dirk H, Mee, Simon, Zheng, Renjian, Schramm, Vern L
Published in Biochemistry (Easton) (31.10.2006)
Published in Biochemistry (Easton) (31.10.2006)
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Syntheses and bio-activities of the L-enantiomers of two potent transition state analogue inhibitors of purine nucleoside phosphorylases
Clinch, K, Evans, GB, Fleet, GWJ, Furneaux, RH, Johnson, SW, Lenz, DH, Mee, SPH, Rands, PR, Schramm, VL, Ringia, EAT, Tyler, PC
Published in Organic & biomolecular chemistry (01.01.2006)
Published in Organic & biomolecular chemistry (01.01.2006)
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Second Generation Transition State Analogue Inhibitors of Human 5‘-Methylthioadenosine Phosphorylase
Evans, Gary B, Furneaux, Richard H, Lenz, Dirk H, Painter, Gavin F, Schramm, Vern L, Singh, Vipender, Tyler, Peter C
Published in Journal of medicinal chemistry (14.07.2005)
Published in Journal of medicinal chemistry (14.07.2005)
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A practical synthesis of (3R,4R)-N-tert-butoxycarbonyl-4-hydroxymethylpyrrolidin-3-ol
Clinch, Keith, Evans, Gary B., Furneaux, Richard H., Lenz, Dirk H., Mason, Jennifer M., Mee, Simon P. H., Tyler, Peter C., Wilcox, Sarah J.
Published in Organic & biomolecular chemistry (01.01.2007)
Published in Organic & biomolecular chemistry (01.01.2007)
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One-pot transformation of glycopyranosylcyanides to N-( t-butoxycarbonyl)methylamines
Lenz, Dirk H, Norris, Gillian E, Taylor, Carol M, Slim, George C
Published in Tetrahedron letters (02.07.2001)
Published in Tetrahedron letters (02.07.2001)
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Journal Article
Femtomolar Transition State Analogue Inhibitors of 5â²-Methylthioadenosine/S-Adenosylhomocysteine Nucleosidase from Escherichia coli
Vipender Singh, Gary B. Evans, Dirk H. Lenz, Jennifer M. Mason, Keith Clinch, Simon Mee, Gavin F. Painter, Peter C. Tyler, Richard H. Furneaux, Jeffrey E. Lee, P. Lynne Howell, Vern L. Schramm
Published in The Journal of biological chemistry (06.05.2005)
Published in The Journal of biological chemistry (06.05.2005)
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Journal Article
Inhibitors of nucleoside phosphorylases and nucleosidases
EVANS GARY B, HUBERT RICHARD, SCHRAMM VERN L, TYLER PETER C, ZUBKOVA OLGA V, LENZ DIRK H
Year of Publication 20.07.2006
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Year of Publication 20.07.2006
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