Mapping phospho-catalytic dependencies of therapy-resistant tumours reveals actionable vulnerabilities
Coppé, Jean-Philippe, Mori, Miki, Pan, Bo, Yau, Christina, Wolf, Denise M, Ruiz-Saenz, Ana, Brunen, Diede, Prahallad, Anirudh, Cornelissen-Steijger, Paulien, Kemper, Kristel, Posch, Christian, Wang, Changjun, Dreyer, Courtney A, Krijgsman, Oscar, Lee, Pei Rong Evelyn, Chen, Zhongzhong, Peeper, Daniel S, Moasser, Mark M, Bernards, René, van 't Veer, Laura J
Published in Nature cell biology (01.06.2019)
Published in Nature cell biology (01.06.2019)
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Journal Article
Heterogeneous drug penetrance of veliparib and carboplatin measured in triple negative breast tumors
Bartelink, Imke H, Prideaux, Brendan, Krings, Gregor, Wilmes, Lisa, Lee, Pei Rong Evelyn, Bo, Pan, Hann, Byron, Coppé, Jean-Philippe, Heditsian, Diane, Swigart-Brown, Lamorna, Jones, Ella F, Magnitsky, Sergey, Keizer, Ron J, de Vries, Niels, Rosing, Hilde, Pawlowska, Nela, Thomas, Scott, Dhawan, Mallika, Aggarwal, Rahul, Munster, Pamela N, Esserman, Laura J, Ruan, Weiming, Wu, Alan H B, Yee, Douglas, Dartois, Véronique, Savic, Radojka M, Wolf, Denise M, van 't Veer, Laura
Published in Breast cancer research : BCR (11.09.2017)
Published in Breast cancer research : BCR (11.09.2017)
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Journal Article
Does the combination of optimal substitutions at the C²-, N⁵- and N⁸-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A₃ adenosine receptors?
Cheong, Siew Lee, Dolzhenko, Anton V, Paoletta, Silvia, Lee, Evelyn Pei Rong, Kachler, Sonja, Federico, Stephanie, Klotz, Karl-Norbert, Dolzhenko, Anna V, Spalluto, Giampiero, Moro, Stefano, Pastorin, Giorgia
Published in Bioorganic & medicinal chemistry (15.10.2011)
Published in Bioorganic & medicinal chemistry (15.10.2011)
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Journal Article
Redefining breast cancer subtypes to guide treatment prioritization and maximize response: Predictive biomarkers across 10 cancer therapies
Wolf, Denise M., Yau, Christina, Wulfkuhle, Julia, Brown-Swigart, Lamorna, Gallagher, Rosa I., Lee, Pei Rong Evelyn, Zhu, Zelos, Magbanua, Mark J., Sayaman, Rosalyn, O’Grady, Nicholas, Basu, Amrita, Delson, Amy, Coppé, Jean Philippe, Lu, Ruixiao, Braun, Jerome, Asare, Smita M., Sit, Laura, Matthews, Jeffrey B., Perlmutter, Jane, Hylton, Nola, Liu, Minetta C., Pohlmann, Paula, Symmans, W. Fraser, Rugo, Hope S., Isaacs, Claudine, DeMichele, Angela M., Yee, Douglas, Berry, Donald A., Pusztai, Lajos, Petricoin, Emanuel F., Hirst, Gillian L., Esserman, Laura J., van 't Veer, Laura J.
Published in Cancer cell (13.06.2022)
Published in Cancer cell (13.06.2022)
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Journal Article
Tumor Drug Penetration Measurements Could Be the Neglected Piece of the Personalized Cancer Treatment Puzzle
Bartelink, Imke H., Jones, Ella F., Shahidi‐Latham, Sheerin K., Lee, Pei Rong Evelyn, Zheng, Yanan, Vicini, Paolo, ‘t Veer, Laura, Wolf, Denise, Iagaru, Andrei, Kroetz, Deanna L., Prideaux, Brendan, Cilliers, Cornelius, Thurber, Greg M., Wimana, Zena, Gebhart, Geraldine
Published in Clinical pharmacology and therapeutics (01.07.2019)
Published in Clinical pharmacology and therapeutics (01.07.2019)
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Journal Article
Abstract 2612: BluePrint Luminal subtype predicts non-response to HER2-targeted therapies in HR+/HER2+ I-SPY 2 breast cancer patients
Lee, Pei Rong Evelyn, Zhu, Zelos, Wolf, Denise, Yau, Christina, Audeh, William, Glas, Annuska, Brown-Swigart, Lamorna, Hirst, Gillian, DeMichele, Angela, Investigators, I-SPY 2 TRIAL, Esserman, Laura, Veer, Laura van 't
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 956: Systematic identification of the actionable kinase dependencies of chemotherapy-resistant triple-negative breast cancer
Coppe, Jean-Philippe F., Bo, Pan, Borden, Carolien van der, Koemans, Nina, Wang, Changjun, Wolf, Denise, Yau, Christina, Bakker, Sietske, Hartog, Marij, Mori, Miki, Ruiz-Saenz, Ana, Chen, Zhongzhong, Olow, Aleksandra, Lee, Pei Rong Evelyn, Veer, Laura van 't
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
An Atlas of the Human Kinome Reveals the Mutational Landscape Underlying Dysregulated Phosphorylation Cascades in Cancer
Olow, Aleksandra, Chen, Zhongzhong, Niedner, R Hannes, Wolf, Denise M, Yau, Christina, Pankov, Aleksandr, Lee, Evelyn Pei Rong, Brown-Swigart, Lamorna, van 't Veer, Laura J, Coppé, Jean-Philippe
Published in Cancer research (Chicago, Ill.) (01.04.2016)
Published in Cancer research (Chicago, Ill.) (01.04.2016)
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Abstract P2-05-09: Functional mapping of the oncogenic kinome activity of triple-negative breast cancer cells
Pan, Bo, Mori, Miki, Lee, Pei Rong Evelyn, Hartog, Marij, Sun, Qiang, van 't Veer, Laura, Coppe, Jean-Philippe
Published in Cancer research (Chicago, Ill.) (01.05.2015)
Published in Cancer research (Chicago, Ill.) (01.05.2015)
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Journal Article
Spatial distribution of veliparib measured by matrix-assisted laser desorption ionization mass spectrometry in triple-negative breast cancer tumors
Bartelink, Imke Heleen, Prideaux, Brendan, Hann, Byron, Krings, Gregor, Coppe, Jean-Philippe, Brown Swigart, Lamorna, Lee, Evelyn Pei Rong, Esserman, Laura, Yee, Douglas, Wolf, Denise, Savic, Rada M.
Published in Journal of clinical oncology (10.09.2014)
Published in Journal of clinical oncology (10.09.2014)
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Journal Article
Abstract P6-11-02: Spatial distribution of veliparib measured by matrix assisted laser desorption ionization mass spectrometry in triple negative breast cancer tumors
Bartelink, Imke H, Prideaux, Brendan, Hann, Byron, Krings, Gregor, Coppe, Jean-Phillippe, Swigart-Brown, Lamorna, Lee, Pei Rong Evelyn, Esserman, Laura, Yee, Douglas, Wolf, Denise, Savic, Rada M, van t Veer, Laura
Published in Cancer research (Chicago, Ill.) (01.05.2015)
Published in Cancer research (Chicago, Ill.) (01.05.2015)
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Journal Article
Does the combination of optimal substitutions at the C super(2-, N) super(5)- and N super(8-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A) sub(3) adenosine receptors?
Cheong, Siew Lee, Dolzhenko, Anton V, Paoletta, Silvia, Lee, Evelyn Pei Rong, Kachler, Sonja, Federico, Stephanie, Klotz, Karl-Norbert, Dolzhenko, Anna V, Spalluto, Giampiero, Moro, Stefano, Pastorin, Giorgia
Published in Bioorganic & medicinal chemistry (15.10.2011)
Published in Bioorganic & medicinal chemistry (15.10.2011)
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Journal Article
Does the combination of optimal substitutions at the C 2-, N 5- and N 8-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A 3 adenosine receptors?
Cheong, Siew Lee, Dolzhenko, Anton V., Paoletta, Silvia, Lee, Evelyn Pei Rong, Kachler, Sonja, Federico, Stephanie, Klotz, Karl-Norbert, Dolzhenko, Anna V., Spalluto, Giampiero, Moro, Stefano, Pastorin, Giorgia
Published in Bioorganic & medicinal chemistry (2011)
Published in Bioorganic & medicinal chemistry (2011)
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