Investigation of amino acid conjugates of (S)-1-[1-(4-aminobenzoyl)-2,3-dihydro-1H-indol-6-sulfonyl]-4-phenyl-imidazolidin-2-one (DW2282) as water soluble anticancer prodrugs
Lee, Ki-Cheul, Venkateswararao, Eeda, Sharma, Vinay Kumar, Jung, Sang-Hun
Published in European journal of medicinal chemistry (10.06.2014)
Published in European journal of medicinal chemistry (10.06.2014)
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Journal Article
Structural requirement(s) of N-phenylthioureas and benzaldehyde thiosemicarbazones as inhibitors of melanogenesis in melanoma B 16 cells
Thanigaimalai, P., Le Hoang, Tuan Anh, Lee, Ki-Cheul, Bang, Seong-Cheol, Sharma, Vinay K., Yun, Cheong-Yong, Roh, Eunmiri, Hwang, Bang-Yeon, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Journal Article
Identification of novel chromenone derivatives as interleukin-5 inhibitors
Venkateswararao, Eeda, Kim, Min-Seok, Sharma, Vinay K., Lee, Ki-Cheul, Subramanian, Santhosh, Roh, Eunmiri, Kim, Youngsoo, Jung, Sang-Hun
Published in European journal of medicinal chemistry (01.01.2013)
Published in European journal of medicinal chemistry (01.01.2013)
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Journal Article
Structural characteristics of thiosemicarbazones as inhibitors of melanogenesis
Lee, Ki-Cheul, Thanigaimalai, Pillaiyar, Sharma, Vinay K., Kim, Min-Seok, Roh, Eunmiri, Hwang, Bang-Yeon, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
Published in Bioorganic & medicinal chemistry letters (15.11.2010)
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Journal Article
Inhibitory effect of novel tetrahydropyrimidine-2(1 H)-thiones on melanogenesis
Thanigaimalai, P., Lee, Ki-Cheul, Bang, Seong-Cheol, Lee, Jee-Hyun, Yun, Cheong-Yong, Roh, Eunmiri, Hwang, Bang-Yeon, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry (01.02.2010)
Published in Bioorganic & medicinal chemistry (01.02.2010)
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Journal Article
Identification of Indoline-2-thione Analogs as Novel Potent Inhibitors of α-Melanocyte Stimulating Hormone Induced Melanogenesis
Thanigaimalai, Pillaiyar, Lee, Ki-Cheul, Sharma, Vinay Kumar, Sharma, Niti, Roh, Eunmiri, Kim, Youngsoo, Jung, Sang-Hun
Published in Chemical & pharmaceutical bulletin (2011)
Published in Chemical & pharmaceutical bulletin (2011)
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Journal Article
Novel Benzo[d]imidazole-2(3H)-thiones as Potent Inhibitors of the α-Melanocyte Stimulating Hormone Induced Melanogenesis in Melanoma B16 Cells
Lee, Jee-Hyun, Thanigaimalai, Pillaiyar, Lee, Ki-Cheul, Bang, Seong-Cheol, Kim, Min-Seok, Sharma, Vinay Kumar, Yun, Cheong-Yong, Roh, Eunmiri, Kim, Youngsoo, Jung, Sang-Hun
Published in Chemical & pharmaceutical bulletin (01.07.2010)
Published in Chemical & pharmaceutical bulletin (01.07.2010)
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Journal Article
A convenient preparation of a disaccharide motif and its role in the cytotoxicity of the triterpenoid saponin, α-hederin
Bang, Seong-Cheol, Seo, Hyun-Hee, Shin, Hye-Rim, Lee, Ki-Cheul, Hoang, Le Tuan Anh, Jung, Sang-Hun
Published in Archives of pharmacal research (01.05.2008)
Published in Archives of pharmacal research (01.05.2008)
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Journal Article
Design and synthesis of novel chromenone derivatives as interleukin-5 inhibitors
Venkateswararao, Eeda, Sharma, Vinay K., Lee, Ki-Cheul, Roh, Eunmiri, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry (01.05.2013)
Published in Bioorganic & medicinal chemistry (01.05.2013)
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Journal Article
Refinement of the pharmacophore of 3,4-dihydroquinazoline-2(1 H)-thiones for their anti-melanogenesis activity
Thanigaimalai, Pillaiyar, Sharma, Vinay K., Lee, Ki-Cheul, Yun, Cheong-Yong, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
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Journal Article
Structural requirement of phenylthiourea analogs for their inhibitory activity of melanogenesis and tyrosinase
Thanigaimalai, Pillaiyar, Lee, Ki-Cheul, Sharma, Vinay K., Joo, Cheonik, Cho, Won-Jea, Roh, Eunmiri, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
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Journal Article
Study on anti-proliferative effect of benzoxathiole derivatives through inactivation of NF-κB in human cancer cells
Venkateswararao, Eeda, Anh, Hoang Le Tuan, Sharma, Vinay K., Lee, Ki-Cheul, Sharma, Niti, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
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Journal Article
Evaluation of 3,4-dihydroquinazoline-2(1H)-thiones as inhibitors of α-MSH-induced melanin production in melanoma B16 cells
Thanigaimalai, P., Lee, Ki-Cheul, Bang, Seong-Cheol, Lee, Jee-Hyun, Yun, Cheong-Yong, Roh, Eunmiri, Hwang, Bang-Yeon, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry (15.02.2010)
Published in Bioorganic & medicinal chemistry (15.02.2010)
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Journal Article
Structure–activity relationship of naphthaldehydethiosemicarbazones in melanogenesis inhibition
Thanigaimalai, Pillaiyar, Rao, Eeda Venkateswara, Lee, Ki-Cheul, Sharma, Vinay K., Roh, Eunmiri, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Journal Article
A SAR study on a series of synthetic lipophilic chalcones as Inhibitor of transcription factor NF-κB
Venkateswararao, Eeda, Sharma, Vinay K., Lee, Ki-Cheul, Sharma, Niti, Park, Sun-Hong, Kim, Youngsoo, Jung, Sang-Hun
Published in European journal of medicinal chemistry (01.08.2012)
Published in European journal of medicinal chemistry (01.08.2012)
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Journal Article
Structural requirements of ( E)-6-benzylidene-4a-methyl-4,4a,5,6,7,8-hexahydronaphthalen-2(3 H)-one derivatives as novel melanogenesis inhibitors
Thanigaimalai, Pillaiyar, Lee, Ki-Cheul, Sharma, Vinay K., Rao, Eeda Vekateswara, Roh, Eunmiri, Kim, Youngsoo, Jung, Sang-Hun
Published in Bioorganic & medicinal chemistry letters (01.04.2011)
Published in Bioorganic & medicinal chemistry letters (01.04.2011)
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Journal Article