Structure-Activity Studies of Cysteine-Rich -Conotoxins that Inhibit High-Voltage-Activated Calcium Channels via GABAB Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B., Berecki, Geza, Daniel, James T., Lee, Han Siean, Jackson, Kathryn A. V., Tae, Han-Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M., Craik, David J., Adams, David J., Clark, Richard J.
Published in Angewandte Chemie International Edition (04.04.2016)
Published in Angewandte Chemie International Edition (04.04.2016)
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Journal Article
Identification, Characterization, and Three-Dimensional Structure of the Novel Circular Bacteriocin, Enterocin NKR-5-3B, from Enterococcus faecium
Himeno, Kohei, Rosengren, K. Johan, Inoue, Tomoko, Perez, Rodney H, Colgrave, Michelle L, Lee, Han Siean, Chan, Lai Y, Henriques, Sónia Troeira, Fujita, Koji, Ishibashi, Naoki, Zendo, Takeshi, Wilaipun, Pongtep, Nakayama, Jiro, Leelawatcharamas, Vichien, Jikuya, Hiroyuki, Craik, David J, Sonomoto, Kenji
Published in Biochemistry (Easton) (11.08.2015)
Published in Biochemistry (Easton) (11.08.2015)
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Journal Article
Posttranslational modifications of α-conotoxins: sulfotyrosine and C-terminal amidation stabilise structures and increase acetylcholine receptor binding
Ho, Thao N. T, Lee, Han Siean, Swaminathan, Shilpa, Goodwin, Lewis, Rai, Nishant, Ushay, Brianna, Lewis, Richard J, Rosengren, K. Johan, Conibear, Anne C
Published in MedChemComm (23.09.2021)
Published in MedChemComm (23.09.2021)
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Journal Article
Development of Relaxin-3 Agonists and Antagonists Based on Grafted Disulfide-Stabilized Scaffolds
Lee, Han Siean, Postan, Michael, Song, Angela, Clark, Richard J, Bathgate, Ross A D, Haugaard-Kedström, Linda M, Rosengren, K Johan
Published in Frontiers in chemistry (18.02.2020)
Published in Frontiers in chemistry (18.02.2020)
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Journal Article
Exploring the Use of Helicogenic Amino Acids for Optimising Single Chain Relaxin-3 Peptide Agonists
Lee, Han Siean, Wang, Shu Hui, Daniel, James T., Hossain, Mohammed Akhter, Clark, Richard J., Bathgate, Ross A. D., Rosengren, K. Johan
Published in Biomedicines (14.10.2020)
Published in Biomedicines (14.10.2020)
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Journal Article
Development of Potent and Selective Agonists for Complement C5a Receptor 1 with In Vivo Activity
Gorman, Declan M, Li, Xaria X, Lee, John D, Fung, Jenny N, Cui, Cedric S, Lee, Han Siean, Rolfe, Barbara E, Woodruff, Trent M, Clark, Richard J
Published in Journal of medicinal chemistry (25.11.2021)
Published in Journal of medicinal chemistry (25.11.2021)
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Journal Article
Structure-Activity Studies of Cysteine-Rich α-Conotoxins that Inhibit High-Voltage-Activated Calcium Channels via GABAB Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B., Berecki, Géza, Daniel, James T., Lee, Han Siean, Jackson, Kathryn A. V., Tae, Han-Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M., Craik, David J., Adams, David J., Clark, Richard J.
Published in Angewandte Chemie (International ed.) (04.04.2016)
Published in Angewandte Chemie (International ed.) (04.04.2016)
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Journal Article
Binding conformation and determinants of a single-chain peptide antagonist at the relaxin-3 receptor RXFP3
Haugaard-Kedström, Linda M., Lee, Han Siean, Jones, Maryon V., Song, Angela, Rathod, Vishaal, Hossain, Mohammed Akhter, Bathgate, Ross A.D., Rosengren, K. Johan
Published in The Journal of biological chemistry (12.10.2018)
Published in The Journal of biological chemistry (12.10.2018)
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Journal Article
Peptide mimic for influenza vaccination using nonnatural combinatorial chemistry
Miles, John J, Tan, Mai Ping, Dolton, Garry, Edwards, Emily Sj, Galloway, Sarah Ae, Laugel, Bruno, Clement, Mathew, Makinde, Julia, Ladell, Kristin, Matthews, Katherine K, Watkins, Thomas S, Tungatt, Katie, Wong, Yide, Lee, Han Siean, Clark, Richard J, Pentier, Johanne M, Attaf, Meriem, Lissina, Anya, Ager, Ann, Gallimore, Awen, Rizkallah, Pierre J, Gras, Stephanie, Rossjohn, Jamie, Burrows, Scott R, Cole, David K, Price, David A, Sewell, Andrew K
Published in The Journal of clinical investigation (01.04.2018)
Published in The Journal of clinical investigation (01.04.2018)
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Journal Article
Structure–Activity Studies of Cysteine‐Rich α‐Conotoxins that Inhibit High‐Voltage‐Activated Calcium Channels via GABA B Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B., Berecki, Géza, Daniel, James T., Lee, Han Siean, Jackson, Kathryn A. V., Tae, Han‐Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M., Craik, David J., Adams, David J., Clark, Richard J.
Published in Angewandte Chemie International Edition (04.04.2016)
Published in Angewandte Chemie International Edition (04.04.2016)
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Journal Article
Structure-Activity Studies of Cysteine-Rich α-Conotoxins that Inhibit High-Voltage-Activated Calcium Channels via GABA(B) Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B, Berecki, Géza, Daniel, James T, Lee, Han Siean, Jackson, Kathryn A V, Tae, Han-Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M, Craik, David J, Adams, David J, Clark, Richard J
Published in Angewandte Chemie International Edition (04.04.2016)
Published in Angewandte Chemie International Edition (04.04.2016)
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Journal Article
Structure–Activity Studies of Cysteine‐Rich α‐Conotoxins that Inhibit High‐Voltage‐Activated Calcium Channels via GABA B Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B., Berecki, Géza, Daniel, James T., Lee, Han Siean, Jackson, Kathryn A. V., Tae, Han‐Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M., Craik, David J., Adams, David J., Clark, Richard J.
Published in Angewandte Chemie (04.04.2016)
Published in Angewandte Chemie (04.04.2016)
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Journal Article
Structure-Activity Studies of Cysteine-Rich [alpha]-Conotoxins that Inhibit High-Voltage-Activated Calcium Channels via GABAB Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B, Berecki, Géza, Daniel, James T, Lee, Han Siean, Jackson, Kathryn A V, Tae, Han-Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M, Craik, David J, Adams, David J, Clark, Richard J
Published in Angewandte Chemie (04.04.2016)
Published in Angewandte Chemie (04.04.2016)
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Journal Article
Structure-Activity Studies of Cysteine-Rich alpha -Conotoxins that Inhibit High-Voltage-Activated Calcium Channels via GABA sub(B) Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B, Berecki, Geza, Daniel, James T, Lee, Han Siean, Jackson, Kathryn AV, Tae, Han-Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M, Craik, David J, Adams, David J, Clark, Richard J
Published in Angewandte Chemie (01.04.2016)
Published in Angewandte Chemie (01.04.2016)
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Journal Article
Structure-Activity Studies of Cysteine-Rich α-Conotoxins that Inhibit High-Voltage-Activated Calcium Channels via GABAB Receptor Activation Reveal a Minimal Functional Motif
Carstens, Bodil B., Berecki, Géza, Daniel, James T., Lee, Han Siean, Jackson, Kathryn A. V., Tae, Han-Shen, Sadeghi, Mahsa, Castro, Joel, O'Donnell, Tracy, Deiteren, Annemie, Brierley, Stuart M., Craik, David J., Adams, David J., Clark, Richard J.
Published in Angewandte Chemie (04.04.2016)
Published in Angewandte Chemie (04.04.2016)
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Journal Article