CRTH2 Antagonist MK-7246: A Synthetic Evolution from Discovery through Development
Molinaro, Carmela, Bulger, Paul G, Lee, Ernest E, Kosjek, Birgit, Lau, Stephen, Gauvreau, Danny, Howard, Melissa E, Wallace, Debra J, O’Shea, Paul D
Published in Journal of organic chemistry (02.03.2012)
Published in Journal of organic chemistry (02.03.2012)
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Regioselective rhodium-catalyzed intermolecular [2+2+2] cycloaddition of alkynes and isocyanates to form pyridones
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Conference Proceeding
Enantioselective Rhodium-Catalyzed [2 + 2 + 2] Cycloadditions of Terminal Alkynes and Alkenyl Isocyanates: Mechanistic Insights Lead to a Unified Model that Rationalizes Product Selectivity
Dalton, Derek M, Oberg, Kevin M, Yu, Robert T, Lee, Ernest E, Perreault, Stéphane, Oinen, Mark Emil, Pease, Melissa L, Malik, Guillaume, Rovis, Tomislav
Published in Journal of the American Chemical Society (04.11.2009)
Published in Journal of the American Chemical Society (04.11.2009)
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Diastereoselective synthesis of fluorinated piperidine quinazoline spirocycles as iNOS selective inhibitors
Walpole, Chris, Liu, Ziping, Lee, Ernest E., Yang, Hua, Zhou, Fei, Mackintosh, Nicole, Sjogren, Magnus, Taylor, David, Shen, Jinyu, Batey, Robert A.
Published in Tetrahedron letters (13.06.2012)
Published in Tetrahedron letters (13.06.2012)
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Effect of acid catalysis on the direct electrophilic fluorination of ketones, ketals, and enamides using Selectfluor
Liu, Jack, Chan, Johann, Bryant, Craig M., Duspara, Petar A., Lee, Ernest E., Powell, David, Yang, Hua, Liu, Ziping, Walpole, Chris, Roberts, Edward, Batey, Robert A.
Published in Tetrahedron letters (13.06.2012)
Published in Tetrahedron letters (13.06.2012)
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Journal Article
Discovery of MK-7246, a selective CRTH2 antagonist for the treatment of respiratory diseases
Gallant, Michel, Beaulieu, Christian, Berthelette, Carl, Colucci, John, Crackower, Michael A., Dalton, Chad, Denis, Danielle, Ducharme, Yves, Friesen, Richard W., Guay, Daniel, Gervais, François G., Hamel, Martine, Houle, Robert, Krawczyk, Connie M., Kosjek, Birgit, Lau, Stephen, Leblanc, Yves, Lee, Ernest E., Levesque, Jean-François, Mellon, Christophe, Molinaro, Carmela, Mullet, Wayne, O’Neill, Gary P., O’Shea, Paul, Sawyer, Nicole, Sillaots, Susan, Simard, Daniel, Slipetz, Deborah, Stocco, Rino, Sørensen, Dan, Truong, Vouy Linh, Wong, Elizabeth, Wu, Jin, Zaghdane, Helmi, Wang, Zhaoyin
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Effect of ethnicity on the risk of developing nonmelanoma skin cancer following long-term PUVA therapy
Murase, Jenny E., Lee, Ernest E., Koo, John
Published in International journal of dermatology (01.12.2005)
Published in International journal of dermatology (01.12.2005)
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Synthesis of oligosaccharide fragments of the glycosylinositolphospholipid of Trypanosoma cruzi: a new selenoglycoside glycosyl donor for the preparation of 4-thiogalactofuranosyl analogues
Randell, Karla D, Johnston, Blair D, Lee, Ernest E, Pinto, B.Mario
Published in Tetrahedron: asymmetry (28.01.2000)
Published in Tetrahedron: asymmetry (28.01.2000)
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Effect of acid catalysis on the direct electrophilic fluorination of ketones, ketals, and enamides using Selectfluorac
Liu, Jack, Chan, Johann, Bryant, Craig M, Duspara, Petar A, Lee, Ernest E, Powell, David, Yang, Hua, Liu, Ziping, Walpole, Chris, Roberts, Edward, Batey, Robert A
Published in Tetrahedron letters (13.06.2012)
Published in Tetrahedron letters (13.06.2012)
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Journal Article
Discovery of Mix-7246, a selective CRTH2 antagonist for the treatment of respiratory diseases
GALLANT, Michel, BEAULIEU, Christian, GERVAIS, François G, HAMEL, Martine, HOULE, Robert, KRAWCZYK, Connie M, KOSJEK, Birgit, LAU, Stephen, LEBLANC, Yves, LEE, Ernest E, LEVESQUE, Jean-François, MELLON, Christophe, BERTHELETTE, Carl, MOLINARO, Carmela, MULLET, Wayne, O'NEILL, Gary P, O'SHEA, Paul, SAWYER, Nicole, SILLAOTS, Susan, SIMARD, Daniel, SLIPETZ, Deborah, STOCCO, Rino, SØRENSEN, Dan, COLUCCI, John, VOUY LINH TRUONG, WONG, Elizabeth, JIN WU, ZAGHDANE, Helmi, ZHAOYIN WANG, CRACKOWER, Michael A, DALTON, Chad, DENIS, Danielle, DUCHARME, Yves, FRIESEN, Richard W, GUAY, Daniel
Published in Bioorganic & medicinal chemistry letters (2011)
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Published in Bioorganic & medicinal chemistry letters (2011)
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