Advanced glycation end-products induce apoptosis of bovine retinal pericytes in culture: involvement of diacylglycerol/ceramide production and oxidative stress induction
Denis, Ulriche, Lecomte, Marc, Paget, Clarisse, Ruggiero, Daniel, Wiernsperger, Nicolas, Lagarde, Michel
Published in Free radical biology & medicine (15.07.2002)
Published in Free radical biology & medicine (15.07.2002)
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Involvement of Arginine 120, Glutamate 524, and Tyrosine 355 in the Binding of Arachidonate and 2-Phenylpropionic Acid Inhibitors to the Cyclooxygenase Active Site of Ovine Prostaglandin Endoperoxide H Synthase-1
Bhattacharyya, D K, Lecomte, M, Rieke, C J, Garavito, M, Smith, W L
Published in The Journal of biological chemistry (26.01.1996)
Published in The Journal of biological chemistry (26.01.1996)
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In vitro and in vivo alterations of enzymatic glycosylation in diabetes
Rellier, Nadège, Ruggiero-Lopez, Daniel, Lecomte, Marc, Lagarde, Michel, Wiernsperger, Nicolas
Published in Life sciences (1973) (19.03.1999)
Published in Life sciences (1973) (19.03.1999)
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Improved Prediction of in Vivo Supersaturation and Precipitation of Poorly Soluble Weakly Basic Drugs Using a Biorelevant Bicarbonate Buffer in a Gastrointestinal Transfer Model
Jede, Christian, Wagner, Christian, Kubas, Holger, Weigandt, Markus, Weber, Christian, Lecomte, Marc, Badolo, Lassina, Koziolek, Mirko, Weitschies, Werner
Published in Molecular pharmaceutics (03.09.2019)
Published in Molecular pharmaceutics (03.09.2019)
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Identification of solubility-limited absorption of oral anticancer drugs using PBPK modeling based on rat PK and its relevance to human
Fink, Christina, Lecomte, Marc, Badolo, Lassina, Wagner, Knut, Mäder, Karsten, Peters, Sheila-Annie
Published in European journal of pharmaceutical sciences (01.09.2020)
Published in European journal of pharmaceutical sciences (01.09.2020)
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Dual A2A/A2B Adenosine Receptor Antagonist M1069 Counteracts Immunosuppressive Mechanisms of Adenosine and Reduces Tumor Growth In Vivo
Schiemann, Kai, Belousova, Natalya, Matevossian, Armine, Nallaparaju, Kalyan C., Kradjian, Giorgio, Pandya, Meghana, Chen, Zhouxiang, Aral, Esengul, Krauel, Eva-Maria, Petrova, Elissaveta, Boesler, Carsten, Kitzing, Thomas, Lecomte, Marc, Wagner, Christian, Blayo, Anne Laure, Schann, Stephan, Huck, Bayard, Moisan, Jacques, Zaynagetdinov, Rinat
Published in Molecular cancer therapeutics (03.09.2024)
Published in Molecular cancer therapeutics (03.09.2024)
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Discovery of Cycloalkyl[c]thiophenes as Novel Scaffolds for Hypoxia-Inducible Factor-2α Inhibitors
Buchstaller, Hans-Peter, Sala-Hojman, Ada, Leiendecker, Matthias, Albers, Joachim, Anlauf, Uwe, Berges, Nina, Dong, Liming, Fuchß, Thomas, Germann, Martina, Knehans, Tim, Krier, Mireille, Lecomte, Marc, Müller, Daniel, Müller, Sandra R., Leuthner, Birgitta, Lindemann, Ralph, Musil, Djordje, Nowak, Mateusz, Reither, Vivian, Rettig, Corinna, Schindler, Christina E. M., Pakulska, Urszula, Spuck, Dieter, Wegener, Ansgar, Zarębski, Adrian
Published in Journal of medicinal chemistry (13.07.2023)
Published in Journal of medicinal chemistry (13.07.2023)
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Dual A2A/ A2B adenosine receptor antagonist M1069 counteracts immuno-suppressive mechanisms of adenosine and reduces tumor growth in vivo
Schiemann, Kai, Belousova, Natalya, Matevossian, Armine, Nallaparaju, Kalyan C, Kradjian, Giorgio, Pandya, Meghana, Chen, Zhouxiang, Aral, Esengul, Krauel, Eva-Maria, Petrova, Elissaveta, Boesler, Carsten, Kitzing, Thomas, Lecomte, Marc, Wagner, Christian, Blayo, Anne Laure, Schann, Stephan, Huck, Bayard, Moisan, Jacques, Zaynagetdinov, Rinat
Published in Molecular cancer therapeutics (20.08.2024)
Published in Molecular cancer therapeutics (20.08.2024)
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Abstract 3499: M1069 as dual A2A/A2B adenosine receptor antagonist counteracts immune-suppressive mechanisms of adenosine and reduces tumor growth in vivo
Zaynagetdinov, Rinat, Schiemann, Kai, Nallaparaju, Kalyan, Belousova, Natalya, Matevossian, Armine, Chen, Zhouxiang, Kradjian, Giorgio, Pandya, Meghana, Dawra, Nemisha, Krauel, Eva-Maria, Petrova, Elissaveta, Poeschke, Oliver, Fischer, David, Lecomte, Marc, Blaukat, Andree, Huck, Bayard, Moisan, Jacques
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Abstract 4516: Evaluation of p70S6K/Akt inhibitor MSC2363318A in patient derived xenograft (PDX) models of breast cancer
Huck, Bayard R., Tian, H, Syed, Sakeena, Lin, Jing, Ma, Jianguo, Clark, Anderson, Kaleta, Remiguisz, Machl, Andreas, Wilker, Erik, Lecomte, Marc
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Reaction of metformin with dicarbonyl compounds. possible implication in the inhibition of advanced glycation end product formation
Ruggiero-Lopez, Daniel, Lecomte, Marc, Moinet, Gérard, Patereau, Gérard, Lagarde, Michel, Wiernsperger, Nicolas
Published in Biochemical pharmacology (01.12.1999)
Published in Biochemical pharmacology (01.12.1999)
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Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11β-hydroxysteroid dehydrogenase type I
Valeur, Eric, Christmann-Franck, Serge, Lepifre, Franck, Carniato, Denis, Cravo, Daniel, Charon, Christine, Bozec, Sophie, Musil, Djordje, Hillertz, Per, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Schultz, Melanie, Roche, Didier
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
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Journal Article
Discovery and structure-guided drug design of inhibitors of 11β-hydroxysteroid-dehydrogenase type I based on a spiro-carboxamide scaffold
Lepifre, Franck, Christmann-Franck, Serge, Roche, Didier, Leriche, Caroline, Carniato, Denis, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
Published in Bioorganic & medicinal chemistry letters (01.07.2009)
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Journal Article
Discovery and structure–activity relationships of pentanedioic acid diamides as potent inhibitors of 11β-hydroxysteroid dehydrogenase type I
Roche, Didier, Carniato, Denis, Leriche, Caroline, Lepifre, Franck, Christmann-Franck, Serge, Graedler, Ulrich, Charon, Christine, Bozec, Sophie, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Valeur, Eric
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Abstract A162: Identification of brain penetrant p70S6K/Akt inhibitor MSC2363318A
Huck, Bayard R., Machl, Andreas, Wilker, Erik, Tian, Hui, Syed, Sakeena, Lin, Jing, Ma, Jianguo, Clark, Anderson, Waterhouse, Roseann, Kaleta, Remiguisz, Micu, Alina, Soughley, Lynne, Li, Long, Groll, Karin, Kroesser, Sonja, Beier, Frank, Hering, Ursula, Lecomte, Marc, Wichert, Katrin, D'Antonio, Mauro, Di Eugenio, Paolo
Published in Molecular cancer therapeutics (01.11.2013)
Published in Molecular cancer therapeutics (01.11.2013)
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Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11[beta]-hydroxysteroid dehydrogenase type I
Valeur, Eric, Christmann-Franck, Serge, Lepifre, Franck, Carniato, Denis, Cravo, Daniel, Charon, Christine, Bozec, Sophie, Musil, Djordje, Hillertz, Per, Doare, Liliane, Schmidlin, Fabien, Lecomte, Marc, Schultz, Melanie, Roche, Didier
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
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Acetylation of human prostaglandin endoperoxide synthase-2 (cyclooxygenase-2) by aspirin
LECOMTE, M, LANEUVILLE, O, CHUAN JI, DEWITT, D. L, SMITH, W. L
Published in The Journal of biological chemistry (06.05.1994)
Published in The Journal of biological chemistry (06.05.1994)
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