Targeted Degradation of Protein Kinase A via a Stapled Peptide PROTAC
Whittaker, Matthew K., Bendzunas, George N., Shirani, Mahsa, LeClair, Timothy J., Shebl, Bassem, Dill, Taylor C., Coffino, Philip, Simon, Sanford M., Kennedy, Eileen J.
Published in ACS chemical biology (20.09.2024)
Published in ACS chemical biology (20.09.2024)
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Allosteric Inhibition of Parkinson’s-Linked LRRK2 by Constrained Peptides
Helton, Leah G, Soliman, Ahmed, von Zweydorf, Felix, Kentros, Michalis, Manschwetus, Jascha T, Hall, Scotty, Gilsbach, Bernd, Ho, Franz Y, Athanasopoulos, Panagiotis S, Singh, Ranjan K, LeClair, Timothy J, Versées, Wim, Raimondi, Francesco, Herberg, Friedrich W, Gloeckner, Christian Johannes, Rideout, Hardy, Kortholt, Arjan, Kennedy, Eileen J
Published in ACS chemical biology (19.11.2021)
Published in ACS chemical biology (19.11.2021)
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Doubly Constrained C‑terminal of Roc (COR) Domain-Derived Peptides Inhibit Leucine-Rich Repeat Kinase 2 (LRRK2) Dimerization
Pathak, Pragya, Alexander, Krista K., Helton, Leah G., Kentros, Michalis, LeClair, Timothy J., Zhang, Xiaojuan, Ho, Franz Y., Moore, Timothy T., Hall, Scotty, Guaitoli, Giambattista, Gloeckner, Christian Johannes, Kortholt, Arjan, Rideout, Hardy, Kennedy, Eileen J.
Published in ACS chemical neuroscience (07.06.2023)
Published in ACS chemical neuroscience (07.06.2023)
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In Silico Optimized Stapled Peptides Targeting WASF3 in Breast Cancer
Limaye, Ameya J, Bendzunas, George N, Whittaker, Matthew K, LeClair, Timothy J, Helton, Leah G, Kennedy, Eileen J
Published in ACS medicinal chemistry letters (14.04.2022)
Published in ACS medicinal chemistry letters (14.04.2022)
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