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An Amino-terminal Variant of the Central Cannabinoid Receptor Resulting from Alternative Splicing
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The Cannabinoid CB1 Receptor Antagonist Rimonabant (SR141716) Inhibits Cell Proliferation and Increases Markers of Adipocyte Maturation in Cultured Mouse 3T3 F442A Preadipocytes
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Structural Features of the Central Cannabinoid CB1 Receptor Involved in the Binding of the Specific CB1 Antagonist SR 141716A
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Stimulation of the β3-Adrenoceptor as a Novel Treatment Strategy for Anxiety and Depressive Disorders
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Published in Neuropsychopharmacology (New York, N.Y.) (25.04.2007)
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SR141716A, a potent and selective antagonist of the brain cannabinoid receptor
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Published in FEBS letters (22.08.1994)
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Role of Peripheral Benzodiazepine Receptors in Mitochondrial, Cellular, and Cardiac Damage Induced by Oxidative Stress and Ischemia-Reperfusion
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Modulation and Functional Involvement of CB2 Peripheral Cannabinoid Receptors During B-Cell Differentiation
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In vitro and in vivo biological activities of SR140333, a novel potent non-peptide tachykinin NK1 receptor antagonist
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Published in European journal of pharmacology (21.12.1993)
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Primary structure and functional expression of mouse pituitary and human brain corticotrophin releasing factor receptors
Vita, Natalio, Laurent, Patrick, Lefort, Sylvie, Chalon, Pascale, Lelias, Jean-Michel, Kaghad, Mourad, Le Fur, Gérard, Caput, Daniel, Ferrara, Pascual
Published in FEBS letters (29.11.1993)
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Neurotensin is an antagonist of the human neurotensin NT2 receptor expressed in Chinese hamster ovary cells
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Published in European journal of pharmacology (06.11.1998)
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Biochemical and Pharmacological Profile of a Potent and Selective Nonpeptide Antagonist of the Neurotensin Receptor
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Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1993)
Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1993)
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Dual intracellular signaling pathways mediated by the human cannabinoid CB1 receptor
CALANDRA, B, PORTIER, M, KERNEIS, A, DELPECH, M, CARILLON, C, LE FUR, G, FERRARA, P, SHIRE, D
Published in European journal of pharmacology (25.06.1999)
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Characterization of NPY receptors controlling lipolysis and leptin secretion in human adipocytes
Serradeil-Le Gal, Claudine, Lafontan, Max, Raufaste, Danielle, Marchand, Jean, Pouzet, Brigitte, Casellas, Pierre, Pascal, Marc, Maffrand, Jean-Pierre, Le Fur, Gérard
Published in FEBS letters (16.06.2000)
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Arousal-enhancing properties of the CB1 cannabinoid receptor antagonist SR 141716A in rats as assessed by electroencephalographic spectral and sleep-waking cycle analysis
Santucci, Vincent, Storme, Jean-jacques, Soubrié, Philippe, Le Fur, Gérard
Published in Life sciences (1973) (1996)
Published in Life sciences (1973) (1996)
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Single and multiple doses of rimonabant antagonize acute effects of smoked cannabis in male cannabis users
HUESTIS, Marilyn A, BOYD, Susan J, HEISHMAN, Stephen J, PRESTON, Kenzie L, BONNET, Denis, LE FUR, Gerard, GORELICK, David A
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Published in Psychopharmacologia (01.11.2007)
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