Stability of G,A triple helices
Debin, A., Laboulais, C., Ouali, M., Malvy, C., Le Bret, M., Svinarchuk, F.
Published in Nucleic acids research (01.07.1999)
Published in Nucleic acids research (01.07.1999)
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A database of 32 DNA triplets to study triple helices by molecular mechanics and dynamics
Piriou, J.M., Ketterlé, Ch, Gabarro-Arpa, J., Cognet, J.A.H., Le Bret, M.
Published in Biophysical chemistry (01.06.1994)
Published in Biophysical chemistry (01.06.1994)
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DNA Polyintercalating Drugs: DNA Binding of Diacridine Derivatives
Le Pecq, Jean-Bernard, Le Bret, Marc, Barbet, Jacques, Roques, Bernard
Published in Proceedings of the National Academy of Sciences - PNAS (01.08.1975)
Published in Proceedings of the National Academy of Sciences - PNAS (01.08.1975)
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Solution Structure of an Oncogenic DNA Duplex, the K- ras Gene and the Sequence Containing a Central C·A or A·G Mismatch as a Function of pH: Nuclear Magnetic Resonance and Molecular Dynamics Studies
Boulard, Y., Cognet, J.A.H., Gabarro-Arpa, J., Le Bret, M, Carbonnaux, C., Fazakerley, G.V.
Published in Journal of molecular biology (01.01.1995)
Published in Journal of molecular biology (01.01.1995)
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The pH dependent configurations of the C.A mispair in DNA
Boulard, Y., Cognet, J.A.H., Gabarro-Arpa, J., Le Bret, M., Sowers, L.C., Fazakerley, G.V.
Published in Nucleic acids research (25.04.1992)
Published in Nucleic acids research (25.04.1992)
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Linker-modified quinoline derivatives targeting HIV-1 integrase: synthesis and biological activity
Bénard, Christophe, Zouhiri, Fatima, Normand-Bayle, Marie, Danet, Michèle, Desmaële, Didier, Leh, Hervé, Mouscadet, Jean-François, Mbemba, Gladys, Thomas, Claire-Marie, Bonnenfant, Sabine, Le Bret, Marc, d'Angelo, Jean
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
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Use of the Kohonen Neural Network for Rapid Screening of Ex Vivo Anti-HIV Activity of Styrylquinolines
Polanski, Jaroslaw, Zouhiri, Fatima, Jeanson, Laurence, Desmaële, Didier, d'Angelo, Jean, Mouscadet, Jean-François, Gieleciak, Rafal, Gasteiger, Johann, Le Bret, Marc
Published in Journal of medicinal chemistry (10.10.2002)
Published in Journal of medicinal chemistry (10.10.2002)
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Mechanism of HIV-1 Integrase Inhibition by Styrylquinoline Derivatives in Vitro
Deprez, Eric, Barbe, Sophie, Kolaski, Macieij, Leh, Hervé, Zouhiri, Fatima, Auclair, Christian, Brochon, Jean-Claude, Le Bret, Marc, Mouscadet, Jean-François
Published in Molecular pharmacology (01.01.2004)
Published in Molecular pharmacology (01.01.2004)
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Structure−Activity Relationships and Binding Mode of Styrylquinolines as Potent Inhibitors of HIV-1 Integrase and Replication of HIV-1 in Cell Culture
Zouhiri, Fatima, Mouscadet, Jean-François, Mekouar, Khalid, Desmaële, Didier, Savouré, Delphine, Leh, Hervé, Subra, Frédéric, Le Bret, Marc, Auclair, Christian, d'Angelo, Jean
Published in Journal of medicinal chemistry (20.04.2000)
Published in Journal of medicinal chemistry (20.04.2000)
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Molecular Modeling of Wild-Type and D816V c-Kit Inhibition Based on ATP-Competitive Binding of Ellipticine Derivatives to Tyrosine Kinases
Vendôme, Jérémie, Letard, Sébastien, Martin, Frédéric, Svinarchuk, Fedor, Dubreuil, Patrice, Auclair, Christian, Le Bret, Marc
Published in Journal of medicinal chemistry (06.10.2005)
Published in Journal of medicinal chemistry (06.10.2005)
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Probing of HIV-1 Integrase/DNA Interactions Using Novel Analogs of Viral DNA
Agapkina, Julia, Smolov, Maksim, Barbe, Sophie, Zubin, Evgenii, Zatsepin, Timofei, Deprez, Eric, Le Bret, Marc, Mouscadet, Jean-François, Gottikh, Marina
Published in The Journal of biological chemistry (28.04.2006)
Published in The Journal of biological chemistry (28.04.2006)
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Functional analysis of novel Sonic Hedgehog gene mutations identified in basal cell carcinomas from xeroderma pigmentosum patients
COUVE-PRIVAT, Sophie, LE BRET, Marc, TRAIFFORT, Elisabeth, QUEILLE, Sophie, COULOMBE, Josée, BOUADJAR, Bakar, AVRIL, Marie Francoise, RUAT, Martial, SARASIN, Alain, DAYA-GROSJEAN, Leela
Published in Cancer research (Chicago, Ill.) (15.05.2004)
Published in Cancer research (Chicago, Ill.) (15.05.2004)
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Modeling of the Inhibition of Retroviral Integrases by Styrylquinoline Derivatives
Ouali, Mohammed, Laboulais, Cyril, Leh, Hervé, Gill, David, Desmaële, Didier, Mekouar, Khalid, Zouhiri, Fatima, d'Angelo, Jean, Auclair, Christian, Mouscadet, Jean-François, Le Bret, Marc
Published in Journal of medicinal chemistry (18.05.2000)
Published in Journal of medicinal chemistry (18.05.2000)
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Intermolecular interactions in the crystal structures of potential HIV-1 integrase inhibitors
Majerz-Maniecka, Katarzyna, Musiol, Robert, Nitek, Wojciech, Oleksyn, Barbara J., Mouscadet, Jean-Francois, Bret, Marc Le, Polanski, Jaroslaw
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Abasic frameshift in DNA. Solution conformation determined by proton NMR and molecular mechanics calculations
Cuniasse, P, Sowers, L. C, Eritja, R, Kaplan, B, Goodman, M. F, Cognet, J. A. H, Le Bret, M, Guschlbauer, W, Fazakerley, G. V
Published in Biochemistry (Easton) (07.03.1989)
Published in Biochemistry (Easton) (07.03.1989)
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HIV-1 replication inhibitors of the styrylquinoline class: incorporation of a masked diketo acid pharmacophore
Zouhiri, Fatima, Desmaële, Didier, d'Angelo, Jean, Ourevitch, Michèle, Mouscadet, Jean-François, Leh, Hervé, Le Bret, Marc
Published in Tetrahedron letters (12.11.2001)
Published in Tetrahedron letters (12.11.2001)
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Comparative molecular surface analysis (CoMSA) for virtual combinatorial library screening of styrylquinoline HIV-1 blocking agents
Niedbala, Halina, Polanski, Jaroslaw, Gieleciak, Rafal, Musiol, Robert, Tabak, Dominik, Podeszwa, Barbara, Bak, Andrzej, Palka, Anna, Mouscadet, Jean-Francois, Gasteiger, Johann, Le Bret, Marc
Published in Combinatorial chemistry & high throughput screening (01.12.2006)
Published in Combinatorial chemistry & high throughput screening (01.12.2006)
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