Bivalent Ligands That Target μ Opioid (MOP) and Cannabinoid1 (CB1) Receptors Are Potent Analgesics Devoid of Tolerance
Le Naour, Morgan, Akgün, Eyup, Yekkirala, Ajay, Lunzer, Mary M, Powers, Mike D, Kalyuzhny, Alexander E, Portoghese, Philip S
Published in Journal of medicinal chemistry (11.07.2013)
Published in Journal of medicinal chemistry (11.07.2013)
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Journal Article
Putative Kappa Opioid Heteromers As Targets for Developing Analgesics Free of Adverse Effects
Le Naour, Morgan, Lunzer, Mary M, Powers, Michael D, Kalyuzhny, Alexander E, Benneyworth, Michael A, Thomas, Mark J, Portoghese, Philip S
Published in Journal of medicinal chemistry (14.08.2014)
Published in Journal of medicinal chemistry (14.08.2014)
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Journal Article
Effect of 6-Benzoyl-benzothiazol-2-one scaffold on the pharmacological profile of α-alkoxyphenylpropionic acid derived PPAR agonists
Hurtevent, Aurélie, Le Naour, Morgan, Leclerc, Veronique, Carato, Pascal, Melnyk, Patricia, Hennuyer, Nathalie, Staels, Bart, Beucher-Gaudin, Monique, Caignard, Daniel-Henri, Dacquet, Catherine, Lebegue, Nicolas
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Journal Article
Effect of Oxime Ether Incorporation in Acyl Indole Derivatives on PPAR Subtype Selectivity
Le Naour, Morgan, Leclerc, Veronique, Farce, Amaury, Caignard, Daniel-Henri, Hennuyer, Nathalie, Staels, Bart, Audinot-Bouchez, Valérie, Boutin, Jean-Albert, Lonchampt, Michel, Dacquet, Catherine, Ktorza, Alain, Berthelot, Pascal, Lebegue, Nicolas
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
A Fentanyl Vaccine Alters Fentanyl Distribution and Protects against Fentanyl-Induced Effects in Mice and Rats
Raleigh, Michael D, Baruffaldi, Federico, Peterson, Samantha J, Le Naour, Morgan, Harmon, Theresa M, Vigliaturo, Jennifer R, Pentel, Paul R, Pravetoni, Marco
Published in The Journal of pharmacology and experimental therapeutics (01.02.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2019)
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Journal Article
Reduced Antinociception of Opioids in Rats and Mice by Vaccination with Immunogens Containing Oxycodone and Hydrocodone Haptens
Pravetoni, Marco, Le Naour, Morgan, Tucker, Ashli M, Harmon, Theresa M, Hawley, Tara M, Portoghese, Philip S, Pentel, Paul R
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Journal Article
COMPOSITIONS AND METHODS RELATED TO TAUOPATHY
Zhao Xiaohui, Le Naour Morgan Clotaire Paul, Hook Derek John, Ashe Karen Hsiao, Walters Michael Anthony
Year of Publication 25.05.2017
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Year of Publication 25.05.2017
Patent
Compositions and methods related to tauopathy
Zhao Xiaohui, Le Naour Morgan Clotaire Paul, Hook Derek John, Ashe Karen Hsiao, Walters Michael Anthony
Year of Publication 28.03.2017
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Year of Publication 28.03.2017
Patent
Nye heterosykliske sykloalkylforbindelser, en fremgangsmate for deres fremstilling og farmasoytiske sammensetninger inneholdende dem
HURTEVENT AURELIE, NAOUR MORGAN LE, DACQUET CATHERINE, L'HELGOUAL'CH JEAN-MARTIAL, CAIGNARD DANIEL-HENRI, LECLERC VERONIQUE, KTORZA ALAIN, CARATO PASCAL, BERTHELOT PASCAL, LEBEGUE NICOLAS
Year of Publication 16.09.2008
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Year of Publication 16.09.2008
Patent
COMPOSITIONS AND METHODS RELATED TO TAUOPATHY
LE NAOUR MORGAN CLOTAIRE PAUL, HOOK DEREK JOHN, WALTERS MICHAEL ANTHONY, ASHE KAREN HSIAO, ZHAO XIAOHUI
Year of Publication 02.06.2016
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Year of Publication 02.06.2016
Patent
Compositions and methods related to tauopathy
LE NAOUR MORGAN CLOTAIRE PAUL, HOOK DEREK JOHN, WALTERS MICHAEL ANTHONY, ASHE KAREN HSIAO, ZHAO XIAOHUI
Year of Publication 01.12.2015
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Year of Publication 01.12.2015
Patent
COMPOSITIONS AND METHODS OF TREATING OPIOID ADDICTION
LE NAOUR MORGAN C.P, PENTEL PAUL RICHARD, PORTOGHESE PHILIP S, PRAVETONI MARCO
Year of Publication 03.04.2014
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Year of Publication 03.04.2014
Patent
COMPOSITIONS AND METHODS RELATED TO TAUOPATHY
LE NAOUR MORGAN CLOTAIRE PAUL, HOOK DEREK JOHN, WALTERS MICHAEL ANTHONY, ASHE KAREN HSIAO, ZHAO XIAOHUI
Year of Publication 19.06.2014
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Year of Publication 19.06.2014
Patent
NOUVEAUX DERIVES HETEROCYCLIQUES, LEUR PROCEDE DE PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES QUI LES CONTIENNENT
DACQUET CATHERINE, LECLERC VERONIQUE, KTORZA ALAIN, BERTHELOT PASCAL, LEBEGUE NICOLAS, LE NAOUR MORGAN, PIRAT CELINE, CAIGNARD DANIEL HENRI
Year of Publication 04.12.2009
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Year of Publication 04.12.2009
Patent
Heterocyclic Cycloalkyl Compounds, a Process for their Preparation and Pharmaceutical Compositions Containing Them
HURTEVENT AURELIE, DACQUET CATHERINE, L'HELGOUAL'CH JEAN-MARTIAL, CAIGNARD DANIEL-HENRI, LECLERC VERONIQUE, KTORZA ALAIN, CARATO PASCAL, BERTHELOT PASCAL, LEBEGUE NICOLAS, LE NAOUR MORGAN
Year of Publication 24.09.2009
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Year of Publication 24.09.2009
Patent
NOVEL HETEROCYCLIC CYCLOALKYL DERIVATIVES, METHOD FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
BERTHELOT, PASCAL, DACQUET, CATHERINE, CARATO, PASCAL, HURTEVENT, AURELIE, L'HELGOUAL'CH, JEAN-MARTIAL, CAIGNARD, DANIEL-HENRI, KTORZA, ALAIN, LE NAOUR, MORGAN, LEBEGUE, NICOLAS, LECLERC, VERONIQUE
Year of Publication 19.11.2008
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Year of Publication 19.11.2008
Patent
NOVEL HETEROCYCLIC CYCLOALKYL DERIVATIVES ¼METHOD FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
HURTEVENT AURELIE, DACQUET CATHERINE, LECLERC VERONIQUE, KTORZA ALAIN, CARATO PASCAL, BERTHELOT PASCAL, L'HELGOUAL'CH JEAN MARTIAL, LEBEGUE NICOLAS, LE NAOUR MORGAN, CAIGNARD DANIEL HENRI
Year of Publication 13.11.2008
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Year of Publication 13.11.2008
Patent
NOUVEAUX DERIVES TETRACYCLIQUES, LEUR PROCEDE DE PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES QUI LES CONTIENNENT
DACQUET CATHERINE, LECLERC VERONIQUE, KTORZA ALAIN, CARATO PASCAL, BERTHELOT PASCAL, L'HELGOUAL'CH JEAN MARTIAL, LEBEGUE NICOLAS, LE NAOUR MORGAN, CAIGNARD DANIEL HENRI
Year of Publication 22.08.2008
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Year of Publication 22.08.2008
Patent
NOUVEAUX DERIVES HETEROCYCLIQUES CYCLOALKYLES, LEUR PROCEDE DE PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES QUI LES CONTIENNENT
HURTEVENT AURELIE, DACQUET CATHERINE, L HELGOUALJEAN MARTIAL, LECLERC VERONIQUE, KTORZA ALAIN, CARATO PASCAL, BERTHELOT PASCAL, LEBEGUE NICOLAS, LE NAOUR MORGAN
Year of Publication 13.06.2008
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Year of Publication 13.06.2008
Patent