Structural basis of organic cation transporter-3 inhibition
Khanppnavar, Basavraj, Maier, Julian, Herborg, Freja, Gradisch, Ralph, Lazzarin, Erika, Luethi, Dino, Yang, Jae-Won, Qi, Chao, Holy, Marion, Jäntsch, Kathrin, Kudlacek, Oliver, Schicker, Klaus, Werge, Thomas, Gether, Ulrik, Stockner, Thomas, Korkhov, Volodymyr M, Sitte, Harald H
Published in Nature communications (07.11.2022)
Published in Nature communications (07.11.2022)
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Journal Article
Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors
Gradisch, Ralph, Schlögl, Katharina, Lazzarin, Erika, Niello, Marco, Maier, Julian, Mayer, Felix P, Alves da Silva, Leticia, Skopec, Sophie M C, Blakely, Randy D, Sitte, Harald H, Mihovilovic, Marko D, Stockner, Thomas
Published in Nature communications (10.01.2024)
Published in Nature communications (10.01.2024)
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A comparative review on the well-studied GAT1 and the understudied BGT-1 in the brain
Bhatt, Manan, Gauthier-Manuel, Laure, Lazzarin, Erika, Zerlotti, Rocco, Ziegler, Christine, Bazzone, Andre, Stockner, Thomas, Bossi, Elena
Published in Frontiers in physiology (13.04.2023)
Published in Frontiers in physiology (13.04.2023)
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Journal Article
Elucidating allosteric communication in the human serotonin transporter
Lazzarin, Erika, Gradisch, Ralph, Alves da Silva, Leticia, Stockner, Thomas
Published in Biophysical journal (11.02.2022)
Published in Biophysical journal (11.02.2022)
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Journal Article
Free energy profile of the substrate-induced occlusion of the human serotonin transporter
Alves da Silva, Leticia, Lazzarin, Erika, Gradisch, Ralph, Clarke, Amy, Stockner, Thomas
Published in Journal of neurochemistry (05.02.2024)
Published in Journal of neurochemistry (05.02.2024)
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Occlusion of the human serotonin transporter is mediated by serotonin-induced conformational changes in the bundle domain
Gradisch, Ralph, Szöllősi, Dániel, Niello, Marco, Lazzarin, Erika, Sitte, Harald H., Stockner, Thomas
Published in The Journal of biological chemistry (01.03.2022)
Published in The Journal of biological chemistry (01.03.2022)
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Journal Article
Insights of hSERT transport mechanism revealed by Markov state models
Alves da Silva, Leticia, Gradisch, Ralph, Lazzarin, Erika, Szöllősi, Dániel, Stockner, Thomas
Published in Biophysical journal (11.02.2022)
Published in Biophysical journal (11.02.2022)
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Unveiling the crucial role of betaine: modulation of GABA homeostasis via SLC6A1 transporter (GAT1)
Bhatt, Manan, Lazzarin, Erika, Alberto-Silva, Ana Sofia, Domingo, Guido, Zerlotti, Rocco, Gradisch, Ralph, Bazzone, Andre, Sitte, Harald H., Stockner, Thomas, Bossi, Elena
Published in Cellular and molecular life sciences : CMLS (01.12.2024)
Published in Cellular and molecular life sciences : CMLS (01.12.2024)
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Journal Article
Interaction of GAT1 with sodium ions: from efficient recruitment to stabilisation of substrate and conformation
Lazzarin, Erika, Gradisch, Ralph, Sophie Mc Skopec, Leticia Alves Da Silva, Sebastianelli-Schoditsch, Chiara, Szollosi, Daniel, Maier, Julian, Sucic, Sonja, Roblek, Marko, Kanner, Baruch, Sitte, Harald H, Stockner, Thomas
Published in bioRxiv (22.02.2024)
Published in bioRxiv (22.02.2024)
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Paper
Interaction of GAT1 with sodium ions: from efficient recruitment to stabilisation of substrate and conformation
Lazzarin, Erika, Gradisch, Ralph, Skopec, Sophie M.C., Alves da Silva, Leticia, Sebastianelli-Schoditsch, Chiara, Szöllősi, Dániel, Maier, Julian, Sucic, Sonja, Roblek, Marko, Kanner, Baruch I., Sitte, Harald H., Stockner, Thomas
Year of Publication 13.10.2023
Year of Publication 13.10.2023
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Structural basis of organic cation transporter-3 inhibition
Khanppnavar, Basavraj, Maier, Julian, Herborg, Freja, Gradisch, Ralph, Lazzarin, Erika, Luethi, Dino, Jae-Won, Yang, Chao, Qi, Holy, Marion, Jaentsch, Kathrin, Kudlacek, Oliver, Schicker, Klaus, Werge, Thomas, Gether, Ulrik, Stockner, Thomas, Korkhov, Volodymyr, Sitte, Harald H
Published in bioRxiv (14.07.2022)
Published in bioRxiv (14.07.2022)
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Paper