Intracellular Released Payload Influences Potency and Bystander-Killing Effects of Antibody-Drug Conjugates in Preclinical Models
Li, Fu, Emmerton, Kim K, Jonas, Mechthild, Zhang, Xinqun, Miyamoto, Jamie B, Setter, Jocelyn R, Nicholas, Nicole D, Okeley, Nicole M, Lyon, Robert P, Benjamin, Dennis R, Law, Che-Leung
Published in Cancer research (Chicago, Ill.) (01.05.2016)
Published in Cancer research (Chicago, Ill.) (01.05.2016)
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Journal Article
Tumor-Associated Macrophages Can Contribute to Antitumor Activity through FcγR-Mediated Processing of Antibody-Drug Conjugates
Li, Fu, Ulrich, Michelle, Jonas, Mechthild, Stone, Ivan J, Linares, Germein, Zhang, Xinqun, Westendorf, Lori, Benjamin, Dennis R, Law, Che-Leung
Published in Molecular cancer therapeutics (01.07.2017)
Published in Molecular cancer therapeutics (01.07.2017)
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Development of orally active inhibitors of protein and cellular fucosylation
Okeley, Nicole M., Alley, Stephen C., Anderson, Martha E., Boursalian, Tamar E., Burke, Patrick J., Emmerton, Kim M., Jeffrey, Scott C., Klussman, Kerry, Law, Che-Leung, Sussman, Django, Toki, Brian E., Westendorf, Lori, Zeng, Weiping, Zhang, Xinqun, Benjamin, Dennis R., Senter, Peter D.
Published in Proceedings of the National Academy of Sciences - PNAS (02.04.2013)
Published in Proceedings of the National Academy of Sciences - PNAS (02.04.2013)
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The Pharmacologic Basis for Antibody-Auristatin Conjugate Activity
Alley, Stephen C, Zhang, Xinqun, Okeley, Nicole M, Anderson, Martha, Law, Che-Leung, Senter, Peter D, Benjamin, Dennis R
Published in The Journal of pharmacology and experimental therapeutics (01.09.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2009)
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Journal Article
Lysosomal Trafficking and Cysteine Protease Metabolism Confer Target-specific Cytotoxicity by Peptide-linked Anti-CD30-Auristatin Conjugates
Sutherland, May S. Kung, Sanderson, Russell J., Gordon, Kristine A., Andreyka, Jamie, Cerveny, Charles G., Yu, Changpu, Lewis, Timothy S., Meyer, Damon L., Zabinski, Roger F., Doronina, Svetlana O., Senter, Peter D., Law, Che-Leung, Wahl, Alan F.
Published in The Journal of biological chemistry (14.04.2006)
Published in The Journal of biological chemistry (14.04.2006)
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Journal Article
Potent Anticarcinoma Activity of the Humanized Anti-CD70 Antibody h1F6 Conjugated to the Tubulin Inhibitor Auristatin via an Uncleavable Linker
OFLAZOGLU, Ezogelin, STONE, Ivan J, GORDON, Kristine, WOOD, Christopher G, REPASKY, Elizabeth A, GREWAL, Iqbal S, LAW, Che-Leung, GERBERA, Hans-Peter
Published in Clinical cancer research (01.10.2008)
Published in Clinical cancer research (01.10.2008)
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Macrophages contribute to the antitumor activity of the anti-CD30 antibody SGN-30
Oflazoglu, Ezogelin, Stone, Ivan J., Gordon, Kristine A., Grewal, Iqbal S., van Rooijen, Nico, Law, Che-Leung, Gerber, Hans-Peter
Published in Blood (15.12.2007)
Published in Blood (15.12.2007)
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Blocking of CD27-CD70 Pathway by Anti-CD70 Antibody Ameliorates Joint Disease in Murine Collagen-Induced Arthritis
Oflazoglu, Ezogelin, Boursalian, Tamar E, Zeng, Weiping, Edwards, Ana C, Duniho, Steve, McEarchern, Julie A, Law, Che-Leung, Gerber, Hans-Peter, Grewal, Iqbal S
Published in The Journal of immunology (1950) (15.09.2009)
Published in The Journal of immunology (1950) (15.09.2009)
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Preclinical Characterization of SGN-70, a Humanized Antibody Directed against CD70
MCEARCHERN, Julie A, SMITH, Leia M, GREWAL, Iqbal S, LAW, Che-Leung, MCDONAGH, Charlotte F, KLUSSMAN, Kerry, GORDON, Kristine A, MORRIS-TILDEN, Carol A, DUNIHO, Steven, RYAN, Maureen, BOURSALIAN, Tamar E, CARTER, Paul J
Published in Clinical cancer research (01.12.2008)
Published in Clinical cancer research (01.12.2008)
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Journal Article
Lymphocyte activation antigen CD70 expressed by renal cell carcinoma is a potential therapeutic target for anti-CD70 antibody-drug conjugates
LAW, Che-Leung, GORDON, Kristine A, SAUTER, Guido, OFLAZOGLU, Ezogelin, DORONINA, Svetlana O, MEYER, Damon L, FRANCISCO, Joseph A, CARTER, Paul, SENTER, Peter D, COPLAND, John A, WOOD, Christopher G, WAHL, Alan F, TOLD, Brian E, YAMANE, Andrew K, HERING, Michelle A, CERVENY, Charles G, PETROZIELLO, Joseph M, RYAN, Maureen C, SMITH, Leia, SIMON, Ronald
Published in Cancer research (Chicago, Ill.) (15.02.2006)
Published in Cancer research (Chicago, Ill.) (15.02.2006)
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CD27-CD70 interactions in the pathogenesis of Waldenström macroglobulinemia
Ho, Allen W., Hatjiharissi, Evdoxia, Ciccarelli, Bryan T., Branagan, Andrew R., Hunter, Zachary R., Leleu, Xavier, Tournilhac, Olivier, Xu, Lian, O'Connor, Kelly, Manning, Robert J., Santos, Daniel Ditzel, Chemaly, Mariana, Patterson, Christopher J., Soumerai, Jacob D., Munshi, Nikhil C., McEarchern, Julie A., Law, Che-Leung, Grewal, Iqbal S., Treon, Steven P.
Published in Blood (01.12.2008)
Published in Blood (01.12.2008)
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Efficient Elimination of B-Lineage Lymphomas by Anti-CD20–Auristatin Conjugates
LAW, Che-Leung, CERVENY, Charles G, SENTER, Peter D, WAHL, Alan F, GORDON, Kristine A, KLUSSMAN, Kerry, MIXAN, Bruce J, CHACE, Dana F, MEYER, Damon L, DORONINA, Svetlana O, SIEGALL, Clay B, FRANCISCO, Joseph A
Published in Clinical cancer research (01.12.2004)
Published in Clinical cancer research (01.12.2004)
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Suppression subtractive hybridization and expression profiling identifies a unique set of genes overexpressed in non-small-cell lung cancer
PETROZIELLO, Joseph, YAMANE, Andrew, WESTENDORF, Lori, THOMPSON, Melissa, MCDONAGH, Charlotte, CERVENY, Charles, LAW, Che-Leung, WAHL, Alan, CARTER, Paul
Published in Oncogene (07.10.2004)
Published in Oncogene (07.10.2004)
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Preclinical Characterization of HPN536, a Trispecific, T-Cell-Activating Protein Construct for the Treatment of Mesothelin-Expressing Solid Tumors
Molloy, Mary Ellen, Austin, Richard J, Lemon, Bryan D, Aaron, Wade H, Ganti, Vaishnavi, Jones, Adrie, Jones, Susan D, Strobel, Kathryn L, Patnaik, Purbasa, Sexton, Kenneth, Tatalick, Laurie, Yu, Timothy Z, Baeuerle, Patrick A, Law, Che-Leung, Wesche, Holger
Published in Clinical cancer research (01.03.2021)
Published in Clinical cancer research (01.03.2021)
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A Potent Anti-CD70 Antibody–Drug Conjugate Combining a Dimeric Pyrrolobenzodiazepine Drug with Site-Specific Conjugation Technology
Jeffrey, Scott C, Burke, Patrick J, Lyon, Robert P, Meyer, David W, Sussman, Django, Anderson, Martha, Hunter, Joshua H, Leiske, Chris I, Miyamoto, Jamie B, Nicholas, Nicole D, Okeley, Nicole M, Sanderson, Russell J, Stone, Ivan J, Zeng, Weiping, Gregson, Stephen J, Masterson, Luke, Tiberghien, Arnaud C, Howard, Philip W, Thurston, David E, Law, Che-Leung, Senter, Peter D
Published in Bioconjugate chemistry (17.07.2013)
Published in Bioconjugate chemistry (17.07.2013)
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Anti-leukemic activity of Lintuzumab (SGN-33) in preclinical models of acute myeloid leukemia
Sutherland, May Kung, Yu, Changpu, Lewis, Timothy S., Miyamoto, Jamie B., Morris-Tilden, Carol A., Jonas, Mechthild, Sutherland, Jennifer, Nesterova, Albina, Gerber, Hans-Peter, Sievers, Eric L., Grewal, Iqbal S., Law, Che-Leung
Published in mAbs (01.09.2009)
Published in mAbs (01.09.2009)
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Journal Article
5-Azacytidine enhances the anti-leukemic activity of lintuzumab (SGN-33) in preclinical models of acute myeloid leukemia
Sutherland, May Kung, Yu, Changpu, Anderson, Martha, Zeng, Weiping, van Rooijen, Nico, Sievers, Eric L., Grewal, Iqbal S., Law, Che-Leung
Published in mAbs (01.07.2010)
Published in mAbs (01.07.2010)
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Brentuximab Vedotin-Driven Microtubule Disruption Results in Endoplasmic Reticulum Stress Leading to Immunogenic Cell Death and Antitumor Immunity
Heiser, Ryan A, Cao, Anthony T, Zeng, Weiping, Ulrich, Michelle, Younan, Patrick, Anderson, Martha E, Trueblood, Esther S, Jonas, Mechthild, Thurman, Robert, Law, Che-Leung, Gardai, Shyra J
Published in Molecular cancer therapeutics (03.01.2024)
Published in Molecular cancer therapeutics (03.01.2024)
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TriTACs, a Novel Class of T-Cell-Engaging Protein Constructs Designed for the Treatment of Solid Tumors
Austin, Richard J, Lemon, Bryan D, Aaron, Wade H, Barath, Manasi, Culp, Patricia A, DuBridge, Robert B, Evnin, Luke B, Jones, Adrie, Panchal, Anand, Patnaik, Purbasa, Ramakrishnan, Vanitha, Rocha, Sony S, Seto, Pui, Sexton, Kenneth, Strobel, Kathryn L, Wall, Russell, Yu, Stephen, Yu, Timothy Z, Law, Che-Leung, Baeuerle, Patrick A, Wesche, Holger
Published in Molecular cancer therapeutics (01.01.2021)
Published in Molecular cancer therapeutics (01.01.2021)
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