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Unsaturated acyl chains dramatically enhanced cellular uptake by direct translocation of a minimalist oligo-arginine lipopeptide
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The Two NK-1 Binding Sites Correspond to Distinct, Independent, and Non-Interconvertible Receptor Conformational States As Confirmed by Plasmon-Waveguide Resonance Spectroscopy
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Relative DNA binding affinity of helix 3 homeodomain analogues, major groove binders, can be rapidly screened by displacement of prebound ethidium bromide. A comparative study
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Analogs of Substance P modified at the C-terminus which are both agonist and antagonist of the NK-1 receptor depending on the second messenger pathway
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Published in The journal of peptide research (01.05.2002)
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Incorporation of vinylogous scaffolds in the C-terminal tripeptide of substance P
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Unsaturated acyl chains dramatically enhanced cellular uptake by direct translocation of a minimalist oligo-arginine lipopeptideElectronic supplementary information (ESI) available: All the experimental procedures are described in SI with the characterization of all the lipopeptides. See DOI: 10.1039/c5cc06116d
Swiecicki, J.-M, Di Pisa, M, Lippi, F, Chwetzoff, S, Mansuy, C, Trugnan, G, Chassaing, G, Lavielle, S, Burlina, F
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Insulin binding to its receptor induces a conformational change in the receptor C-terminus
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Published in Biochemistry (Easton) (15.05.1990)
Published in Biochemistry (Easton) (15.05.1990)
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Distinct presynaptic control of dopamine release in striosomal- and matrix-enriched areas of the rat striatum by selective agonists of NK1, NK2 and NK3 tachykinin receptors
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Published in Regulatory peptides (02.07.1993)
Published in Regulatory peptides (02.07.1993)
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Analysis of tachykinin binding site interactions using constrained analogues of tachykinins
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Published in Biochemical pharmacology (01.01.1988)
Published in Biochemical pharmacology (01.01.1988)
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