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Published in Bioorganic & medicinal chemistry (01.07.2008)
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Phytosphingosine 1-phosphate: a high affinity ligand for the S1P4/Edg-6 receptor
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Published in Biochemical and biophysical research communications (01.09.2002)
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Design and synthesis of conformationally constrained tri-substituted ureas as potent antagonists of the human glucagon receptor
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Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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Discovery of novel, potent, and orally active spiro-urea human glucagon receptor antagonists
Shen, Dong-Ming, Zhang, Fengqi, Brady, Edward J., Candelore, Mari Rios, Dallas-Yang, Qing, Ding, Victor D.-H., Dragovic, Jasminka, Feeney, William P., Jiang, Guoquiang, McCann, Peggy E., Mock, Steve, Qureshi, Sajjad A., Saperstein, Richard, Shen, Xiaolan, Tamvakopoulos, Constantin, Tong, Xinchun, Tota, Laurie M., Wright, Michael J., Yang, Xiaodong, Zheng, Song, Chapman, Kevin T., Zhang, Bei B., Tata, James R., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (15.10.2005)
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Direct observation (NMR) of the efficacy of glucagon receptor antagonists in murine liver expressing the human glucagon receptor
Cohen, Sheila M., Duffy, Joseph L., Miller, Corin, Kirk, Brian A., Candelore, Mari Rios, Ding, Victor D.H., Kaczorowski, Gregory, Tota, Laurie M., Werrmann, Jeffrey G., Wright, Michael, Parmee, Emma R., Tata, James R., Zhang, Bei B.
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Published in Journal of medicinal chemistry (19.10.2000)
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Potent, selective human β3 adrenergic receptor agonists containing a substituted indoline-5-sulfonamide pharmacophore
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Published in Bioorganic & medicinal chemistry letters (01.07.1999)
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Parmee, Emma R., Ok, Hyun O., Candelore, Mari R., Tota, Laurie, Deng, Liping, Strader, Catherine D., Wyvratt, Matthew J., Fisher, Michael H., Weber, Ann E.
Published in Bioorganic & medicinal chemistry letters (01.05.1998)
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A novel series of indazole-/indole-based glucagon receptor antagonists
Lin, Songnian, Zhang, Fengqi, Jiang, Guoqiang, Qureshi, Sajjad A., Yang, Xiaodong, Chicchi, Gary G., Tota, Laurie, Bansal, Alka, Brady, Edward, Trujillo, Maria, Salituro, Gino, Miller, Corey, Tata, James R., Zhang, Bei B., Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (01.10.2015)
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Human β 3-adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides
Brockunier, Linda L, Parmee, Emma R, Ok, Hyun O, Candelore, Mari R, Cascieri, Margaret A, Colwell, Lawrence F, Deng, Liping, Feeney, William P, Forrest, Michael J, Hom, Gary J, MacIntyre, D.Euan, Tota, Laurie, Wyvratt, Matthew J, Fisher, Michael H, Weber, Ann E
Published in Bioorganic & medicinal chemistry letters (18.09.2000)
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Discovery of cyclic guanidines as potent, orally active, human glucagon receptor antagonists
Sinz, Christopher, Chang, Jiang, Lins, Ashley Rouse, Brady, Ed, Candelore, Mari, Dallas-Yang, Qing, Ding, Victor, Jiang, Guoqiang, Lin, Zhen, Mock, Steven, Qureshi, Sajjad, Salituro, Gino, Saperstein, Richard, Shang, Jackie, Szalkowski, Deborah, Tota, Laurie, Vincent, Stella, Wright, Michael, Xu, Shiyao, Yang, Xiaodong, Zhang, Bei, Tata, James, Kim, Ronald, Parmee, Emma
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
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Human β3-Adrenergic receptor agonists containing 1,2,3-triazole-substituted benzenesulfonamides
BROCKUNIER, Linda L, PARMEE, Emma R, MACINTYRE, D. Euan, TOTA, Laurie, WYVRATT, Matthew J, FISHER, Michael H, WEBER, Ann E, OK, Hyun O, CANDELORE, Mari R, CASCIERI, Margaret A, COLWELL, Lawrence F, LIPING DENG, FEENEY, William P, FORREST, Michael J, HOM, Gary J
Published in Bioorganic & medicinal chemistry letters (01.09.2000)
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Sinz, Christopher, Bittner, Amy, Brady, Ed, Candelore, Mari, Dallas-Yang, Qing, Ding, Victor, Jiang, Guoqiang, Lin, Zhen, Qureshi, Sajjad, Salituro, Gino, Saperstein, Richard, Shang, Jackie, Szalkowski, Deborah, Tota, Laurie, Vincent, Stella, Wright, Michael, Xu, Shiyao, Yang, Xiaodong, Zhang, Bei, Tata, James, Kim, Ronald, Parmee, Emma R.
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
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Potent, selective benzenesulfonamide agonists of the human β3 adrenergic receptor
WEBER, A. E, MATHVINK, R. J, PERKINS, L, HUTCHINS, J. E, CANDELORE, M. R, TOTA, L, STRADER, C. D, WYVRATT, M. J, FISHER, M. H
Published in Bioorganic & medicinal chemistry letters (01.05.1998)
Published in Bioorganic & medicinal chemistry letters (01.05.1998)
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Phytosphingosine 1-phosphate: a high affinity ligand for the S1P(4)/Edg-6 receptor
Candelore, Mari Rios, Wright, Michael J, Tota, Laurie M, Milligan, James, Shei, Gan-ju, Bergstrom, James D, Mandala, Suzanne M
Published in Biochemical and biophysical research communications (27.09.2002)
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Published in Biochemical and biophysical research communications (27.09.2002)
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Phytosphingosine 1-phosphate: a high affinity ligand for the S1P 4/Edg-6 receptor
Rios Candelore, Mari, Wright, Michael J, Tota, Laurie M, Milligan, James, Shei, Gan-ju, Bergstrom, James D, Mandala, Suzanne M
Published in Biochemical and biophysical research communications (2002)
Published in Biochemical and biophysical research communications (2002)
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