The Heptahelical Domain of GABAB2 Is Activated Directly by CGP7930, a Positive Allosteric Modulator of the GABAB Receptor
Virginie Binet, Carole Brajon, Laurent Le Corre, Francine Acher, Jean-Philippe Pin, Laurent Prézeau
Published in The Journal of biological chemistry (09.07.2004)
Published in The Journal of biological chemistry (09.07.2004)
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A Single Subunit (GB2) Is Required for G-protein Activation by the Heterodimeric GABAB Receptor
Duthey, Béatrice, Caudron, Sara, Perroy, Julie, Bettler, Bernhard, Fagni, Laurent, Pin, Jean-Philippe, Prézeau, Laurent
Published in The Journal of biological chemistry (01.02.2002)
Published in The Journal of biological chemistry (01.02.2002)
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Asymmetric Functioning of Dimeric Metabotropic Glutamate Receptors Disclosed by Positive Allosteric Modulators
Goudet, Cyril, Kniazeff, Julie, Hlavackova, Veronika, Malhaire, Fanny, Maurel, Damien, Acher, Francine, Blahos, Jaroslav, Prézeau, Laurent, Pin, Jean-Philippe
Published in The Journal of biological chemistry (01.07.2005)
Published in The Journal of biological chemistry (01.07.2005)
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CPCCOEt, a Noncompetitive Metabotropic Glutamate Receptor 1 Antagonist, Inhibits Receptor Signaling Without Affecting Glutamate Binding
Litschig, S, Gasparini, F, Rueegg, D, Stoehr, N, Flor, P J, Vranesic, I, Prézeau, L, Pin, J P, Thomsen, C, Kuhn, R
Published in Molecular pharmacology (01.03.1999)
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Published in Molecular pharmacology (01.03.1999)
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BAY36-7620: A Potent Non-Competitive mGlu1 Receptor Antagonist with Inverse Agonist Activity
Carroll, F Y, Stolle, A, Beart, P M, Voerste, A, Brabet, I, Mauler, F, Joly, C, Antonicek, H, Bockaert, J, Müller, T, Pin, J P, Prézeau, L
Published in Molecular pharmacology (01.05.2001)
Published in Molecular pharmacology (01.05.2001)
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Real-Time Analysis of Agonist-Induced Activation of Protease-Activated Receptor 1/Gαi1 Protein Complex Measured by Bioluminescence Resonance Energy Transfer in Living Cells
Mohammed A. Ayoub, Damien Maurel, Virginie Binet, Michel Fink, Laurent Prézeau, Hervé Ansanay, Jean-Philippe Pin
Published in Molecular pharmacology (01.05.2007)
Published in Molecular pharmacology (01.05.2007)
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Amino-Pyrrolidine Tricarboxylic Acids Give New Insight into Group III Metabotropic Glutamate Receptor Activation Mechanism
Frauli, Mélanie, Hubert, Nadia, Schann, Stephan, Triballeau, Nicolas, Bertrand, Hugues-Olivier, Acher, Francine, Neuville, Pascal, Pin, Jean-Philippe, Prézeau, Laurent
Published in Molecular pharmacology (01.03.2007)
Published in Molecular pharmacology (01.03.2007)
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The Second Intracellular Loop of Metabotropic Glutamate Receptors Recognizes C Termini of G-protein α-Subunits
Michaela Havlickova, Jaroslav Blahos, Isabelle Brabet, Jianfeng Liu, Bohdana Hruskova, Laurent Prézeau, Jean-Philippe Pin
Published in The Journal of biological chemistry (12.09.2003)
Published in The Journal of biological chemistry (12.09.2003)
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A Cluster of Basic Residues in the Carboxyl-terminal Tail of the Short Metabotropic Glutamate Receptor 1 Variants Impairs Their Coupling to Phospholipase C
Mary, Sophie, Gomeza, Jesus, Prézeau, Laurent, Bockaert, Joël, Pin, Jean-Philippe
Published in The Journal of biological chemistry (02.01.1998)
Published in The Journal of biological chemistry (02.01.1998)
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Mapping the Agonist-binding Site of GABAB Type 1 Subunit Sheds Light on the Activation Process of GABABReceptors
Galvez, Thierry, Prézeau, Laurent, Milioti, Gérald, Franek, Miloslav, Joly, Cécile, Froestl, Wolfgang, Bettler, Bernhard, Bertrand, Hugues-Olivier, Blahos, Jaroslav, Pin, Jean-Philippe
Published in The Journal of biological chemistry (29.12.2000)
Published in The Journal of biological chemistry (29.12.2000)
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Ca2+ Requirement for High-Affinity γ-Aminobutyric Acid (GABA) Binding at GABAB Receptors: Involvement of Serine 269 of the GABABR1 Subunit
Thierry Galvez, Stephan Urwyler, Laurent Prézeau, Johannes Mosbacher, Cécile Joly, Barbara Malitschek, Jakob Heid, Isabelle Brabet, Wolfgang Froestl, Bernhard Bettler, Klemens Kaupmann, Jean-Philippe Pin
Published in Molecular pharmacology (01.03.2000)
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Published in Molecular pharmacology (01.03.2000)
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