Evaluation of the effects of RP5063, a novel, multimodal, serotonin receptor modulator, as single-agent therapy and co-administrated with sildenafil, bosentan, and treprostinil in a monocrotaline-induced pulmonary arterial hypertension rat model
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Published in European journal of pharmacology (15.05.2018)
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Dual antiplatelet and anticoagulant APAC prevents experimental ischemia–reperfusion-induced acute kidney injury
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Published in Frontiers in cardiovascular medicine (14.12.2022)
Published in Frontiers in cardiovascular medicine (14.12.2022)
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RP5063, a novel, multimodal, serotonin receptor modulator, prevents monocrotaline-induced pulmonary arterial hypertension in rats
Bhat, Laxminarayan, Hawkinson, Jon, Cantillon, Marc, Reddy, Dasharatha G., Bhat, Seema R., Laurent, Charles E., Bouchard, Annie, Biernat, Marzena, Salvail, Dany
Published in European journal of pharmacology (05.09.2017)
Published in European journal of pharmacology (05.09.2017)
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Prostanoid receptor subtypes involved in treprostinil-mediated vasodilation of rat pulmonary arteries and in treprostinil-mediated inhibition of collagen gene expression of human lung fibroblasts
Corboz, Michel R., Salvail, William, Gagnon, Sandra, LaSala, Daniel, Laurent, Charles E., Salvail, Dany, Chen, Kuan-Ju, Cipolla, David, Perkins, Walter R., Chapman, Richard W.
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Published in Prostaglandins & other lipid mediators (01.02.2021)
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RP5063, a novel, multimodal, serotonin receptor modulator, prevents Sugen 5416-hypoxia–induced pulmonary arterial hypertension in rats
Bhat, Laxminarayan, Hawkinson, Jon, Cantillon, Marc, Reddy, Dasharatha G., Bhat, Seema R., Laurent, Charles E., Bouchard, Annie, Biernat, Marzena, Salvail, Dany
Published in European journal of pharmacology (05.09.2017)
Published in European journal of pharmacology (05.09.2017)
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Preclinical Pharmacology and Pharmacokinetics of Inhaled Hexadecyl-Treprostinil (C16TR), a Pulmonary Vasodilator Prodrug
Corboz, Michel R, Li, Zhili, Malinin, Vladimir, Plaunt, Adam J, Konicek, Donna M, Leifer, Franziska G, Chen, Kuan-Ju, Laurent, Charles E, Yin, Han, Biernat, Marzena C, Salvail, Dany, Zhuang, Jianguo, Xu, Fadi, Curran, Aidan, Perkins, Walter R, Chapman, Richard W
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Published in The Journal of pharmacology and experimental therapeutics (01.12.2017)
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Inhaled Treprostinil-Prodrug Lipid Nanoparticle Formulations Provide Long-Acting Pulmonary Vasodilation
Leifer, Franziska G, Konicek, Donna M, Chen, Kuan-Ju, Plaunt, Adam J, Salvail, Dany, Laurent, Charles E, Corboz, Michel R, Li, Zhili, Chapman, Richard W, Perkins, Walter R, S Malinin, Vladimir
Published in Drug research (01.11.2018)
Published in Drug research (01.11.2018)
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Inhaled hexadecyl-treprostinil provides pulmonary vasodilator activity at significantly lower plasma concentrations than infused treprostinil
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Functional desensitization to isoproterenol without reducing cAMP production in canine failing cardiocytes
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Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.02.2001)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.02.2001)
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Functional desensitization to isoproterenol without reducing cAMP production in canine failing cardiocytes
LAURENT, Charles-E, CARDINAL, René, ROUSSEAU, Guy, VERMEULEN, Michel, BOUCHARD, Caroline, WILKINSON, Michael, ARMOUR, J. Andrew, BOUVIER, Michel
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.02.2001)
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Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.02.2001)
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Hypoxia-induced release of prostaglandins: mechanisms and sources of production in coronary resistance vessels of the isolated rabbit heart
Nakhostine, N, Laurent, C E, Nadeau, R, Cardinal, R, Lamontagne, D
Published in Canadian journal of physiology and pharmacology (01.12.1995)
Published in Canadian journal of physiology and pharmacology (01.12.1995)
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