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Abu Rabe, Dina, Chdid, Lhoucine, Lamson, David R, Laudeman, Christopher P, Tarpley, Michael, Elsayed, Naglaa, Smith, Ginger R, Zheng, Weifan, Dixon, Maria S, Williams, Kevin P
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Published in Molecules (Basel, Switzerland) (28.06.2024)
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Structure-Activity Relationships of a Series of Echinocandins and the Discovery of CD101, a Highly Stable and Soluble Echinocandin with Distinctive Pharmacokinetic Properties
James, Kenneth D, Laudeman, Christopher P, Malkar, Navdeep B, Krishnan, Radha, Polowy, Karen
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Published in Antimicrobial agents and chemotherapy (01.02.2017)
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N-substituted phenylbenzamides of the niclosamide chemotype attenuate obesity related changes in high fat diet fed mice
Bhagat, Hiral A, Compton, Sarah A, Musso, David L, Laudeman, Christopher P, Jackson, Kimberly M P, Yi, Na Young, Nierobisz, Lidia S, Forsberg, Lawrence, Brenman, Jay E, Sexton, Jonathan Z
Published in PloS one (25.10.2018)
Published in PloS one (25.10.2018)
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Identification of harmine and β-carboline analogs from a high-throughput screen of an approved drug collection; profiling as differential inhibitors of DYRK1A and monoamine oxidase A and for in vitro and in vivo anti-cancer studies
Tarpley, Michael, Oladapo, Helen O., Strepay, Dillon, Caligan, Thomas B., Chdid, Lhoucine, Shehata, Hassan, Roques, Jose R., Thomas, Rhashad, Laudeman, Christopher P., Onyenwoke, Rob U., Darr, David B., Williams, Kevin P.
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Published in European journal of pharmaceutical sciences (01.07.2021)
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Discovery of 5-[[4-[(2,3-Dimethyl-2H-indazol-6-yl)methylamino]-2-pyrimidinyl]amino]-2-methyl-benzenesulfonamide (Pazopanib), a Novel and Potent Vascular Endothelial Growth Factor Receptor Inhibitor
Harris, Philip A, Boloor, Amogh, Cheung, Mui, Kumar, Rakesh, Crosby, Renae M, Davis-Ward, Ronda G, Epperly, Andrea H, Hinkle, Kevin W, Hunter, Robert N, Johnson, Jennifer H, Knick, Victoria B, Laudeman, Christopher P, Luttrell, Deirdre K, Mook, Robert A, Nolte, Robert T, Rudolph, Sharon K, Szewczyk, Jerzy R, Truesdale, Anne T, Veal, James M, Wang, Liping, Stafford, Jeffrey A
Published in Journal of medicinal chemistry (14.08.2008)
Published in Journal of medicinal chemistry (14.08.2008)
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Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120)
Sparks, Steven M., Chen, Grace, Collins, Jon L., Danger, Dana, Dock, Steven T., Jayawickreme, Channa, Jenkinson, Stephen, Laudeman, Christopher, Leesnitzer, M. Anthony, Liang, Xi, Maloney, Patrick, McCoy, David C., Moncol, David, Rash, Vincent, Rimele, Thomas, Vulimiri, Padmaja, Way, James M., Ross, Sean
Published in Bioorganic & medicinal chemistry letters (15.07.2014)
Published in Bioorganic & medicinal chemistry letters (15.07.2014)
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Discovery of small molecule agonists for the bombesin receptor subtype 3 (BRS-3) based on an omeprazole lead
Carlton, David L., Collin-Smith, Lissa J., Daniels, Alejandro J., Deaton, David N., Goetz, Aaron S., Laudeman, Christopher P., Littleton, Thomas R., Musso, David L., Morgan, Ronda J. Ott, Szewczyk, Jerzy R., Zhang, Cunyu
Published in Bioorganic & medicinal chemistry (15.10.2008)
Published in Bioorganic & medicinal chemistry (15.10.2008)
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Journal Article
Discovery of 5-[[4-[(2,3-dimethyl-2H-indazol-6-yl)methylamino]-2-pyrimidinyl]amino]-2-methylbenzenesulfonamide (pazopanib), a novel and potent vascular endothelial growth factor receptor inhibitor
Harris, Philip A., Boloor, Amogh, Cheung, Mui, Kumar, Rakesh, Crosby, Renae M., Davis-Ward, Ronda G., Epperly, Andrea H., Hinkle, Kevin W., Hunter, Robert N., Johnson, Jennifer H., Knick, Victoria B., Laudeman, Christopher P., Luttrell, Deirdre K., Mook, Robert A., Nolte, Robert T., Rudolph, Sharon K., Szewczyk, Jerzy R., Truesdale, Anne T., Veal, James M., Wang, Liping, Stafford, Jeffrey A.
Published in Journal of medicinal chemistry (14.08.2008)
Published in Journal of medicinal chemistry (14.08.2008)
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Journal Article
1H-INDOLE-2-CARBOXYLIC ACID DERIVATIVES USEFUL AS PPAR MODULATORS
OPLINGER JEFFREY ALAN, LAUDEMAN CHRISTOPHER P, RAY JOHN A, BANKER PIERETTE, SPEARING PAUL KENNETH, LAMBERT MILLARD HURST, SZEWCZYK JERZY R
Year of Publication 06.07.2009
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Year of Publication 06.07.2009
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MALKAR, Navdeep Balkrishna, LAUDEMAN, Christopher Patrick, JAMES, JR., Kenneth Duke, RADHAKRISHNAN, Balasingam
Year of Publication 26.05.2022
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Year of Publication 26.05.2022
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Year of Publication 09.12.2020
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Year of Publication 09.12.2020
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Year of Publication 30.07.2018
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Year of Publication 30.07.2018
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ANTIFUNGAL AGENTS AND USES THEREOF
RADHAKRISHNAN, BALASINGHAM, JAMES, KENNETH DUKE, LAUDEMAN, CHRISTOPHER PATRICK, MALKAR, NAVDEEP BALKRISHNA
Year of Publication 08.10.2019
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Year of Publication 08.10.2019
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R-BIND 2.0: An Updated Database of Bioactive RNA-Targeting Small Molecules and Associated RNA Secondary Structures
Donlic, Anita, Swanson, Emily G, Liang-Yuan, Chiu, Wicks, Sarah L, Juru, Aline Umuhire, Cai, Zhengguo, Kassam, Kamillah J, Laudeman, Christopher, Sanaba, Bilva, Sugarman, Andrew, Han, Eunseong, Tolbert, Blanton S, Hargrove, Amanda E
Published in bioRxiv (15.03.2022)
Published in bioRxiv (15.03.2022)
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Paper
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Radhakrishnan, Balasingam, Malkar, Navdeep Balkrishna, James, Kenneth Duke, Laudeman, Christopher Patrick
Year of Publication 14.12.2018
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Year of Publication 14.12.2018
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MALKAR, Navdeep Balkrishna, LAUDEMAN, Christopher Patrick, JAMES, Kenneth Duke, RADHAKRISHNAN, Balasingam
Year of Publication 28.09.2018
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Year of Publication 28.09.2018
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Malkar, Navdeep Balkrishna, Radhakrishnan, Balasingham, James, Kenneth Duke, Laudeman, Christopher Patrick
Year of Publication 09.02.2018
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Year of Publication 09.02.2018
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RADHAKRISHNAN, BALASINGHAM, LAUDEMAN, CHRISTOPHER, PATRICK, MALKAR, NAVDEEP, BALKRISHNA, JAMES, KENNETH, DUKE, JR
Year of Publication 31.01.2018
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Year of Publication 31.01.2018
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ANTIFUNGAL AGENTS AND USES THEREOF
JAMES, KENNETH DUKE JR, LAUDEMAN, CHRISTOPHER PATRICK, MALKAR, NAVDEEP BALKRISHNA, RADHAKRISHNAN, BALASINGAM
Year of Publication 31.01.2018
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Year of Publication 31.01.2018
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