TH1902, a new docetaxel‐peptide conjugate for the treatment of sortilin‐positive triple‐negative breast cancer
Demeule, Michel, Charfi, Cyndia, Currie, Jean‐Christophe, Larocque, Alain, Zgheib, Alain, Kozelko, Sophie, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer science (01.10.2021)
Published in Cancer science (01.10.2021)
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New Peptide-Drug Conjugates for Precise Targeting of SORT1-Mediated Vasculogenic Mimicry in the Tumor Microenvironment of TNBC-Derived MDA-MB-231 Breast and Ovarian ES-2 Clear Cell Carcinoma Cells
Charfi, Cyndia, Demeule, Michel, Currie, Jean-Christophe, Larocque, Alain, Zgheib, Alain, Danalache, Bogdan Alexandru, Ouanouki, Amira, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Frontiers in oncology (22.10.2021)
Published in Frontiers in oncology (22.10.2021)
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Journal Article
The Peptide-Drug Conjugate TH1902: A New Sortilin Receptor-Mediated Cancer Therapeutic against Ovarian and Endometrial Cancers
Currie, Jean-Christophe, Demeule, Michel, Charfi, Cyndia, Zgheib, Alain, Larocque, Alain, Danalache, Bogdan Alexandru, Ouanouki, Amira, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancers (08.04.2022)
Published in Cancers (08.04.2022)
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Journal Article
Abstract 6362: TH1901, a novel curcumin-peptide conjugate for the treatment of Sortilin-positive (SORT1+) cancer
Annabi, Borhane, Demeule, Michel, Currie, Jean-Christophe, Larocque, Alain, Zgheib, Alain, Marsolais, Christian, Béliveau, Richard
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
Abstract 685: Sortilin receptor-mediated novel cancer therapy: A targeted approach to inhibit vasculogenic mimicry in ovarian and breast cancers
Currie, Jean-Christophe, Demeule, Michel, Larocque, Alain, Zgheib, Alain, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
Abstract 1313: TH1902, a docetaxel peptide-drug conjugate, shows pre-clinical efficacy in several Sortilin-positive (SORT1+) cancers
Marsolais, Christian, Currie, Jean-Christophe, Demeule, Michel, Charfi, Cyndia, Larocque, Alain, Zgheib, Alain, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article
Abstract 1439: Increasing potency of anticancer drugs through SORT1+ technology: A new targeted approach for the treatment of ovarian and endometrial cancers
Demeule, Michel, Currie, Jean-Christophe, Charfi, Cyndia, Larocque, Alain, Zgheib, Alain, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Use of a Noninvasive Brain-Penetrating Peptide-Drug Conjugate Strategy to Improve the Delivery of Opioid Pain Relief Medications to the Brain
Eiselt, Émilie, Otis, Valérie, Belleville, Karine, Yang, Gaoqiang, Larocque, Alain, Régina, Anthony, Demeule, Michel, Sarret, Philippe, Gendron, Louis
Published in The Journal of pharmacology and experimental therapeutics (01.07.2020)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2020)
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Journal Article
Increasing potency and safety of anticancer drugs through sortilin receptor-mediated cancer therapy: A new targeted approach for the treatment of ovarian cancer
Annabi, Borhane, Demeule, Michel, Currie, Jean-Christophe, Larocque, Alain, Charfi, Cyndia, Béliveau, Richard
Published in Journal of clinical oncology (20.05.2019)
Published in Journal of clinical oncology (20.05.2019)
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Journal Article
Abstract 1061: Increasing potency of anticancer drugs through Sortilin receptor-mediated cancer therapy: A new targeted approach for the treatment of ovarian cancer
Demeule, Michel, Currie, Jean-Christophe, Charfi, Cyndia, Larocque, Alain, Zgheib, Alain, Kozelko, Sophie, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
Abstract 2910: A novel Sortilin-targeted docetaxel peptide conjugate (TH1902), for the treatment of Sortilin-positive (SORT1+) triple-negative breast cancer
Marsolais, Christian, Charfi, Cyndia, Demeule, Michel, Currie, Jean-Christophe, Larocque, Alain, Zgheib, Alain, Duquette, Natacha, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Journal Article
Abstract P3-10-07: Receptor-mediated chemotherapy using a new Docetaxel-peptide conjugate for Sortilin-positive triple-negative breast cancer
Demeule, Michel, Charfi, Cyndia, Currie, Jean-Christophe C, Larocque, Alain, Zgheib, Alain, Marsolais, Christian, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.02.2020)
Published in Cancer research (Chicago, Ill.) (15.02.2020)
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소틸린 결합 접합체 화합물, 조성물 및 암을 치료하기 위한 이들의 용도
MARSOLAIS CHRISTIAN, DEMEULE MICHEL, CURRIE JEAN CHRISTOPHE, LAROCQUE ALAIN
Year of Publication 17.08.2022
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Year of Publication 17.08.2022
Patent
Abstract 5146: Increasing penetration of anticancer drugs through sortilin receptor-mediated cancer therapy: A new targeted and personalized Approach in the treatment of ovarian cancer
Demeule, Michel, Curie, Jean-Christophe, Larocque, Alain, Charfi, Cyndia, Béliveau, Richard, Vezeau, Claude, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Conjugation of a brain-penetrant peptide with neurotensin provides antinociceptive properties
Demeule, Michel, Beaudet, Nicolas, Régina, Anthony, Besserer-Offroy, Élie, Murza, Alexandre, Tétreault, Pascal, Belleville, Karine, Ché, Christian, Larocque, Alain, Thiot, Carine, Béliveau, Richard, Longpré, Jean-Michel, Marsault, Éric, Leduc, Richard, Lachowicz, Jean E, Gonias, Steven L, Castaigne, Jean-Paul, Sarret, Philippe
Published in The Journal of clinical investigation (01.03.2014)
Published in The Journal of clinical investigation (01.03.2014)
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암 줄기 세포를 표적화하기 위한 방법 및 소르틸린 결합 접합체 화합물
ANNABI BORHANE, MARSOLAIS CHRISTIAN, DEMEULE MICHEL, CURRIE JEAN CHRISTOPHE, LAROCQUE ALAIN, CHARFI CYNDIA, ZGHEIB ALAIN, BELIVEAU RICHARD
Year of Publication 07.12.2023
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Year of Publication 07.12.2023
Patent
Abstract 1076: The peptide-drug conjugate TH1902 inhibits growth of subcutaneous melanoma xenografts and formation of lung metastases in a syngeneic mouse model
Demeule, Michel, Currie, Jean-Christophe, Charfi, Cyndia, Larocque, Alain, Zgheib, Alain, Kozelko, Sophie, Béliveau, Richard, Marsolais, Christian, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
Abstract 1853: TH1902, a SORT1 docetaxel peptide-drug conjugate, inhibits tumor growth of human cancer stem-like cells (CD133+) from both triple-negative breast cancers and ovarian cancers
Marsolais, Christian, Charfi, Cyndia, Demeule, Michel, Currie, Jean-Christophe, Zgheib, Alain, Larocque, Alain, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
Abstract 1079: Anti-cancer efficacy of TH1902, a SORT1 docetaxel peptide-drug conjugate, against ovarian and endometrial cancers xenografts alone or in combination with carboplatin
Marsolais, Christian, Demeule, Michel, Charfi, Cyndia, Currie, Jean-Christophe, Larocque, Alain, Zgheib, Alain, Béliveau, Richard, Annabi, Borhane
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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