The discovery of quinoline-3-carboxamides as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors
Deaton, David N., Do, Young, Holt, Jason, Jeune, Michael R., Kramer, H. Fritz, Larkin, Andrew L., Orband-Miller, Lisa A., Peckham, Gregory E., Poole, Chuck, Price, Daniel J., Schaller, Lee T., Shen, Ying, Shewchuk, Lisa M., Stewart, Eugene L., Stuart, J. Darren, Thomson, Stephen A., Ward, Paris, Wilson, Joseph W., Xu, Tianshun, Guss, Jeffrey H., Musetti, Caterina, Rendina, Alan R., Affleck, Karen, Anders, David, Hancock, Ashley P., Hobbs, Heather, Hodgson, Simon T., Hutchinson, Jonathan, Leveridge, Melanie V., Nicholls, Harry, Smith, Ian E.D., Somers, Don O., Sneddon, Helen F., Uddin, Sorif, Cleasby, Anne, Mortenson, Paul N., Richardson, Caroline, Saxty, Gordon
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Published in Bioorganic & medicinal chemistry (15.04.2019)
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Directed ortho Metalation−Boronation and Suzuki−Miyaura Cross Coupling of Pyridine Derivatives: A One-Pot Protocol to Substituted Azabiaryls
Alessi, Manlio, Larkin, Andrew L, Ogilvie, Kevin A, Green, Laine A, Lai, Sunny, Lopez, Simon, Snieckus, Victor
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Opioid receptor modulation of hedonic taste preference and food intake: a single-dose safety, pharmacokinetic, and pharmacodynamic investigation with GSK1521498, a novel μ-opioid receptor inverse agonist
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Published in Journal of clinical pharmacology (01.04.2012)
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H-PGDS 억제제로서의 퀴놀린-3-카르복스아미드
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Year of Publication 27.08.2018
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Year of Publication 27.08.2018
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Regulation of ingestive behaviors in the rat by GSK1521498, a novel micro-opioid receptor-selective inverse agonist
Ignar, Diane M, Goetz, Aaron S, Noble, Kimberly Nichols, Carballo, Luz Helena, Stroup, Andrea E, Fisher, Julie C, Boucheron, Joyce A, Brainard, Tracy A, Larkin, Andrew L, Epperly, Andrea H, Shearer, Todd W, Sorensen, Scott D, Speake, Jason D, Hommel, Jonathan D
Published in The Journal of pharmacology and experimental therapeutics (01.10.2011)
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Chemical Compounds
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Year of Publication 13.01.2022
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Year of Publication 13.01.2022
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Year of Publication 14.05.2020
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Year of Publication 14.05.2020
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CHEMICAL COMPOUNDS
CADILLA, RODOLFO, LARKIN, ANDREW L, DEATON, DAVID NORMAN, SCHULTE, CHRISTIE, SMALLEY JR, TERRENCE L
Year of Publication 14.05.2020
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Year of Publication 14.05.2020
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Quinoline-3-carboxamides as H-PGDS inhibitors
Saxty, Gordon, Mortenson, Paul N, Deaton, Dave Norman, Wilson, Joseph Wendell, Price, Daniel J, Cadilla, Rodolfo, Thomson, Stephen Andrew, Hodgson, Simon Teanby, Larkin, Andrew L, Le, Joelle, Schaller, Lee T, Smith, Ian Edward David, Hancock, Ashley Paul, Hobbs, Heather, Schulte, Christie
Year of Publication 25.07.2019
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Year of Publication 25.07.2019
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Chemical compounds
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Year of Publication 01.11.2020
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Year of Publication 01.11.2020
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Quinoline-3-carboxamides as H-PGDS inhibitors
Saxty, Gordon, Mortenson, Paul N, Deaton, Dave Norman, Wilson, Joseph Wendell, Price, Daniel J, Cadilla, Rodolfo, Thomson, Stephen Andrew, Hodgson, Simon Teanby, Larkin, Andrew L, Le, Joelle, Schaller, Lee T, Smith, Ian Edward David, Hancock, Ashley Paul, Hobbs, Heather, Schulte, Christie
Year of Publication 14.06.2018
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Year of Publication 14.06.2018
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NUEVOS COMPUESTOS INHIBIDORES DE LA PROSTAGLANDINA D SINTASA HEMATOPOYÉTICA (H-PGDS)
Andrew L LARKIN, Terrence L. SMALLEY Jr, CADILLA Rodolfo, David Norman DEATON, SCHULTE Christie
Year of Publication 29.05.2020
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Year of Publication 29.05.2020
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QUINOLINE-3-CARBOXAMIDES AS H-PGDS INHIBITORS
HANCOCK, Ashley Paul, PRICE, Daniel J, HODGSON, Simon Teanby, DEATON, Dave Norman, MORTENSON, Paul N, LE, Joelle, SAXTY, Gordon, SMITH, Ian Edward David, THOMSON, Stephen Andrew, WILSON, Joseph Wendell, HOBBS, Heather, SCHULTE, Christie, LARKIN, Andrew L, CADILLA, Rodolfo, SCHALLER, Lee T
Year of Publication 24.10.2018
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Year of Publication 24.10.2018
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QUINOLINE-3-CARBOXAMIDES AS H-PGDS INHIBITORS
HANCOCK, Ashley Paul, PRICE, Daniel J, HODGSON, Simon Teanby, DEATON, Dave Norman, MORTENSON, Paul N, LE, Joelle, SAXTY, Gordon, SMITH, Ian Edward David, THOMSON, Stephen Andrew, WILSON, Joseph Wendell, HOBBS, Heather, SCHULTE, Christie, LARKIN, Andrew L, CADILLA, Rodolfo, SCHALLER, Lee T
Year of Publication 22.06.2017
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Year of Publication 22.06.2017
Patent
QUINOLINE-3-CARBOXAMIDES AS H-PGDS INHIBITORS
HODGSON, SIMON TEANBY, DEATON, DAVE NORMAN, LE, JOELLE, SAXTY, GORDON, THOMSON, STEPHEN ANDREW, HANCOCK, ASHLEY PAUL, PRICE, DANIEL J, SMITH, IAN EDWARD DAVID, WILSON, JOSEPH WENDELL, CADILLA, RODOLFO, LARKIN, ANDREW L, SCHULTE, CHRISTIE, SCHALLER, LEE T, HOBBS, HEATHER, MORTENSON, PAUL N
Year of Publication 22.06.2017
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Year of Publication 22.06.2017
Patent
Directed ortho-Metalation-Boronation and Suzuki-Miyaura Cross-Coupling of Pyridine Derivatives: A One-Pot Protocol to Substituted Azabiaryls
Alessi, Manlio, Larkin, Andrew L., Ogilvie, Kevin A., Green, Laine A., Lai, Sunny, Lopez, Simon, Snieckus, Victor
Published in ChemInform (10.07.2007)
Published in ChemInform (10.07.2007)
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Journal Article
quinolina-3-carboxamidas como inibidores da h-pgds
LEE T. SCHALLER, ANDREW L. LARKIN, STEPHEN ANDREW THOMSON, RODOLFO CADILLA, IAN EDWARD DAVID SMITH, DANIEL J. PRICE, SIMON TEANBY HODGSON, CHRISTIE SCHULTE, JOELLE LE, GORDON SAXTY, HEATHER HOBBS, PAUL N. MORTENSON, DAVE NORMAN DEATON, JOSEPH WENDELL WILSON, ASHLEY PAUL HANCOCK
Year of Publication 18.12.2018
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Year of Publication 18.12.2018
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Aniline derivatives as selective androgen receptor modulators
TURNBULL PHILIP S, KALDOR ISTVAN, STEWART EUGENE L, CADILLA RODOLFO, COWAN DAVID J, LARKIN ANDREW L
Year of Publication 16.08.2007
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Year of Publication 16.08.2007
Patent
QUINOLINE-3-CARBOXAMIDES AS H-PGDS INHIBITORS
SMITH IAN EDWARD DAVID, THOMSON STEPHEN ANDREW, CADILLA RODOLFO, HODGSON SIMON TEANBY, SCHALLER LEE T, PRICE DANIEL J, HOBBS HEATHER, SCHULTE CHRISTIE, WILSON JOSEPH WENDELL, LARKIN ANDREW L, HANCOCK ASHLEY PAUL, DEATON DAVE NORMAN, LE JOELLE, SAXTY GORDON, MORTENSON PAUL N
Year of Publication 21.08.2018
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Year of Publication 21.08.2018
Patent
COMPUESTO DE QUINOLIN-3-CARBOXAMIDA, COMPOSICIÓN FARMACÉUTICA QUE LO COMPRENDE Y SU USO PARA PREPARARLA
LEE T. SCHALLER, STEPHEN ANDREW THOMSON, ANDREW L. LARKIN, RODOLFO CADILLA, IAN EDWARD DAVID SMITH, SIMON TEANBY HODGSON, DANIEL J. PRICE, JOELLE LE, CHRISTIE SCHULTE, GORDON SAXTY, HEATHER HOBBS, PAUL N. MORTENSON, DAVE NORMAN DEATON, JOSEPH WENDELL WILSON, ASHLEY PAUL HANCOCK
Year of Publication 14.03.2018
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Year of Publication 14.03.2018
Patent