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Published in Nature communications (11.07.2016)
Published in Nature communications (11.07.2016)
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A new inhibitor of the β-arrestin/AP2 endocytic complex reveals interplay between GPCR internalization and signalling
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Published in Nature communications (18.04.2017)
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Dynamic spatiotemporal determinants modulate GPCR:G protein coupling selectivity and promiscuity
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Functional selectivity profiling of the angiotensin II type 1 receptor using pathway-wide BRET signaling sensors
Namkung, Yoon, LeGouill, Christian, Kumar, Sahil, Cao, Yubo, Teixeira, Larissa B, Lukasheva, Viktoriya, Giubilaro, Jenna, Simões, Sarah C, Longpré, Jean-Michel, Devost, Dominic, Hébert, Terence E, Piñeyro, Graciela, Leduc, Richard, Costa-Neto, Claudio M, Bouvier, Michel, Laporte, Stéphane A
Published in Science signaling (04.12.2018)
Published in Science signaling (04.12.2018)
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Intrinsic bias at non-canonical, β-arrestin-coupled seven transmembrane receptors
Pandey, Shubhi, Kumari, Punita, Baidya, Mithu, Kise, Ryoji, Cao, Yubo, Dwivedi-Agnihotri, Hemlata, Banerjee, Ramanuj, Li, Xaria X., Cui, Cedric S., Lee, John D., Kawakami, Kouki, Maharana, Jagannath, Ranjan, Ashutosh, Chaturvedi, Madhu, Jhingan, Gagan Deep, Laporte, Stéphane A., Woodruff, Trent M., Inoue, Asuka, Shukla, Arun K.
Published in Molecular cell (18.11.2021)
Published in Molecular cell (18.11.2021)
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The experimental power of FR900359 to study Gq-regulated biological processes
Schrage, Ramona, Schmitz, Anna-Lena, Gaffal, Evelyn, Annala, Suvi, Kehraus, Stefan, Wenzel, Daniela, Büllesbach, Katrin M, Bald, Tobias, Inoue, Asuka, Shinjo, Yuji, Galandrin, Ségolène, Shridhar, Naveen, Hesse, Michael, Grundmann, Manuel, Merten, Nicole, Charpentier, Thomas H, Martz, Matthew, Butcher, Adrian J, Slodczyk, Tanja, Armando, Sylvain, Effern, Maike, Namkung, Yoon, Jenkins, Laura, Horn, Velten, Stößel, Anne, Dargatz, Harald, Tietze, Daniel, Imhof, Diana, Galés, Céline, Drewke, Christel, Müller, Christa E, Hölzel, Michael, Milligan, Graeme, Tobin, Andrew B, Gomeza, Jesús, Dohlman, Henrik G, Sondek, John, Harden, T Kendall, Bouvier, Michel, Laporte, Stéphane A, Aoki, Junken, Fleischmann, Bernd K, Mohr, Klaus, König, Gabriele M, Tüting, Thomas, Kostenis, Evi
Published in Nature communications (14.12.2015)
Published in Nature communications (14.12.2015)
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Manifold roles of β-arrestins in GPCR signaling elucidated with siRNA and CRISPR/Cas9
Luttrell, Louis M, Wang, Jialu, Plouffe, Bianca, Smith, Jeffrey S, Yamani, Lama, Kaur, Suneet, Jean-Charles, Pierre-Yves, Gauthier, Christophe, Lee, Mi-Hye, Pani, Biswaranjan, Kim, Jihee, Ahn, Seungkirl, Rajagopal, Sudarshan, Reiter, Eric, Bouvier, Michel, Shenoy, Sudha K, Laporte, Stéphane A, Rockman, Howard A, Lefkowitz, Robert J
Published in Science signaling (25.09.2018)
Published in Science signaling (25.09.2018)
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Allosteric modulation of GPCR-induced β-arrestin trafficking and signaling by a synthetic intrabody
Baidya, Mithu, Chaturvedi, Madhu, Dwivedi-Agnihotri, Hemlata, Ranjan, Ashutosh, Devost, Dominic, Namkung, Yoon, Stepniewski, Tomasz Maciej, Pandey, Shubhi, Baruah, Minakshi, Panigrahi, Bhanupriya, Sarma, Parishmita, Yadav, Manish K, Maharana, Jagannath, Banerjee, Ramanuj, Kawakami, Kouki, Inoue, Asuka, Selent, Jana, Laporte, Stéphane A, Hébert, Terence E, Shukla, Arun K
Published in Nature communications (08.08.2022)
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Molecular insights into intrinsic transducer-coupling bias in the CXCR4-CXCR7 system
Sarma, Parishmita, Carino, Carlo Marion C, Seetharama, Deeksha, Pandey, Shubhi, Dwivedi-Agnihotri, Hemlata, Rui, Xue, Cao, Yubo, Kawakami, Kouki, Kumari, Poonam, Chen, Yu-Chih, Luker, Kathryn E, Yadav, Prem N, Luker, Gary D, Laporte, Stéphane A, Chen, Xin, Inoue, Asuka, Shukla, Arun K
Published in Nature communications (09.08.2023)
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Structure-toxicity relationships of saturated and unsaturated free fatty acids for elucidating the lipotoxic effects in human EndoC-βH1 beta-cells
Plötz, T., von Hanstein, A.S., Krümmel, B., Laporte, A., Mehmeti, I., Lenzen, S.
Published in Biochimica et biophysica acta. Molecular basis of disease (01.11.2019)
Published in Biochimica et biophysica acta. Molecular basis of disease (01.11.2019)
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Differential β-arrestin-dependent conformational signaling and cellular responses revealed by angiotensin analogs
Zimmerman, Brandon, Beautrait, Alexandre, Aguila, Benjamin, Charles, Ricardo, Escher, Emanuel, Claing, Audrey, Bouvier, Michel, Laporte, Stéphane A
Published in Science signaling (24.04.2012)
Published in Science signaling (24.04.2012)
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Genetic code expansion and photocross-linking identify different β-arrestin binding modes to the angiotensin II type 1 receptor
Gagnon, Laurence, Cao, Yubo, Cho, Aaron, Sedki, Dana, Huber, Thomas, Sakmar, Thomas P., Laporte, Stéphane A.
Published in The Journal of biological chemistry (15.11.2019)
Published in The Journal of biological chemistry (15.11.2019)
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Discovery of a dual Ras and ARF6 inhibitor from a GPCR endocytosis screen
Giubilaro, Jenna, Schuetz, Doris A., Stepniewski, Tomasz M., Namkung, Yoon, Khoury, Etienne, Lara-Márquez, Mónica, Campbell, Shirley, Beautrait, Alexandre, Armando, Sylvain, Radresa, Olivier, Duchaine, Jean, Lamarche-Vane, Nathalie, Claing, Audrey, Selent, Jana, Bouvier, Michel, Marinier, Anne, Laporte, Stéphane A.
Published in Nature communications (03.08.2021)
Published in Nature communications (03.08.2021)
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Prostaglandin F2α and angiotensin II type 1 receptors exhibit differential cognate G protein coupling regulation
Sedki, Dana, Cho, Aaron, Cao, Yubo, Nikolajev, Ljiljana, Atmuri, N. D. Prasad, Lubell, William D., Laporte, Stéphane A.
Published in The Journal of biological chemistry (01.09.2022)
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β-Arrestin-mediated Angiotensin II Signaling Controls the Activation of ARF6 Protein and Endocytosis in Migration of Vascular Smooth Muscle Cells
Charles, Ricardo, Namkung, Yoon, Cotton, Mathieu, Laporte, Stéphane A., Claing, Audrey
Published in The Journal of biological chemistry (19.02.2016)
Published in The Journal of biological chemistry (19.02.2016)
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β-Arrestin 2: A Receptor-Regulated MAPK Scaffold for the Activation of JNK3
McDonald, Patricia H., Chow, Chi-Wing, Miller, William E., Laporte, Stéphane A., Field, Michael E., Lin, Fang-Tsyr, Davis, Roger J., Lefkowitz, Robert J.
Published in Science (American Association for the Advancement of Science) (24.11.2000)
Published in Science (American Association for the Advancement of Science) (24.11.2000)
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Risk Score Derived from Pre-operative Data Analysis Predicts the Need for Biventricular Mechanical Circulatory Support
Fitzpatrick, J. Raymond, MD, Frederick, John R., MD, Hsu, Vivian M., MD, Kozin, Elliott D., BA, O'Hara, Mary Lou, MSN, Howell, Elan, BSN, Dougherty, Deborah, BSN, McCormick, Ryan C., BS, Laporte, Carine A., BA, Cohen, Jeffrey E., BA, Southerland, Kevin W., BS, Howard, Jessica L., BS, Jessup, Mariell L., MD, Morris, Rohinton J., MD, Acker, Michael A., MD, Woo, Y. Joseph, MD
Published in The Journal of heart and lung transplantation (01.12.2008)
Published in The Journal of heart and lung transplantation (01.12.2008)
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