Brain accumulation of sunitinib is restricted by P-glycoprotein (ABCB1) and breast cancer resistance protein (ABCG2) and can be enhanced by oral elacridar and sunitinib coadministration
Tang, Seng Chuan, Lagas, Jurjen S., Lankheet, Nienke A.G., Poller, Birk, Hillebrand, Michel J., Rosing, Hilde, Beijnen, Jos H., Schinkel, Alfred H.
Published in International journal of cancer (01.01.2012)
Published in International journal of cancer (01.01.2012)
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Dose recommendations for anticancer drugs in patients with renal or hepatic impairment
Krens, Stefanie D, Lassche, Gerben, Jansman, Frank G A, Desar, Ingrid M E, Lankheet, Nienke A G, Burger, David M, van Herpen, Carla M L, van Erp, Nielka P
Published in The lancet oncology (01.04.2019)
Published in The lancet oncology (01.04.2019)
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Plasma concentrations of tyrosine kinase inhibitors imatinib, erlotinib, and sunitinib in routine clinical outpatient cancer care
Lankheet, Nienke A G, Knapen, Lotte M, Schellens, Jan H M, Beijnen, Jos H, Steeghs, Neeltje, Huitema, Alwin D R
Published in Therapeutic drug monitoring (01.06.2014)
Published in Therapeutic drug monitoring (01.06.2014)
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The QT interval prolongation potential of anticancer and supportive drugs: a comprehensive overview
Giraud, Eline L, Ferrier, Kaylee R M, Lankheet, Nienke A G, Desar, Ingrid M E, Steeghs, Neeltje, Beukema, Rypko J, van Erp, Nielka P, Smolders, Elise J
Published in The lancet oncology (01.09.2022)
Published in The lancet oncology (01.09.2022)
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Relatively mild symptoms after chronic overdose with a double-dose encorafenib: a case report
Mian, Paola, Meussen, Elvera, Piersma, Djura, Lankheet, Nienke A G
Published in Anti-cancer drugs (01.06.2021)
Published in Anti-cancer drugs (01.06.2021)
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Optimizing the dose in cancer patients treated with imatinib, sunitinib and pazopanib
Lankheet, Nienke A. G., Desar, Ingrid M. E., Mulder, Sasja F., Burger, David M., Kweekel, Dinemarie M., Herpen, Carla M. L., Graaf, Winette T. A., Erp, Nielka P.
Published in British journal of clinical pharmacology (01.10.2017)
Published in British journal of clinical pharmacology (01.10.2017)
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P-glycoprotein (ABCB1) and breast cancer resistance protein (ABCG2) restrict brain accumulation of the active sunitinib metabolite N-desethyl sunitinib
Tang, Seng Chuan, Lankheet, Nienke A G, Poller, Birk, Wagenaar, Els, Beijnen, Jos H, Schinkel, Alfred H
Published in The Journal of pharmacology and experimental therapeutics (01.04.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2012)
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Concentrations of Erlotinib in Tumor Tissue and Plasma in Non–Small-Cell Lung Cancer Patients After Neoadjuvant Therapy
Lankheet, Nienke A.G, Schaake, Eva E, Burgers, Sjaak A, van Pel, Renée, Beijnen, Jos H, Huitema, Alwin D.R, Klomp, Houke
Published in Clinical lung cancer (01.07.2015)
Published in Clinical lung cancer (01.07.2015)
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Quantification of sunitinib and N-desethyl sunitinib in human EDTA plasma by liquid chromatography coupled with electrospray ionization tandem mass spectrometry: validation and application in routine therapeutic drug monitoring
Lankheet, Nienke A G, Steeghs, N, Rosing, H, Schellens, J H M, Beijnen, J H, Huitema, A D R
Published in Therapeutic drug monitoring (01.04.2013)
Published in Therapeutic drug monitoring (01.04.2013)
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Brain Accumulation of Dasatinib Is Restricted by P-Glycoprotein (ABCB1) and Breast Cancer Resistance Protein (ABCG2) and Can Be Enhanced by Elacridar Treatment
LAGAS, Jurjen S, VAN WATERSCHOOT, Robert A. B, VAN TILBURG, VickyA. C. J, HILLEBRAND, Michel J, LANKHEET, Nienke, ROSING, Hilde, BEIJNEN, Jos H, SCHINKEL, Alfred H
Published in Clinical cancer research (01.04.2009)
Published in Clinical cancer research (01.04.2009)
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Dasatinib in combination with fludarabine in patients with refractory chronic lymphocytic leukemia: A multicenter phase 2 study
Kater, Arnon P, Spiering, Marjolein, Liu, Roberto D, Doreen te Raa, G, Slinger, E, Tonino, Sanne H, Beckers, Marielle M, Daenen, Simon, Doorduijn, Jeanette K, Lankheet, Nienke A.G, Luijks, Dieuwertje M, Eldering, Eric, van Oers, Marinus H.J
Published in Leukemia research (01.01.2014)
Published in Leukemia research (01.01.2014)
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Use of the Child-Pugh score in anticancer drug dosing decision making: proceed with caution – Authors' reply
Krens, Stefanie D, Lassche, Gerben, Jansman, Frank G A, Desar, Ingrid M E, Lankheet, Nienke A G, Burger, David M, van Herpen, Carla M L, van Erp, Nielka P
Published in The lancet oncology (01.06.2019)
Published in The lancet oncology (01.06.2019)
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The effect of seasonal variation and secretion of sunitinib in sweat on the development of hand–foot syndrome
Lankheet, Nienke A. G., Huitema, Alwin D. R., Mallo, Henk, Adriaansz, Sandra, Haanen, John B. A. G., Schellens, Jan H. M., Beijnen, Jos H., Blank, Christian U.
Published in European journal of clinical pharmacology (01.12.2013)
Published in European journal of clinical pharmacology (01.12.2013)
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Erlotinib and pantoprazole: a relevant interaction or not?
Ter Heine, Rob, Fanggiday, James C., Lankheet, Nienke A. G., Beijnen, Jos H., Van Der Westerlaken, Monique M. L., Staaks, Gerald H. A., Malingré, Mirte M.
Published in British journal of clinical pharmacology (01.12.2010)
Published in British journal of clinical pharmacology (01.12.2010)
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Determination of Sunitinib and Its Active Metabolite N-Desethylsunitinib in Sweat of a Patient
Lankheet, Nienke A.G., Blank, Christian U., Mallo, Henk, Adriaansz, Sandra, Rosing, Hilde, Schellens, Jan H.M., Huitema, Alwin D.R., Beijnen, Jos H.
Published in Journal of analytical toxicology (01.10.2011)
Published in Journal of analytical toxicology (01.10.2011)
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Phase 1 Study of Combination Treatment with PTK 787/ZK 222584 and Cetuximab for Patients with Advanced Solid Tumors: Safety, Pharmacokinetics, Pharmacodynamics Analysis
Langenberg, Marlies H.G., Witteveen, Petronella O., Lankheet, Nienke A.G., Roodhart, Jeanine M.L., Rosing, Hilde, van den Heuvel, Ingeborg J.G.M., Beijnen, Jos H., Voest, Emile E.
Published in Neoplasia (New York, N.Y.) (01.02.2010)
Published in Neoplasia (New York, N.Y.) (01.02.2010)
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Relatively mild symptoms after an olanzapine intoxication in a 2-year-old girl with excessively high serum levels
Lankheet, Nienke A G, Padberg, Roos D, de Kluiver, Evelyne M, Wilhelm, Abraham J, van Woensel, Job B M, Beijnen, Jos H, Huitema, Alwin D R
Published in Journal of child and adolescent psychopharmacology (01.02.2011)
Published in Journal of child and adolescent psychopharmacology (01.02.2011)
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Sunitinib in Refractory Adrenocortical Carcinoma: A Phase II, Single-Arm, Open-Label Trial
Kroiss, Matthias, Quinkler, Marcus, Johanssen, Sarah, van Erp, Nielka P, Lankheet, Nienke, Pöllinger, Alexander, Laubner, Katharina, Strasburger, Christian J, Hahner, Stefanie, Müller, Hans-Helge, Allolio, Bruno, Fassnacht, Martin
Published in The journal of clinical endocrinology and metabolism (01.10.2012)
Published in The journal of clinical endocrinology and metabolism (01.10.2012)
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Development of an online drug-drug interaction resource to support safe prescription of oncolytics
Van Erp, Nielka P., Ferrier, Kaylee R.M., Gibbons, Sarah E., Burger, David, McAllister, Katie, Martin, Jasmine L.M., Khoo, Saye H., Jansman, Frank, Lankheet, Nienke A.G.
Published in Journal of clinical oncology (20.05.2018)
Published in Journal of clinical oncology (20.05.2018)
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Abstract 1518: P-glycoprotein (ABCB1) and breast cancer resistance protein (ABCG2) limit sunitinib brain accumulation which can be enhanced by oral elacridar treatment
Tang, Seng Chuan, Lagas, Jurjen S., Lankheet, Nienke, Rosing, Hilde, Beijnen, Jos H., Schinkel, Alfred H.
Published in Cancer research (Chicago, Ill.) (15.04.2010)
Published in Cancer research (Chicago, Ill.) (15.04.2010)
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