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Published in SLAS discovery (01.06.2020)
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Published in Nucleic acids research (01.01.2005)
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Quantitative Comparison of Enrichment from DNA-Encoded Chemical Library Selections
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Published in Bioorganic & medicinal chemistry letters (01.07.2018)
Published in Bioorganic & medicinal chemistry letters (01.07.2018)
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Discovery and Optimization of Quinolinone Derivatives as Potent, Selective, and Orally Bioavailable Mutant Isocitrate Dehydrogenase 1 (mIDH1) Inhibitors
Lin, Jian, Lu, Wei, Caravella, Justin A, Campbell, Ann Marie, Diebold, R. Bruce, Ericsson, Anna, Fritzen, Edward, Gustafson, Gary R, Lancia, David R, Shelekhin, Tatiana, Wang, Zhongguo, Castro, Jennifer, Clarke, Andrea, Gotur, Deepali, Josephine, Helen R, Katz, Marie, Diep, Hien, Kershaw, Mark, Yao, Lili, Kauffman, Goss, Hubbs, Stephen E, Luke, George P, Toms, Angela V, Wang, Liann, Bair, Kenneth W, Barr, Kenneth J, Dinsmore, Christopher, Walker, Duncan, Ashwell, Susan
Published in Journal of medicinal chemistry (25.07.2019)
Published in Journal of medicinal chemistry (25.07.2019)
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Discovery and optimization of novel piperazines as potent inhibitors of fatty acid synthase (FASN)
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Published in Bioorganic & medicinal chemistry letters (15.04.2019)
Published in Bioorganic & medicinal chemistry letters (15.04.2019)
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ACTIVATING PYRUVATE KINASE R
DAVID RICHARD, ANNA ERICKSON, ZHENG XIAOZHANG, LORNA MITCHELL, TATIANA SHELEKHIN, DABID R LANCIA JR, GARY GUSTAFSON, NEAL GREEN, LIN JIAN
Year of Publication 01.02.2024
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Year of Publication 30.01.2024
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HDAC 억제제로서의 이소인돌린
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PYRROLOPYRROLE COMPOSITION AS PYRUVATE KINASE (PKR) ACTIVATOR
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Year of Publication 05.12.2019
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PKR PYRROLOPYRROLE COMPOSITIONS AS PYRUVATE KINASE PKR ACTIVATORS
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Year of Publication 06.11.2017
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Activating pyruvate kinase R
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Year of Publication 22.10.2024
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Year of Publication 22.10.2024
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BICYCLIC [4,6,0] HYDROXAMIC ACIDS AS HDAC INHIBITORS
Lancia, JR., David R, Ng, Pui Yee, Rudnitskaya, Aleksandra, Zheng, Xiaozhang
Year of Publication 09.11.2023
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Year of Publication 09.11.2023
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Bicyclic [4,6,0] hydroxamic acids as HDAC inhibitors
Lancia, Jr., David R, Ng, Pui Yee, Rudnitskaya, Aleksandra, Zheng, Xiaozhang
Year of Publication 18.07.2023
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Year of Publication 18.07.2023
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