Novel Rapidly Diversifiable Antimicrobial RNA Polymerase Switch Region Inhibitors with Confirmed Mode of Action in Haemophilus influenzae
Buurman, Ed T, Foulk, Melinda A, Gao, Ning, Laganas, Valerie A, McKinney, David C, Moustakas, Demetri T, Rose, Jonathan A, Shapiro, Adam B, Fleming, Paul R
Published in Journal of Bacteriology (01.10.2012)
Published in Journal of Bacteriology (01.10.2012)
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Characterization of novel respiratory syncytial virus inhibitors identified by high throughput screen
Laganas, Valerie A., Dunn, Ewan F., McLaughlin, Robert E., Tiong-Yip, Choi Lai, Yuzhakov, Olga, Isabella, Vincent M., Hill, Pamela, Yu, Qin
Published in Antiviral research (01.03.2015)
Published in Antiviral research (01.03.2015)
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The Role of a Novel Auxiliary Pocket in Bacterial Phenylalanyl-tRNA Synthetase Druggability
Abibi, Ayome, Ferguson, Andrew D., Fleming, Paul R., Gao, Ning, Hajec, Laurel I., Hu, Jun, Laganas, Valerie A., McKinney, David C., McLeod, Sarah M., Prince, D.Bryan, Shapiro, Adam B., Buurman, Ed T.
Published in The Journal of biological chemistry (01.08.2014)
Published in The Journal of biological chemistry (01.08.2014)
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Negishi cross-coupling enabled synthesis of novel NAD+-dependent DNA ligase inhibitors and SAR development
Murphy-Benenato, Kerry E., Gingipalli, Lakshmaiah, Boriack-Sjodin, P. Ann, Martinez-Botella, Gabriel, Carcanague, Dan, Eyermann, Charles J., Gowravaram, Madhu, Harang, Jenna, Hale, Michael R., Ioannidis, Georgine, Jahic, Harris, Johnstone, Michele, Kutschke, Amy, Laganas, Valerie A., Loch, James T., Miller, Matthew D., Oguto, Herbert, Patel, Sahil Joe
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
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Antimicrobial Activity of Adenine-Based Inhibitors of NAD+-Dependent DNA Ligase
Buurman, Ed T, Laganas, Valerie A, Liu, Ce Feng, Manchester, John I
Published in ACS medicinal chemistry letters (09.08.2012)
Published in ACS medicinal chemistry letters (09.08.2012)
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From fragments to leads: novel bacterial NAD+-dependent DNA ligase inhibitors
Hale, Michael R., Brassington, Claire, Carcanague, Dan, Embrey, Kevin, Eyermann, Charles J., Giacobbe, Robert A., Gingipalli, Lakshmaiah, Gowravaram, Madhusudhan, Harang, Jenna, Howard, Tina, Ioannidis, Georgine, Jahic, Haris, Kutschke, Amy, Laganas, Valerie A., Loch, James, Miller, Matthew D., Murphy-Benenato, Kerry E., Oguto, Herbert, Otterbein, Ludovic, Patel, Sahil Joe, Shapiro, Adam B., Boriack-Sjodin, P. Ann
Published in Tetrahedron letters (03.06.2015)
Published in Tetrahedron letters (03.06.2015)
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