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Fader, Lee D., Bethell, Richard, Bonneau, Pierre, Bös, Michael, Bousquet, Yves, Cordingley, Michael G., Coulombe, René, Deroy, Patrick, Faucher, Anne-Marie, Gagnon, Alexandre, Goudreau, Nathalie, Grand-Maître, Chantal, Guse, Ingrid, Hucke, Oliver, Kawai, Stephen H., Lacoste, Jean-Eric, Landry, Serge, Lemke, Christopher T., Malenfant, Eric, Mason, Stephen, Morin, Sébastien, O’Meara, Jeff, Simoneau, Bruno, Titolo, Steve, Yoakim, Christiane
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Novel Inhibitor Binding Site Discovery on HIV‑1 Capsid N‑Terminal Domain by NMR and X‑ray Crystallography
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Published in ACS chemical biology (17.05.2013)
Published in ACS chemical biology (17.05.2013)
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Monitoring binding of HIV-1 capsid assembly inhibitors using (19)F ligand-and (15)N protein-based NMR and X-ray crystallography: early hit validation of a benzodiazepine series
Goudreau, Nathalie, Coulombe, René, Faucher, Anne-Marie, Grand-Maître, Chantal, Lacoste, Jean-Eric, Lemke, Christopher T, Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean-François, Titolo, Steve, Mason, Stephen W
Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series
Goudreau, Nathalie, Coulombe, René, Faucher, Anne-Marie, Grand-Maître, Chantal, Lacoste, Jean-Eric, Lemke, Christopher T., Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean-François, Titolo, Steve, Mason, Stephen W.
Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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Identification of benzofurano[3,2-d]pyrimidin-2-ones, a new series of HIV-1 nucleotide-competing reverse transcriptase inhibitors
Tremblay, Martin, Bethell, Richard C., Cordingley, Michael G., DeRoy, Patrick, Duan, Jianmin, Duplessis, Martin, Edwards, Paul J., Faucher, Anne-Marie, Halmos, Ted, James, Clint A., Kuhn, Cyrille, Lacoste, Jean-Éric, Lamorte, Louie, LaPlante, Steven R., Malenfant, Éric, Minville, Joannie, Morency, Louis, Morin, Sébastien, Rajotte, Daniel, Salois, Patrick, Simoneau, Bruno, Tremblay, Sonia, Sturino, Claudio F.
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
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Preparation of 2-alkenylperhydro-1,3-benzoxazines and application for 2-isoxazolines synthesis
Poisson, Carl, Lacoste, Jean-Éric, Rochon, Fernande D., Breau, Livain
Published in Tetrahedron: asymmetry (04.11.2009)
Published in Tetrahedron: asymmetry (04.11.2009)
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2 IMIDAZOPYRIDAZINES USEFUL AS INHIBITORS OF THE PAR-2 SIGNALING PATHWAY
FOURNIER PIERRE ANDRE, FARMER LUC J, LACOSTE JEAN ERIC, LESSARD STEPHANIE, BUBENIK MONICA, STURINO CLAUDIO, LIU BINGCAN, VALLEE FREDERIC, RAMTOHUL YEEMAN, SZYCHOWSKI JANEK, YANNOPOULOS CONSTANTIN, ST ONGE MIGUEL, MARTEL JULIEN, SAYEGH CAMIL ELIE
Year of Publication 27.05.2016
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Year of Publication 27.05.2016
Patent
INHIBITORS OF HIV REPLICATION
JAMES CLINT, DEROY PATRICK, HALMOS TEDDY, MORENCY LOUIS, TREMBLAY MARTIN, LACOSTE JEAN ERIC, FAUCHER ANNE MARIE, STURINO CLAUDIO, DUPLESSIS MARTIN, YOAKIM CHRISTIANE, MALENFANT ERIC, MORIN SEBASTIEN, MINVILLE JOANNIE, EDWARDS PAUL J
Year of Publication 12.04.2012
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Year of Publication 12.04.2012
Patent
Inside Cover: Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series (ChemMedChem 3/2013)
Goudreau, Nathalie, Coulombe, René, Faucher, Anne‐Marie, Grand‐Maître, Chantal, Lacoste, Jean‐Eric, Lemke, Christopher T., Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean‐François, Titolo, Steve, Mason, Stephen W.
Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using super(19)F Ligand-and super(15)N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series
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Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series
Goudreau, Nathalie, Coulombe, René, Faucher, Anne‐Marie, Grand‐Maître, Chantal, Lacoste, Jean‐Eric, Lemke, Christopher T., Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean‐François, Titolo, Steve, Mason, Stephen W.
Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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Inside Cover: Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series (ChemMedChem 3/2013)
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Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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2-Vinyl- trans-octahydro-1,3-benzoxazine: Cyclization and 1,3-dipolar cycloaddition of nitrile oxides
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Published in Tetrahedron letters (10.12.1998)
Published in Tetrahedron letters (10.12.1998)
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Year of Publication 06.04.2023
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Year of Publication 06.04.2023
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Year of Publication 26.10.2022
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Year of Publication 26.10.2022
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Cycloalkyl-containing carboxylic acids and uses thereof
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Year of Publication 11.08.2022
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Year of Publication 11.08.2022
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CYCLOALKYL-CONTAINING CARBOXYLIC ACIDS AND USES THEREOF
MARTEL, JULIEN, DUCEPPE, JEAN-SIMON, GAGNON, LYNE, THIBODEAU, JEAN-FRANCOIS, LEBLOND, FRANCOIS, LACOSTE, JEAN-ERIC, ZACHARIE, BOULOS, DOYLE, CHRIS, GEERTS, LILIANNE
Year of Publication 24.06.2021
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Year of Publication 24.06.2021
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