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The discovery of potent and selective 4-aminothienopyridines as B-Raf kinase inhibitors
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The Effects of the Novel, Reversible Epidermal Growth Factor Receptor/ErbB-2 Tyrosine Kinase Inhibitor, GW2016, on the Growth of Human Normal and Tumor-derived Cell Lines in Vitro and in Vivo
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Knowledge-based design of 7-azaindoles as selective B-Raf inhibitors
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Published in Bioorganic & medicinal chemistry (15.08.2008)
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Oxindole-Based Inhibitors of Cyclin-Dependent Kinase 2 (CDK2): Design, Synthesis, Enzymatic Activities, and X-ray Crystallographic Analysis
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Published in Journal of medicinal chemistry (06.12.2001)
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Small molecule inhibitors of the class 1 receptor tyrosine kinase family
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Published in Current topics in medicinal chemistry (01.09.2002)
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RET Activation Inhibits Doxorubicin-induced Apoptosis in SK-N-MC Cells
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Published in Anticancer research (01.07.2008)
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Published in Science (American Association for the Advancement of Science) (05.01.2001)
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Published in Bioorganic & medicinal chemistry letters (15.08.2005)
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Synthesis and Antitumor Activity of Novel Water Soluble Derivatives of Camptothecin as Specific Inhibitors of Topoisomerase I
Luzzio, Michael J, Besterman, Jeffrey M, Emerson, David L, Evans, Michael G, Lackey, Karen, Leitner, Peter L, McIntyre, Gordon, Morton, Bradley, Myers, Peter L, Peel, Michael, Sisco, Jay M, Sternbach, Daniel D, Tong, Wei-Qin, Truesdale, Ann, Uehling, David E, Vuong, Alan, Yates, Julie
Published in Journal of medicinal chemistry (01.02.1995)
Published in Journal of medicinal chemistry (01.02.1995)
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A Unique Structure for Epidermal Growth Factor Receptor Bound to GW572016 (Lapatinib)
Wood, Edgar R., Truesdale, Anne T., McDonald, Octerloney B., Yuan, Derek, Hassell, Anne, Dickerson, Scott H., Ellis, Byron, Pennisi, Christopher, Horne, Earnest, Lackey, Karen, Alligood, Krystal J., Rusnak, David W., Gilmer, Tona M., Shewchuk, Lisa
Published in Cancer research (Chicago, Ill.) (15.09.2004)
Published in Cancer research (Chicago, Ill.) (15.09.2004)
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