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Published in Journal of the American Chemical Society (13.01.1999)
Published in Journal of the American Chemical Society (13.01.1999)
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Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. IV. Discovery of 1-[(4,6-Dimethyl-5-pyrimidinyl)carbonyl]- 4-[4-{2-methoxy-1(R)-4-(trifluoromethyl)phenyl}ethyl-3(S)-methyl-1-piperazinyl]- 4-methylpiperidine (Sch-417690/Sch-D), a Potent, Highly Selective, and Orally Bioavailable CCR5 Antagonist
Tagat, Jayaram R, McCombie, Stuart W, Nazareno, Dennis, Labroli, Marc A, Xiao, Yushi, Steensma, Ruo W, Strizki, Julie M, Baroudy, Bahige M, Cox, Kathleen, Lachowicz, Jean, Varty, Geoffrey, Watkins, Robert
Published in Journal of medicinal chemistry (06.05.2004)
Published in Journal of medicinal chemistry (06.05.2004)
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Discovery of potent wall teichoic acid early stage inhibitors
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Published in Bioorganic & medicinal chemistry letters (15.08.2016)
Published in Bioorganic & medicinal chemistry letters (15.08.2016)
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The identification of novel 5′-amino gemcitabine analogs as potent RRM1 inhibitors
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Published in Bioorganic & medicinal chemistry (01.04.2014)
Published in Bioorganic & medicinal chemistry (01.04.2014)
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10-Formyl-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid (10-formyl-ddacthf) : A potent cytotoxic agent acting by selective inhibition of human GAR Tfase and the de novo purine biosynthetic pathway
MARSILJE, Thomas H, LABROLI, Marc A, WILSON, Ian A, BEARDSLEY, G. Peter, BENKOVIC, Stephen J, BOGER, Dale L, HEDRICK, Michael P, QING JIN, DESHARNAIS, Joel, BAKER, Stephen J, GOOLJARSINGH, Lata T, RAMCHARAN, Joseph, TAVASSOLI, Ali, YAN ZHANG
Published in Bioorganic & medicinal chemistry (01.08.2002)
Published in Bioorganic & medicinal chemistry (01.08.2002)
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A convergent preparation of the CHK1 inhibitor MK-8776 (SCH 900776)
Labroli, Marc A., Dwyer, Michael P., Poker, Cory, Keertikar, Kerry M., Rossman, Randall, Guzi, Timothy J.
Published in Tetrahedron letters (15.06.2016)
Published in Tetrahedron letters (15.06.2016)
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ChemInform Abstract: Syntheses of 5′-Amino-2′,5′-dideoxy-2′,2′-difluorocytidine Derivatives as Novel Anticancer Nucleoside Analogues
Labroli, Marc A., Dwyer, Michael P., Shen, Ruichao, Popovici-Muller, Janeta, Pu, Qinglin, Richard, Judson, Rosner, Kristen, Paruch, Kamil, Guzi, Timothy J.
Published in ChemInform (24.06.2014)
Published in ChemInform (24.06.2014)
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Syntheses of 5′-amino-2′,5′-dideoxy-2′,2′-difluorocytidine derivatives as novel anticancer nucleoside analogs
Labroli, Marc A., Dwyer, Michael P., Shen, Ruichao, Popovici-Muller, Janeta, Pu, Qinglin, Richard, Judson, Rosner, Kristen, Paruch, Kamil, Guzi, Timothy J.
Published in Tetrahedron letters (15.01.2014)
Published in Tetrahedron letters (15.01.2014)
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Journal Article
Syntheses of 5'-amino-2',5'-dideoxy-2',2'-dif luorocytidine derivatives as novel anticancer nucleoside analogs
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Published in Tetrahedron letters (01.01.2014)
Published in Tetrahedron letters (01.01.2014)
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AMIDO-SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPES VIRUSES
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Year of Publication 29.11.2023
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Year of Publication 29.11.2023
Patent
Piperazine-based CCR5 antagonists as HIV-1 inhibitors. IV. Discovery of 1-[(4,6-dimethyl-5-pyrimidinyl)carbonyl]- 4-[4-[2-methoxy-1(R)-4-(trifluoromethyl)phenyl]ethyl-3(S)-methyl-1-piperazinyl]- 4-methylpiperidine (Sch-417690/Sch-D), a potent, highly selective, and orally bioavailable CCR5 antagonist
Tagat, Jayaram R, McCombie, Stuart W, Nazareno, Dennis, Labroli, Marc A, Xiao, Yushi, Steensma, Ruo W, Strizki, Julie M, Baroudy, Bahige M, Cox, Kathleen, Lachowicz, Jean, Varty, Geoffrey, Watkins, Robert
Published in Journal of medicinal chemistry (06.05.2004)
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Published in Journal of medicinal chemistry (06.05.2004)
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AMIDO-SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPES VIRUSES
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Year of Publication 16.03.2023
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Year of Publication 16.03.2023
Patent
AMIDO-SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPES VIRUSES
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Year of Publication 26.10.2022
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Year of Publication 26.10.2022
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OXAZOLIDINONES AS TARO INHIBITORS
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Year of Publication 13.12.2023
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Year of Publication 13.12.2023
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INHIBITORS OF MSBA AS ANTIBIOTICS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
LI, Sarah W, TONG, Ling, LABROLI, Marc A, ZHANG, Li-Kang, BALIBAR, Carl J, SKUDLAREK, Jason W, WANG, Hao, WU, Zhe, MITCHELL, Helen, BABAOGLU, Kerim, COOKE, Andrew J, FORSTER, Ashley, WU, Chengwei, RAHEEM, Izzat, BUEVICH, Alexei, HUNTER, David N, SHAW, Anthony W
Year of Publication 23.11.2023
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Year of Publication 23.11.2023
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INHIBITORS OF MSBA AS ANTIBIOTICS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
TONG, Ling, LABROLI, Marc A, ZHANG, Li-Kang, BALIBAR, Carl J, SKUDLAREK, Jason W, WANG, Hao, LIU, Jian, WU, Zhe, MITCHELL, Helen, BABAOGLU, Kerim, COOKE, Andrew J, FORSTER, Ashley, WU, Chengwei, RAHEEM, Izzat, BUEVICH, Alexei, SHAW, Anthony W
Year of Publication 23.11.2023
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Year of Publication 23.11.2023
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