Recent advances in the development of dual topoisomerase I and II inhibitors as anticancer drugs
Salerno, S, Da Settimo, F, Taliani, S, Simorini, F, La Motta, C, Fornaciari, G, Marini, A M
Published in Current medicinal chemistry (01.12.2010)
Published in Current medicinal chemistry (01.12.2010)
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Receptor tyrosine kinase kit and gastrointestinal stromal tumours: an overview
Sartini, S, Dario, B, Morelli, M, Da Settimo, F, La Motta, C
Published in Current medicinal chemistry (01.06.2011)
Published in Current medicinal chemistry (01.06.2011)
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Inhibition of Ocular Aldose Reductase by a New Benzofuroxane Derivative Ameliorates Rat Endotoxic Uveitis
Sartini, S., Novellino, Ettore, Gesualdo, C., Simonelli, Francesca, Rossi, S., D'Amico, Michele, La Motta, Concettina, Ferraraccio, Franca, Ferraro, B., Maione, Sabatino, Trotta, M. C., Maisto, R., Zippo, M. V., Di Filippo, Clara, Cosconati, Sandro
Published in Mediators of Inflammation (01.01.2014)
Published in Mediators of Inflammation (01.01.2014)
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Allosteric modulators for adenosine receptors: an alternative to the orthosteric ligands
La Motta, C, Sartini, S, Morelli, M, Taliani, S, Da Settimo, F
Published in Current topics in medicinal chemistry (01.07.2010)
Published in Current topics in medicinal chemistry (01.07.2010)
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Journal Article
Effects of the New Aldose Reductase Inhibitor Benzofuroxane Derivative BF-5m on High Glucose Induced Prolongation of Cardiac QT Interval and Increase of Coronary Perfusion Pressure
D'Amico, Michele, Rossi, Francesco, La Motta, Concettina, Sartini, S., Di Carluccio, N., Trotta, M. C., Maisto, R., Ferraro, B., Di Filippo, Clara, Ferraraccio, Franca
Published in Journal of Diabetes Research (01.01.2016)
Published in Journal of Diabetes Research (01.01.2016)
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Journal Article
[1,2,4]Triazino[4,3-a]benzimidazole Acetic Acid Derivatives: A New Class of Selective Aldose Reductase Inhibitors
Da Settimo, Federico, Primofiore, Giampaolo, Da Settimo, Antonio, La Motta, Concettina, Taliani, Sabrina, Simorini, Francesca, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Boldrini, Enrico
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
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Journal Article
3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: A New Class of Selective A1 Adenosine Receptor Antagonists
Da Settimo, Federico, Primofiore, Giampaolo, Taliani, Sabrina, Marini, Anna Maria, La Motta, Concettina, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Trincavelli, Letizia, Martini, Claudia
Published in Journal of medicinal chemistry (01.02.2001)
Published in Journal of medicinal chemistry (01.02.2001)
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Journal Article
Synthesis and biological activity of 1,4-dihydrobenzothiopyrano[4,3- c]pyrazole derivatives, novel pro-apoptotic mitochondrial targeted agents
Dalla Via, L., Marini, A.M., Salerno, S., La Motta, C., Condello, M., Arancia, G., Agostinelli, E., Toninello, A.
Published in Bioorganic & medicinal chemistry (2009)
Published in Bioorganic & medicinal chemistry (2009)
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Journal Article
Synthesis of pyrrolo[3,4- c]pyridine derivatives possessing an acid group and their in vitro and in vivo evaluation as aldose reductase inhibitors
Da Settimo, A, Primofiore, G, Da Settimo, F, Simorini, F, La Motta, C, Martinelli, A, Boldrini, E
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
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Journal Article
Nanostructured ultra-thin patches for ultrasound-modulated delivery of anti-restenotic drug
Vannozzi, Lorenzo, Ricotti, Leonardo, Filippeschi, Carlo, Sartini, Stefania, Coviello, Vito, Piazza, Vincenzo, Pingue, Pasqualantonio, La Motta, Concettina, Dario, Paolo, Menciassi, Arianna
Published in International journal of nanomedicine (01.01.2016)
Published in International journal of nanomedicine (01.01.2016)
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Journal Article
Novel, Highly Potent Adenosine Deaminase Inhibitors Containing the Pyrazolo[3,4-d]pyrimidine Ring System. Synthesis, Structure−Activity Relationships, and Molecular Modeling Studies
Da Settimo, Federico, Primofiore, Giampaolo, La Motta, Concettina, Taliani, Sabrina, Simorini, Francesca, Marini, Anna Maria, Mugnaini, Laura, Lavecchia, Antonio, Novellino, Ettore, Tuscano, Daniela, Martini, Claudia
Published in Journal of medicinal chemistry (11.08.2005)
Published in Journal of medicinal chemistry (11.08.2005)
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2-(Benzimidazol-2-yl)quinoxalines: A novel class of selective antagonists at human A(1) and A(3) adenosine receptors designed by 3D database searching
Novellino, E, Cosimelli, B, Ehlardo, M, Greco, G, Iadanza, M, Lavecchia, A, Rimoli, MG, Sala, A, Da Settimo, A, Primofiore, G, Da Settimo, F, Taliani, S, La Motta, C, Klotz, KN, Tuscano, D, Trincavelli, ML, Martini, C
Published in Journal of medicinal chemistry (29.12.2005)
Published in Journal of medicinal chemistry (29.12.2005)
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Journal Article
Naphtho[1,2-d]isothiazole Acetic Acid Derivatives as a Novel Class of Selective Aldose Reductase Inhibitors
Da Settimo, Federico, Primofiore, Giampaolo, La Motta, Concettina, Sartini, Stefania, Taliani, Sabrina, Simorini, Francesca, Marini, Anna Maria, Lavecchia, Antonio, Novellino, Ettore, Boldrini, Enrico
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
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Journal Article
Medicinal chemistry of indolylglyoxylamide TSPO high affinity ligands with anxiolytic-like effects
Simorini, Francesca, Marini, Anna Maria, Taliani, Sabrina, La Motta, Concettina, Salerno, Silvia, Pugliesi, Isabella, Da Settimo, Federico
Published in Current topics in medicinal chemistry (01.02.2012)
Published in Current topics in medicinal chemistry (01.02.2012)
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Journal Article
Spirohydantoin derivatives of thiopyrano[2,3- b]pyridin-4(4 H)-one as potent in vitro and in vivo aldose reductase inhibitors
Da Settimo, Federico, Primofiore, Giampaolo, La Motta, Concettina, Salerno, Silvia, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Laneri, Sonia, Boldrini, Enrico
Published in Bioorganic & medicinal chemistry (17.01.2005)
Published in Bioorganic & medicinal chemistry (17.01.2005)
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Journal Article
3-aryl[1,2,4]triazino[4,3-alpha]benzimidazol-4(10H)-ones: A new class of selective A(1) adenosine receptor antagonists
Da Settimo, F, Primofiore, G, Taliani, S, Marini, AM, La Motta, C, Novellino, E, Greco, G, Lavecchia, A, Trincavelli, L, Martini, C
Published in Journal of medicinal chemistry (01.02.2001)
Published in Journal of medicinal chemistry (01.02.2001)
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Journal Article
Refinement of the Benzodiazepine Receptor Site Topology by Structure−Activity Relationships of New N-(Heteroarylmethyl)indol-3-ylglyoxylamides
Primofiore, Giampaolo, Da Settimo, Federico, Marini, Anna Maria, Taliani, Sabrina, La Motta, Concettina, Simorini, Francesca, Novellino, Ettore, Greco, Giovanni, Cosimelli, Barbara, Ehlardo, Marina, Sala, Annalisa, Besnard, François, Montali, Marina, Martini, Claudia
Published in Journal of medicinal chemistry (20.04.2006)
Published in Journal of medicinal chemistry (20.04.2006)
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Journal Article
Novel, Highly Potent Aldose Reductase Inhibitors: Cyano(2-oxo-2,3-dihydroindol-3-yl)acetic Acid Derivatives
Da Settimo, Federico, Primofiore, Giampaolo, Da Settimo, Antonio, La Motta, Concettina, Simorini, Francesca, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Boldrini, Enrico
Published in Journal of medicinal chemistry (10.04.2003)
Published in Journal of medicinal chemistry (10.04.2003)
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Journal Article
New Fluorescent 2-Phenylindolglyoxylamide Derivatives as Probes Targeting the Peripheral-Type Benzodiazepine Receptor: Design, Synthesis, and Biological Evaluation
Taliani, Sabrina, Simorini, Francesca, Sergianni, Valentina, La Motta, Concettina, Da Settimo, Federico, Cosimelli, Barbara, Abignente, Enrico, Greco, Giovanni, Novellino, Ettore, Rossi, Leonardo, Gremigni, Vittorio, Spinetti, Francesca, Chelli, Beatrice, Martini, Claudia
Published in Journal of medicinal chemistry (25.01.2007)
Published in Journal of medicinal chemistry (25.01.2007)
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