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Published in Journal of the American Chemical Society (12.02.2020)
Published in Journal of the American Chemical Society (12.02.2020)
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Discovery of orally active pyrrolopyridine- and aminopyridine-based Met kinase inhibitors
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Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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Photocatalytic Dearomative Intermolecular [2+2] Cycloaddition of Heterocycles for Building Molecular Complexity
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Published in Journal of organic chemistry (15.01.2021)
Published in Journal of organic chemistry (15.01.2021)
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Direct displacement of –OH by nucleophiles in hydroxymethylimidazoles
Macor, John E, Cornelius, Lyndon A.M, Roberge, Jacques Y
Published in Tetrahedron letters (15.04.2000)
Published in Tetrahedron letters (15.04.2000)
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Synthesis of 1‑(tert-Butyl) 4‑Methyl (1R,2S,4R)‑2-Methylcyclohexane-1,4-dicarboxylate from Hagemann’s tert-Butyl Ester for an Improved Synthesis of BMS-986251
Cornelius, Lyndon A. M, Li, Jianqing, Smith, Daniel, Krishnananthan, Subramaniam, Yip, Shiuhang, Wu, Dauh-Rurng, Pawluczyk, Joseph, Aulakh, Darpandeep, Sarjeant, Amy A, Kempson, James, Tino, Joseph A, Mathur, Arvind, Murali Dhar, T. G, Cherney, Robert J
Published in Journal of organic chemistry (21.08.2020)
Published in Journal of organic chemistry (21.08.2020)
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Discovery of N-(2-Chloro-6-methyl- phenyl)-2-(6-(4-(2-hydroxyethyl)- piperazin-1-yl)-2-methylpyrimidin-4- ylamino)thiazole-5-carboxamide (BMS-354825), a Dual Src/Abl Kinase Inhibitor with Potent Antitumor Activity in Preclinical Assays
Lombardo, Louis J, Lee, Francis Y, Chen, Ping, Norris, Derek, Barrish, Joel C, Behnia, Kamelia, Castaneda, Stephen, Cornelius, Lyndon A. M, Das, Jagabandhu, Doweyko, Arthur M, Fairchild, Craig, Hunt, John T, Inigo, Ivan, Johnston, Kathy, Kamath, Amrita, Kan, David, Klei, Herbert, Marathe, Punit, Pang, Suhong, Peterson, Russell, Pitt, Sidney, Schieven, Gary L, Schmidt, Robert J, Tokarski, John, Wen, Mei-Li, Wityak, John, Borzilleri, Robert M
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
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Discovery of N-(4-(2-Amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide (BMS-777607), a Selective and Orally Efficacious Inhibitor of the Met Kinase Superfamily
Schroeder, Gretchen M, An, Yongmi, Cai, Zhen-Wei, Chen, Xiao-Tao, Clark, Cheryl, Cornelius, Lyndon A. M, Dai, Jun, Gullo-Brown, Johnni, Gupta, Ashok, Henley, Benjamin, Hunt, John T, Jeyaseelan, Robert, Kamath, Amrita, Kim, Kyoung, Lippy, Jonathan, Lombardo, Louis J, Manne, Veeraswamy, Oppenheimer, Simone, Sack, John S, Schmidt, Robert J, Shen, Guoxiang, Stefanski, Kevin, Tokarski, John S, Trainor, George L, Wautlet, Barri S, Wei, Donna, Williams, David K, Zhang, Yingru, Zhang, Yueping, Fargnoli, Joseph, Borzilleri, Robert M
Published in Journal of medicinal chemistry (12.03.2009)
Published in Journal of medicinal chemistry (12.03.2009)
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Discovery of BMS-986251: A Clinically Viable, Potent, and Selective ROR gamma t Inverse Agonist
Cherney, Robert J., Cornelius, Lyndon A. M., Srivastava, Anurag, Weigelt, Carolyn A., Marcoux, David, Duan, James J-W, Shi, Qing, Batt, Douglas G., Liu, Qingjie, Yip, Shiuhang, Wu, Dauh-Rurng, Ruzanov, Max, Sack, John, Khan, Javed, Wang, Jinhong, Yarde, Melissa, Cvijic, Mary Ellen, Mathur, Arvind, Li, Sha, Shuster, David, Khandelwal, Purnima, Borowski, Virna, Xie, Jenny, Obermeier, Mary, Fura, Aberra, Stefanski, Kevin, Cornelius, Georgia, Tino, Joseph A., Macor, John E., Salter-Cid, Luisa, Denton, Rex, Zhao, Qihong, Carter, Percy H., Dhar, T. G. Murali
Published in ACS medicinal chemistry letters (11.06.2020)
Published in ACS medicinal chemistry letters (11.06.2020)
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Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitors
Qin, Lan-Ying, Ruan, Zheming, Cherney, Robert J., Dhar, T.G. Murali, Neels, James, Weigelt, Carolyn A., Sack, John S., Srivastava, Anurag S., Cornelius, Lyndon A.M., Tino, Joseph A., Stefanski, Kevin, Gu, Xiaomei, Xie, Jenny, Susulic, Vojkan, Yang, Xiaoxia, Yarde-Chinn, Melissa, Skala, Stacey, Bosnius, Ruth, Goldstein, Christine, Davies, Paul, Ruepp, Stefan, Salter-Cid, Luisa, Bhide, Rajeev S., Poss, Michael A.
Published in Bioorganic & medicinal chemistry letters (15.02.2017)
Published in Bioorganic & medicinal chemistry letters (15.02.2017)
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TRICYCLIC SULFONES AS ROR? MODULATORS
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Year of Publication 12.05.2022
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Year of Publication 07.03.2023
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Year of Publication 07.03.2023
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Nonsteroidal Progesterone Receptor Ligands. 2. High-Affinity Ligands with Selectivity for Bone Cell Progesterone Receptors
Combs, Donald W, Reese, Kimberly, Cornelius, Lyndon A. M, Gunnet, Joseph W, Cryan, Ellen V, Granger, Kay S, Jordan, Jerold J, Demarest, Keith T
Published in Journal of medicinal chemistry (01.12.1995)
Published in Journal of medicinal chemistry (01.12.1995)
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HETEROCYCLIC SULFONES AS ROR GAMMA MODULATORS
Dhar, T.G. Murali, Xiao, Hai-Yun, Cornelius, Lyndon A.M, Li, Jianqing, Cherney, Robert J, Qin, Lan-ying, LIU, Qingjie
Year of Publication 03.10.2019
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Year of Publication 03.10.2019
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Year of Publication 28.07.2021
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Year of Publication 28.07.2021
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CORNELIUS, Lyndon A.M, SHI, Qing, WEIGELT, Carolyn A, BATT, Douglas G, CHERNEY, Robert J, DHAR, T.G. Murali, MARCOUX, David, DUAN, Jingwu, BEAUDOIN BERTRAND, Myra, LIU, Qingjie, SRIVASTAVA, Anurag S
Year of Publication 17.03.2021
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Year of Publication 17.03.2021
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HETEROCYCLIC SULFONES AS ROR GAMMA MODULATORS
CORNELIUS, Lyndon A.M, CHERNEY, Robert, J, QIN, Lan-ying, DHAR, T.G. Murali, XIAO, Hai-Yun, LIU, Qingjie, LI, Jianqing
Year of Publication 21.08.2019
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Year of Publication 21.08.2019
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