Therapeutic efficacy of the small molecule GS-5734 against Ebola virus in rhesus monkeys
Warren, Travis K, Jordan, Robert, Lo, Michael K, Ray, Adrian S, Mackman, Richard L, Soloveva, Veronica, Siegel, Dustin, Perron, Michel, Bannister, Roy, Hui, Hon C, Larson, Nate, Strickley, Robert, Wells, Jay, Stuthman, Kelly S, Van Tongeren, Sean A, Garza, Nicole L, Donnelly, Ginger, Shurtleff, Amy C, Retterer, Cary J, Gharaibeh, Dima, Zamani, Rouzbeh, Kenny, Tara, Eaton, Brett P, Grimes, Elizabeth, Welch, Lisa S, Gomba, Laura, Wilhelmsen, Catherine L, Nichols, Donald K, Nuss, Jonathan E, Nagle, Elyse R, Kugelman, Jeffrey R, Palacios, Gustavo, Doerffler, Edward, Neville, Sean, Carra, Ernest, Clarke, Michael O, Zhang, Lijun, Lew, Willard, Ross, Bruce, Wang, Queenie, Chun, Kwon, Wolfe, Lydia, Babusis, Darius, Park, Yeojin, Stray, Kirsten M, Trancheva, Iva, Feng, Joy Y, Barauskas, Ona, Xu, Yili, Wong, Pamela, Braun, Molly R, Flint, Mike, McMullan, Laura K, Chen, Shan-Shan, Fearns, Rachel, Swaminathan, Swami, Mayers, Douglas L, Spiropoulou, Christina F, Lee, William A, Nichol, Stuart T, Cihlar, Tomas, Bavari, Sina
Published in Nature (London) (17.03.2016)
Published in Nature (London) (17.03.2016)
Get full text
Journal Article
Discovery and Synthesis of a Phosphoramidate Prodrug of a Pyrrolo[2,1‑f][triazin-4-amino] Adenine C‑Nucleoside (GS-5734) for the Treatment of Ebola and Emerging Viruses
Siegel, Dustin, Hui, Hon C, Doerffler, Edward, Clarke, Michael O, Chun, Kwon, Zhang, Lijun, Neville, Sean, Carra, Ernest, Lew, Willard, Ross, Bruce, Wang, Queenie, Wolfe, Lydia, Jordan, Robert, Soloveva, Veronica, Knox, John, Perry, Jason, Perron, Michel, Stray, Kirsten M, Barauskas, Ona, Feng, Joy Y, Xu, Yili, Lee, Gary, Rheingold, Arnold L, Ray, Adrian S, Bannister, Roy, Strickley, Robert, Swaminathan, Swami, Lee, William A, Bavari, Sina, Cihlar, Tomas, Lo, Michael K, Warren, Travis K, Mackman, Richard L
Published in Journal of Medicinal Chemistry (09.03.2017)
Published in Journal of Medicinal Chemistry (09.03.2017)
Get full text
Journal Article
Web Resource
Development of a Scalable Lanthanide Halide/Quaternary Ammonium Salt System for the Nucleophilic Addition of Grignard Reagents to Carbonyl Groups and Application to the Synthesis of a Remdesivir Intermediate
Stevens, Andrew C, Brak, Katrien, Bremner, W. Stacy, Brown, Angela M, Chtchemelinine, Andrei, Heumann, Lars, Kerschen, James A, Subotkowski, Witold, Vieira, Tiago, Wolfe, Lydia C, Xu, Boran, Yu, Chia-Yun
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
Get full text
Journal Article
Nickel or Phenanthroline Mediated Intramolecular Arylation of sp3 C–H Bonds Using Aryl Halides
Wertjes, William C, Wolfe, Lydia C, Waller, Peter J, Kalyani, Dipannita
Published in Organic letters (06.12.2013)
Published in Organic letters (06.12.2013)
Get full text
Journal Article
Discovery and Synthesis of a Phosphoramidate Prodrug of a Pyrrolo(2,1-f][triazin-4-amino] Adenine C-Nucleoside (GS-5734) for the Treatment of Ebola and Emerging Viruses
Siegel, Dustin, Hui, Hon C., Doerffler, Edward, Clarke, Michael O., Chun, Kwon, Zhang, Lijun, Neville, Sean, Carra, Ernest, Lew, Willard, Ross, Bruce, Wang, Queenie, Wolfe, Lydia, Jordan, Robert, Soloveva, Veronica, Knox, John, Perry, Jason, Perron, Michel, Stray, Kirsten M., Barauskas, Ona, Feng, Joy Y., Xu, Yili, Lee, Gary, Rheingold, Arnold L., Ray, Adrian S., Bannister, Roy, Strickley, Robert, Swaminathan, Swami, Lee, William A., Bavari, Sina, Cihlar, Tomas, Lo, Michael K., Warren, Travis K., Mackman, Richard L.
Published in Journal of medicinal chemistry (09.03.2017)
Published in Journal of medicinal chemistry (09.03.2017)
Get full text
Journal Article
Nickel or Phenanthroline Mediated Intramolecular Arylation of sp(3) C-H Bonds Using Aryl Halides
Wertjes, William C., Wolfe, Lydia C., Waller, Peter J., Kalyani, Dipannita
Published in Organic letters (06.12.2013)
Published in Organic letters (06.12.2013)
Get full text
Journal Article
Nickel or Phenanthroline Mediated Intramolecular Arylation of sp 3 C–H Bonds Using Aryl Halides
Wertjes, William C., Wolfe, Lydia C., Waller, Peter J., Kalyani, Dipannita
Published in Organic letters (06.12.2013)
Published in Organic letters (06.12.2013)
Get full text
Journal Article
METHODS FOR PREPARING RIBOSIDES
WANG XIANGHONG, ERICK RUEDEN, WILLARD LEW, MORIN MAE FRICK, TIAGO VIEIRA, ROBERT WILLIAM SCOTT, LYDIA WOLFE, BRITTANIE HOANG, GAO DETIAN, ANDREW C STEVENS, ANDREI CHTELININE, ANDREW W WALTMAN, YU CHIA-YUN, SILVIO CAMPAGNA, DUSTIN SIEGEL, STEVEN DONALD AXT, BRUCE ROSS, LARS V HEUMANN, KATRIEN BRAK, ROBERT RONALD MILBURN, PAVEL ROBERTOVICH BADALOV, MARK CHARLES WHITCOMB, EDWARD DOERFFLER, CLARISSA TADEUS, SEAN TIMOTHY NEVILLE
Year of Publication 25.06.2020
Get full text
Year of Publication 25.06.2020
Patent
METHODS FOR PREPARATION OF RIBOSIDES
WANG XIANGHONG, ERICK RUEDEN, WILLARD LEW, MORIN MAE FRICK, TIAGO VIEIRA, ROBERT WILLIAM SCOTT, LYDIA WOLFE, BRITTANIE HOANG, GAO DETIAN, ANDREW C STEVENS, ANDREI CHTELININE, ANDREW W WALTMAN, YU CHIA-YUN, SILVIO CAMPAGNA, DUSTIN SIEGEL, STEVEN DONALD AXT, BRUCE ROSS, LARS V HEUMANN, KATRIEN BRAK, ROBERT RONALD MILBURN, PAVEL ROBERTOVICH BADALOV, MARK CHARLES WHITCOMB, EDWARD DOERFFLER, CLARISSA TADEUS, SEAN TIMOTHY NEVILLE
Year of Publication 28.03.2019
Get full text
Year of Publication 28.03.2019
Patent
METHODS FOR PREPARATION OF RIBOSIDES
WANG XIANGHONG, ERICK RUEDEN, WILLARD LEW, MORIN MAE FRICK, TIAGO VIEIRA, ROBERT WILLIAM SCOTT, LYDIA WOLFE, BRITTANIE HOANG, GAO DETIAN, ANDREW C STEVENS, ANDREI CHTELININE, ANDREW W WALTMAN, YU CHIA-YUN, SILVIO CAMPAGNA, DUSTIN SIEGEL, STEVEN DONALD AXT, BRUCE ROSS, LARS V HEUMANN, KATRIEN BRAK, ROBERT RONALD MILBURN, PAVEL ROBERTOVICH BADALOV, MARK CHARLES WHITCOMB, EDWARD DOERFFLER, CLARISSA TADEUS, SEAN TIMOTHY NEVILLE
Year of Publication 08.11.2018
Get full text
Year of Publication 08.11.2018
Patent
Methods for the preparation of ribosides
Campagna, Silvio, Waltman, Andrew W, Heumann, Lars V, Lew, Willard, Milburn, Robert Ronald, Rueden, Erick, Ross, Bruce, Tadeus, Clarissa, Wolfe, Lydia, Scott, Robert William, Axt, Steven Donald, Gao, Detian, Frick, Morin Mae, Doerffler, Edward, Chtchemelinine, Andrei, Wang, Xianghong, Brak, Katrien, Neville, Sean Timothy, Yu, Chia-Yun, Siegel, Dustin, Hoang, Brittanie, Badalov, Pavel Robertovich, Vieira, Tiago, Whitcomb, Mark Charles, Stevens, Andrew C
Year of Publication 18.05.2023
Get full text
Year of Publication 18.05.2023
Patent
METHODS FOR THE PREPARATION OF RIBOSIDES
ROSS, BRUCE, LEW, WILLARD, TADEUS, CLARISSA, CHTELININE, ANDREI, CAMPAGNA, SILVIO, GAO, DETIAN, VIEIRA, TIAGO, NEVILLE, SEAN TIMOTHY, WALTMAN, ANDREW W, SCOTT, ROBERT WILLIAM, BADALOV, PAVEL ROBERTOVICH, WANG, XIANGHONG, BRAK, KATRIEN, HEUMANN, LARS V, YU, CHIA-YUN, SIEGEL, DUSTIN, WOLFE, LYDIA, WHITCOMB, MARK CHARLES, DOERFFLER, EDWARD, HOANG, BRITTANIE, STEVENS, ANDREW C, AXT, STEVEN DONALD, MILBURN, ROBERT RONALD, RUEDEN, ERIK, FRICK, MORIN MAE
Year of Publication 04.04.2023
Get full text
Year of Publication 04.04.2023
Patent
Methods for the preparation of ribosides
Campagna, Silvio, Waltman, Andrew W, Heumann, Lars V, Lew, Willard, Milburn, Robert Ronald, Rueden, Erick, Ross, Bruce, Tadeus, Clarissa, Wolfe, Lydia, Scott, Robert William, Axt, Steven Donald, Gao, Detian, Frick, Morin Mae, Doerffler, Edward, Chtchemelinine, Andrei, Wang, Xianghong, Brak, Katrien, Neville, Sean Timothy, Yu, Chia-Yun, Siegel, Dustin, Hoang, Brittanie, Badalov, Pavel Robertovich, Vieira, Tiago, Whitcomb, Mark Charles, Stevens, Andrew C
Year of Publication 02.02.2023
Get full text
Year of Publication 02.02.2023
Patent
METHODS FOR THE PREPARATION OF RIBOSIDES
Campagna, Silvio, Waltman, Andrew W, Heumann, Lars V, Lew, Willard, Milburn, Robert Ronald, Ross, Bruce, Tadeus, Clarissa, Wolfe, Lydia, Scott, Robert William, Axt, Steven Donald, Gao, Detian, Frick, Morin Mae, Doerffler, Edward, Chtchemelinine, Andrei, Wang, Xianghong, Brak, Katrien, Neville, Sean Timothy, Yu, Chia-Yun, Siegel, Dustin, Hoang, Brittanie, Badalov, Pavel Robertovich, Rueden, Erik, Vieira, Tiago, Whitcomb, Mark Charles, Stevens, Andrew C
Year of Publication 10.11.2022
Get full text
Year of Publication 10.11.2022
Patent
METHODS FOR THE PREPARATION OF RIBOSIDES
FRICK, Morin Mae, GAO, Detian, BRAK, Katrien, HEUMANN, Lars V, MILBURN, Robert Ronald, NEVILLE, Sean Timothy, TADEUS, Clarissa, VIERA, Tiago, YU, Chia-Yun, STEVENS, Andrew C, CAMPAGNA, Silvio, CHTELININE, Andrei, ROSS, Bruce, HOANG, Brittanie, RUEDEN, Erick, SCOTT, Robert William, AXT, Steven Donald, WHITCOMB, Mark Charles, SIEGEL, Dustin, BADALOV, Pavel Robertovich, WOLFE, Lydia, DOERFFLER, Edward, LEW, Willard, WANG, Xianghong, WALTMAN, Andrew W
Year of Publication 03.08.2022
Get full text
Year of Publication 03.08.2022
Patent
Methods for the preparation of ribosides
Campagna, Silvio, Waltman, Andrew W, Heumann, Lars V, Lew, Willard, Milburn, Robert Ronald, Ross, Bruce, Tadeus, Clarissa, Wolfe, Lydia, Scott, Robert William, Axt, Steven Donald, Gao, Detian, Frick, Morin Mae, Doerffler, Edward, Chtchemelinine, Andrei, Wang, Xianghong, Brak, Katrien, Neville, Sean Timothy, Yu, Chia-Yun, Siegel, Dustin, Hoang, Brittanie, Badalov, Pavel Robertovich, Rueden, Erik, Vieira, Tiago, Whitcomb, Mark Charles, Stevens, Andrew C
Year of Publication 31.05.2022
Get full text
Year of Publication 31.05.2022
Patent
METHODS FOR THE PREPARATION OF RIBOSIDES
ROSS, BRUCE, LEW, WILLARD, TADEUS, CLARISSA, CHTELININE, ANDREI, CAMPAGNA, SILVIO, GAO, DETIAN, VIEIRA, TIAGO, NEVILLE, SEAN TIMOTHY, WALTMAN, ANDREW W, SCOTT, ROBERT WILLIAM, BADALOV, PAVEL ROBERTOVICH, WANG, XIANGHONG, BRAK, KATRIEN, HEUMANN, LARS V, YU, CHIA-YUN, SIEGEL, DUSTIN, RUEDEN, ERICK, WOLFE, LYDIA, WHITCOMB, MARK CHARLES, DOERFFLER, EDWARD, HOANG, BRITTANIE, STEVENS, ANDREW C, AXT, STEVEN DONALD, MILBURN, ROBERT RONALD, FRICK, MORIN MAE
Year of Publication 28.02.2022
Get full text
Year of Publication 28.02.2022
Patent
METHODS FOR THE PREPARATION OF RIBOSIDES
VIEIRA Tiago, GAO Detian, NEVILLE Sean Timothy, SCOTT Robert William, STEVENS Andrew C, WALTMAN Andrew W, AXT Steven Donald, DOERFFLER Edward, MILBURN Robert Ronald, CAMPAGNA Silvio, SIEGEL Dustin, ROSS Bruce, TADEUS Clarissa, RUEDEN Erick, YU Chia-Yun, FRICK Morin Mae, CHTELININE Andrei, HOANG Brittanie, BADALOV Pavel Robertovich, WOLFE Lydia, WANG Xianghong, HEUMANN Lars V, BRAK Katrien, WHITCOMB Mark Charles, LEW Willard
Year of Publication 31.01.2022
Get full text
Year of Publication 31.01.2022
Patent