Phase I Study of TLK286 (Glutathione S-Transferase P1-1 Activated Glutathione Analogue) in Advanced Refractory Solid Malignancies
ROSEN, Lee S, BROWN, Joseph, MASCAVAGE, Julie C, DOMBROSKI, Jacqueline A, GOMEZ, Reinaldo F, BROWN, Gail L, LAXA, Bernadette, BOULOS, Leny, REISWIG, Laura, HENNER, William D, LUM, Robert T, SCHOW, Steve R, MAACK, Christopher A, KECK, James G
Published in Clinical cancer research (01.05.2003)
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Published in Clinical cancer research (01.05.2003)
Journal Article
A Novel Small Molecule That Directly Sensitizes the Insulin Receptor In Vitro and In Vivo
VARA PRASAD MANCHEM, GOLDFINE, Ira D, VILLAR, Hugo O, WICK, Michael M, KOZLOWSKI, Michael R, KOHANSKI, Ronald A, CRISTOBAL, Cristina P, LUM, Robert T, SCHOW, Steven R, SHI, Songyuan, SPEVAK, Wayne R, LABORDE, Edgardo, TOAVS, Deborah K
Published in Diabetes (New York, N.Y.) (01.04.2001)
Published in Diabetes (New York, N.Y.) (01.04.2001)
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Journal Article
Design, Synthesis, and Structure−Activity Relationships of Novel Insulin Receptor Tyrosine Kinase Activators
Lum, Robert T, Cheng, Mingshan, Cristobal, Cristina P, Goldfine, Ira D, Evans, Joseph L, Keck, James G, Macsata, Robert W, Manchem, Vara Prasad, Matsumoto, Yukiharu, Park, Sophia J, Rao, Sandhya S, Robinson, Louise, Shi, Songyuan, Spevak, Wayne R, Schow, Steven R
Published in Journal of medicinal chemistry (09.10.2008)
Published in Journal of medicinal chemistry (09.10.2008)
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Journal Article
Synthesis, structure, and reactions of a zirconocene-cyclohexyne complex
Buchwald, Stephen L, Lum, Robert T, Dewan, John C
Published in Journal of the American Chemical Society (01.11.1986)
Published in Journal of the American Chemical Society (01.11.1986)
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Journal Article
A general method for the preparation of zirconocene complexes of substituted benzynes: in situ generation, coupling reactions, and use in the synthesis of polyfunctionalized aromatic compounds
Buchwald, Stephen L, Watson, Brett T, Lum, Robert T, Nugent, William A
Published in Journal of the American Chemical Society (01.11.1987)
Published in Journal of the American Chemical Society (01.11.1987)
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Journal Article
Target-related affinity profiling: Telik's lead discovery technology
Beroza, Paul, Damodaran, Komath, Lum, Robert T
Published in Current topics in medicinal chemistry (01.01.2005)
Published in Current topics in medicinal chemistry (01.01.2005)
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Journal Article
5-Substituted isophthalamides as insulin receptor sensitizers
Robinson, Louise, Bajjalieh, Sonia, Cairns, Nicholas, Lum, Robert T., Macsata, Robert W., Manchem, Vara Prasad, Park, Sophia J., Rao, Sandhya, Schow, Steven R., Shi, Songyuan, Spevak, Wayne R.
Published in Bioorganic & medicinal chemistry (15.06.2008)
Published in Bioorganic & medicinal chemistry (15.06.2008)
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Journal Article
In vitro and in vivo prevention of HIV protease inhibitor-induced insulin resistance by a novel small molecule insulin receptor activator
Cheng, Mingshan, Chen, Seiyu, Schow, Steven R., Manchem, Vara Prasad, Spevak, Wayne R., Cristobal, Cristina P., Shi, Songyuan, Macsata, Robert W., Lum, Robert T., Goldfine, Ira D., Keck, James G.
Published in Journal of cellular biochemistry (15.08.2004)
Published in Journal of cellular biochemistry (15.08.2004)
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Journal Article
Synthesis and Biological Evaluation of the Enantiomers of the Potent and Selective A1-Adenosine Antagonist 1,3-Dipropyl-8-[2-(5,6-epoxynorbonyl)]- xanthine
Pfister, Jürg R, Belardinelli, Luiz, Lee, Gavin, Lum, Robert T, Milner, Peter, Stanley, William C, Linden, Joel, Baker, Stephen P, Schreiner, George
Published in Journal of medicinal chemistry (06.06.1997)
Published in Journal of medicinal chemistry (06.06.1997)
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Journal Article
A New Structural Class of Proteasome Inhibitors that Prevent NF-κB Activation
Lum, Robert T, Kerwar, Suresh S, Meyer, Stephanie M, Nelson, Marek G, Schow, Steven R, Shiffman, Dov, Wick, Michael M, Joly, Alison
Published in Biochemical pharmacology (01.05.1998)
Published in Biochemical pharmacology (01.05.1998)
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Journal Article
Novel Cyclooxygenase-1 Inhibitors Discovered Using Affinity Fingerprints
Hsu, Nancy, Cai, Danying, Damodaran, Komath, Gomez, Reinaldo F, Keck, James G, Laborde, Edgardo, Lum, Robert T, Macke, Thomas J, Martin, Graeme, Schow, Steven R, Simon, Reyna J, Villar, Hugo O, Wick, Michael M, Beroza, Paul
Published in Journal of medicinal chemistry (23.09.2004)
Published in Journal of medicinal chemistry (23.09.2004)
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Journal Article
Selective inhibition of the chymotrypsin-like activity of the 20S proteasome by 5-methoxy-1-indanone dipeptide benzamides
Lum, Robert T., Nelson, Marek G., Joly, Alison, Horsma, Amy G., Lee, Gavin, Meyer, Stephanie M., Wick, Michael M., Schow, Steven R.
Published in Bioorganic & medicinal chemistry letters (03.02.1998)
Published in Bioorganic & medicinal chemistry letters (03.02.1998)
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Journal Article
Synthesis and antiviral activity of a novel class of HIV-1 protease inhibitors containing a heterocyclic P1′-P2′ amide bond isostere
Thompson, Scott K., Eppley, Alecia M., Frazee, James S., Darcy, Michael G., Lum, Robert T., Tomaszek, Thaddeus A., Ivanoff, Lucinda A., Morris, Jane F., Sternberg, Edmund J., Lambert, Dennis M., Fernandez, Annabellee V., Petteway, Stephen R., Meek, Thomas D, Metcalf, Brian W., Gleason, John G.
Published in Bioorganic & medicinal chemistry letters (01.10.1994)
Published in Bioorganic & medicinal chemistry letters (01.10.1994)
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Journal Article
Oxygen-atom transfer from nitrous oxide. Synthesis and structure of a zirconocene oxametallacyclobutene complex
Vaughan, G. Alan, Hillhouse, Gregory L., Lum, Robert T., Buchwald, Stephen L., Rheingold, Arnold L.
Published in Journal of the American Chemical Society (01.10.1988)
Published in Journal of the American Chemical Society (01.10.1988)
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Journal Article
Synthesis and activity of 2,6,9-trisubstituted purines
Schow, Steven R., Mackman, Richard L., Blum, Cheri L., Brooks, Eric, Horsma, Amy G., Joly, Alison, Kerwar, Suresh S., Lee, Gavin, Shiffman, Dov, Nelson, Marek G., Wang, Xingbo, Wick, Michael M., Zhang, Xiaoming, Lum, Robert T.
Published in Bioorganic & medicinal chemistry letters (04.11.1997)
Published in Bioorganic & medicinal chemistry letters (04.11.1997)
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Journal Article