Reduction of myocardial infarction by calpain inhibitors A-705239 and A-705253 in isolated perfused rabbit hearts
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Published in Biological chemistry (01.11.2004)
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Potent and selective oxindole-based vasopressin 1b receptor antagonists with improved pharmacokinetic properties
Oost, Thorsten, Backfisch, Gisela, Bhowmik, Swati, van Gaalen, Marcel M., Geneste, Hervé, Hornberger, Wilfried, Lubisch, Wilfried, Netz, Astrid, Unger, Liliane, Wernet, Wolfgang
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Discovery and SAR of 2-(1-propylpiperidin-4-yl)-1H-benzimidazole-4-carboxamide: A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer
Penning, Thomas D, Zhu, Gui-Dong, Gandhi, Viraj B, Gong, Jianchun, Thomas, Sheela, Lubisch, Wilfried, Grandel, Roland, Wernet, Wolfgang, Park, Chang H, Fry, Elizabeth H, Liu, Xuesong, Shi, Yan, Klinghofer, Vered, Johnson, Eric F, Donawho, Cherrie K, Frost, David J, Bontcheva-Diaz, Velitchka, Bouska, Jennifer J, Olson, Amanda M, Marsh, Kennan C, Luo, Yan, Rosenberg, Saul H, Giranda, Vincent L
Published in Bioorganic & medicinal chemistry (15.07.2008)
Published in Bioorganic & medicinal chemistry (15.07.2008)
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CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS
SEEMANN DIETMAR, NIMMRICH VOLKER, MACK HELMUT, KLING ANDREAS, MOELLER ACHIM, HORNBERGER WILFRIED, LUBISCH WILFRIED
Year of Publication 05.08.2015
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Year of Publication 05.08.2015
Patent
CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS
SEEMANN DIETMAR, NIMMRICH VOLKER, MACK HELMUT, KLING ANDREAS, MOELLER ACHIM, HORNBERGER WILFRIED, LUBISCH WILFRIED
Year of Publication 05.08.2015
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Year of Publication 05.08.2015
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Benzoylalanine-Derived Ketoamides Carrying Vinylbenzyl Amino Residues: Discovery of Potent Water-Soluble Calpain Inhibitors with Oral Bioavailability
Lubisch, Wilfried, Beckenbach, Edith, Bopp, Sabina, Hofmann, Hans-Peter, Kartal, Arzu, Kästel, Claudia, Lindner, Tanja, Metz-Garrecht, Marion, Reeb, Jutta, Regner, Ferdinand, Vierling, Michael, Möller, Achim
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Synthesis and SAR of highly potent and selective dopamine D 3-receptor antagonists: Quinolin(di)one and benzazepin(di)one derivatives
Geneste, Hervé, Backfisch, Gisela, Braje, Wilfried, Delzer, Jürgen, Haupt, Andreas, Hutchins, Charles W., King, Linda L., Lubisch, Wilfried, Steiner, Gerd, Teschendorf, Hans-Jürgen, Unger, Liliane, Wernet, Wolfgang
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Discovery and SAR of 2-(1-propylpiperidin-4-yl)-1 H-benzimidazole-4-carboxamide: A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer
Penning, Thomas D., Zhu, Gui-Dong, Gandhi, Viraj B., Gong, Jianchun, Thomas, Sheela, Lubisch, Wilfried, Grandel, Roland, Wernet, Wolfgang, Park, Chang H., Fry, Elizabeth H., Liu, Xuesong, Shi, Yan, Klinghofer, Vered, Johnson, Eric F., Donawho, Cherrie K., Frost, David J., Bontcheva-Diaz, Velitchka, Bouska, Jennifer J., Olson, Amanda M., Marsh, Kennan C., Luo, Yan, Rosenberg, Saul H., Giranda, Vincent L.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Discovery and SAR of 2-(l-propylpiperidin-4-yl)-lH-benzimidazole-4-carboxamide : A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer
PENNING, Thomas D, ZHU, Gui-Dong, XUESONG LIU, YAN SHI, KLINGHOFER, Vered, JOHNSON, Eric F, DONAWHO, Cherrie K, FROST, David J, BONTCHEVA-DIAZ, Velitchka, BOUSKA, Jennifer J, OLSON, Amanda M, MARSH, Kennan C, GANDHI, Viraj B, YAN LUO, ROSENBERG, Saul H, GIRANDA, Vincent L, JIANCHUN GONG, THOMAS, Sheela, LUBISCH, Wilfried, GRANDEL, Roland, WERNET, Wolfgang, PARK, Chang H, FRY, Elizabeth H
Published in Bioorganic & medicinal chemistry (2008)
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Published in Bioorganic & medicinal chemistry (2008)
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Synthesis and SAR of highly potent and selective dopamine D(3)-receptor antagonists: Quinolin(di)one and benzazepin(di)one derivatives. herve.geneste@abbott.com
Geneste, Hervé, Backfisch, Gisela, Braje, Wilfried, Delzer, Jürgen, Haupt, Andreas, Hutchins, Charles W, King, Linda L, Lubisch, Wilfried, Steiner, Gerd, Teschendorf, Hans-Jürgen, Unger, Liliane, Wernet, Wolfgang
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Synthesis and SAR of highly potent and selective dopamine D3-receptor antagonists : Quinolin(di)one and benzazepin(di)one derivatives
GENESTE, Hervé, BACKFISCH, Gisela, UNGER, Liliane, WERNET, Wolfgang, BRAJE, Wilfried, DELZER, Jürgen, HAUPT, Andreas, HUTCHINS, Charles W, KING, Linda L, LUBISCH, Wilfried, STEINER, Gerd, TESCHENDORF, Hans-Jürgen
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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A Novel Water-Soluble and Cell-Permeable Calpain Inhibitor Protects Myocardial and Mitochondrial Function in Postischemic Reperfusion
Neuhof, C., Götte, O., Trumbeckaite, S., Attenberger, M., Kuzkaya, N., Gellerich, F., Möller, A., Lubisch, W., Speth, M., Tillmanns, H., Neuhof, H.
Published in Biological chemistry (01.12.2003)
Published in Biological chemistry (01.12.2003)
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