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Published in Biochemistry (Easton) (02.06.2009)
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Aminoethylenes: A Tetrahedral Intermediate Isostere Yielding Potent Inhibitors of the Aspartyl Protease BACE-1
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Published in Journal of medicinal chemistry (09.02.2006)
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Design and synthesis of 2-amino-pyrazolopyridines as Polo-like kinase 1 inhibitors
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A diaminocyclohexyl analog of SNS-032 with improved permeability and bioavailability properties
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Discovery of Dihydrobenzoxazepinone (GS-6615) Late Sodium Current Inhibitor (Late I Nai), a Phase II Agent with Demonstrated Preclinical Anti-Ischemic and Antiarrhythmic Properties
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Published in Journal of medicinal chemistry (13.10.2016)
Published in Journal of medicinal chemistry (13.10.2016)
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Discovery of Dihydrobenzoxazepinone (GS-6615) Late Sodium Current Inhibitor (Late I(Na)i), a Phase II Agent with Demonstrated Preclinical Anti-Ischemic and Antiarrhythmic Properties
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Published in Journal of medicinal chemistry (13.10.2016)
Published in Journal of medicinal chemistry (13.10.2016)
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compostos para o tratamento de dependência química
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