Biphenyl amide p38 kinase inhibitors 4: DFG-in and DFG-out binding modes
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Published in Bioorganic & medicinal chemistry (01.08.2008)
Published in Bioorganic & medicinal chemistry (01.08.2008)
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3,5-Disubstituted-indole-7-carboxamides: The discovery of a novel series of potent, selective inhibitors of IKK-β
Miller, David D., Bamborough, Paul, Christopher, John A., Baldwin, Ian R., Champigny, Aurelie C., Cutler, Geoffrey J., Kerns, Jeffrey K., Longstaff, Timothy, Mellor, Geoffrey W., Morey, James V., Morse, Mary A., Nie, Hong, Rumsey, William L., Taggart, John J.
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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3,5-Disubstituted-indole-7-carboxamides: The discovery of a novel series of potent, selective inhibitors of IIK-β
MILLER, David D, BAMBOROUGH, Paul, MORSE, Mary A, HONG NIE, RUMSEY, William L, TAGGART, John J, CHRISTOPHER, John A, BALDWIN, Ian R, CHAMPIGNY, Aurelie C, CUTLER, Geoffrey J, KERNS, Jeffrey K, LONGSTAFF, Timothy, MELLOR, Geoffrey W, MOREY, James V
Published in Bioorganic & medicinal chemistry letters (2011)
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Published in Bioorganic & medicinal chemistry letters (2011)
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Fused heteroaryl derivatives for use as P38 kinase inhibitors
DEBOECK NIGEL MARC, ANGELL RICHARD MARTYN, LONGSTAFF TIMOTHY, BAMBOROUGH PAUL, BALDWIN IAN ROBERT, SWANSON STEPHEN
Year of Publication 05.01.2010
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Year of Publication 05.01.2010
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Fused heteroaryl derivatives for use as P38 kinase inhibitors
Angell, Richard Martyn, Baldwin, Ian Robert, Bamborough, Paul, Deboeck, Nigel Marc, Longstaff, Timothy, Swanson, Stephen
Year of Publication 05.01.2010
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Year of Publication 05.01.2010
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INDOL-DERIVATE UND IHRE VERWENDUNG ALS KINASE- HEMMER, INSBESONDERE IKK2-HEMMER
CHRISTOPHER, JOHN, MILLER, DAVID, BALDWIN, IAN, BAMBOROUGH, PAUL, KERNS, JEFFREY, LONGSTAFF, TIMOTHY
Year of Publication 15.11.2008
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Year of Publication 15.11.2008
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