4-[3-(4-Cyclopropanecarbonylpiperazine-1-carbonyl)-4-fluorobenzyl]-2H-phthalazin-1-one: A Novel Bioavailable Inhibitor of Poly(ADP-ribose) Polymerase-1
Menear, Keith A, Adcock, Claire, Boulter, Robert, Cockcroft, Xiao-ling, Copsey, Louise, Cranston, Aaron, Dillon, Krystyna J, Drzewiecki, Jan, Garman, Sheila, Gomez, Sylvie, Javaid, Hashim, Kerrigan, Frank, Knights, Charlotte, Lau, Alan, Loh, Vincent M, Matthews, Ian T. W, Moore, Stephen, O’Connor, Mark J, Smith, Graeme C. M, Martin, Niall M. B
Published in Journal of medicinal chemistry (23.10.2008)
Published in Journal of medicinal chemistry (23.10.2008)
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Phthalazinones. Part 1: The design and synthesis of a novel series of potent inhibitors of poly(ADP-ribose)polymerase
Loh, Vincent M., Cockcroft, Xiao-ling, Dillon, Krystyna J., Dixon, Lesley, Drzewiecki, Jan, Eversley, Penny J., Gomez, Sylvie, Hoare, Janet, Kerrigan, Frank, Matthews, Ian T.W., Menear, Keith A., Martin, Niall M.B., Newton, Roger F., Paul, Jane, Smith, Graeme C.M., Vile, Julia, Whittle, Alan J.
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
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Phthalazinones 2: Optimisation and synthesis of novel potent inhibitors of poly(ADP-ribose)polymerase
Cockcroft, Xiao-ling, Dillon, Krystyna J., Dixon, Lesley, Drzewiecki, Jan, Kerrigan, Frank, Loh, Vincent M., Martin, Niall M.B., Menear, Keith A., Smith, Graeme C.M.
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Ftalazinonderivater, anvendelse derav samt farmasøytisk preparat omfattende en slik forbindelse
Cockcroft, Xiao-Ling Fan, Menear, Keith Allan, Matthews, Ian Timothy William, Martin, Niall Morrison Barr, Kerrigan, Frank, Smith, Graeme Cameron Murray, Loh Jr, Vincent M, Ashworth, Alan, Jackson, Stephen Philip
Year of Publication 10.04.2012
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Year of Publication 10.04.2012
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Phthalazinones 2: Optimization and Synthesis of Novel Potent Inhibitors of Poly(ADP-Ribose)polymerase
Cockcroft, Xiao-ling, Dillon, Krystyna J., Dixon, Lesley, Drzewiecki, Jan, Kerrigan, Frank, Loh, Vincent M. Jr, Martin, Niall M. B., Menear, Keith A., Smith, Graeme C. M.
Published in ChemInform (23.05.2006)
Published in ChemInform (23.05.2006)
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Ftalazinonderivater
SMITH GRAEME CAMERON MURRAY, MARTIN NIALL MORRISON BARR, JACKSON STEPHEN PHILIP, ASHWORTH ALAN, MENEAR KEITH ALLAN, KERRIGAN FRANK, MATTHEWS IAN TIMOTHY WILLIAM, LOH JR VINCENT M, COCKCROFT XIAO-LING FAN
Year of Publication 11.11.2005
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Year of Publication 11.11.2005
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