Rearrangement of 3,3-Disubstituted Indolenines and Synthesis of 2,3-Substituted Indoles
Liu, Kevin G, Robichaud, Albert J, Lo, Jennifer R, Mattes, James F, Cai, Yanxuan
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Published in Organic letters (07.12.2006)
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Identification of a series of benzoxazoles as potent 5-HT6 ligands
Liu, Kevin G, Lo, Jennifer R, Comery, Thomas A, Zhang, Guo Ming, Zhang, Jean Y, Kowal, Dianne M, Smith, Deborah L, Di, Li, Kerns, Edward H, Schechter, Lee E, Robichaud, Albert J
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Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Discovery of Lanraplenib (GS-9876): A Once-Daily Spleen Tyrosine Kinase Inhibitor for Autoimmune Diseases
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5-Piperazinyl-3-sulfonylindazoles as Potent and Selective 5-Hydroxytryptamine-6 Antagonists
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Published in Journal of medicinal chemistry (11.11.2010)
Published in Journal of medicinal chemistry (11.11.2010)
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Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT6 antagonists
Liu, Kevin G., Robichaud, Albert J., Greenfield, Alexander A., Lo, Jennifer R., Grosanu, Cristina, Mattes, James F., Cai, Yanxuan, Zhang, Guo Ming, Zhang, Jean Y., Kowal, Dianne M., Smith, Deborah L., Di, Li, Kerns, Edward H., Schechter, Lee E., Comery, Thomas A.
Published in Bioorganic & medicinal chemistry (01.01.2011)
Published in Bioorganic & medicinal chemistry (01.01.2011)
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A regiospecific synthesis of a series of 1-sulfonyl azepinoindoles as potent 5-HT6 ligands
LIU, Kevin G, LO, Jennifer R, ROBICHAUD, Albert J, COMERY, Thomas A, GUO MING ZHANG, ZHANG, Jean Y, KOWAL, Dianne M, SMITH, Deborah L, LI DI, KERNS, Edward H, SCHECHTER, Lee E
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
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Identification of a novel series of 3-piperidinyl-5-sulfonylindazoles as potent 5-HT 6 ligands
Liu, Kevin G., Lo, Jennifer R., Comery, Thomas A., Zhang, Guo Ming, Zhang, Jean Y., Kowal, Dianne M., Smith, Deborah L., Di, Li, Kerns, Edward H., Schechter, Lee E., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
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Journal Article
1-Sulfonylindazoles as potent and selective 5-HT6 ligands
LIU, Kevin G, LO, Jennifer R, ROBICHAUD, Albert J, COMERY, Thomas A, GUO MING ZHANG, ZHANG, Jean Y, KOWAL, Dianne M, SMITH, Deborah L, LI DI, KERNS, Edward H, SCHECHTER, Lee E
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Journal Article
Identification of a novel series of 3-piperidinyl-5-sulfonylindazoles as potent 5-HT6 ligands
LIU, Kevin G, LO, Jennifer R, ROBICHAUD, Albert J, COMERY, Thomas A, GUO MING ZHANG, ZHANG, Jean Y, KOWAL, Dianne M, SMITH, Deborah L, LI DI, KERNS, Edward H, SCHECHTER, Lee E
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
Published in Bioorganic & medicinal chemistry letters (15.06.2009)
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Journal Article
Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT sub(6) antagonists
Liu, Kevin G, Robichaud, Albert J, Greenfield, Alexander A, Lo, Jennifer R, Grosanu, Cristina, Mattes, James F, Cai, Yanxuan, Zhang, Guo Ming, Zhang, Jean Y, Kowal, Dianne M, Smith, Deborah L, Di, Li, Kerns, Edward H, Schechter, Lee E, Comery, Thomas A
Published in Bioorganic & medicinal chemistry (01.01.2011)
Published in Bioorganic & medicinal chemistry (01.01.2011)
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Journal Article
1-Sulfonylindazoles as potent and selective 5-HT 6 ligands
Liu, Kevin G., Lo, Jennifer R., Comery, Thomas A., Zhang, Guo Ming, Zhang, Jean Y., Kowal, Dianne M., Smith, Deborah L., Di, Li, Kerns, Edward H., Schechter, Lee E., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Journal Article
Identification of a series of benzoxazoles as potent 5-HT 6 ligands
Liu, Kevin G., Lo, Jennifer R., Comery, Thomas A., Zhang, Guo Ming, Zhang, Jean Y., Kowal, Dianne M., Smith, Deborah L., Di, Li, Kerns, Edward H., Schechter, Lee E., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Journal Article
A regiospecific synthesis of a series of 1-sulfonyl azepinoindoles as potent 5-HT sub(6) ligands
Liu, Kevin G, Lo, Jennifer R, Comery, Thomas A, Zhang, Guo Ming, Zhang, Jean Y, Kowal, Dianne M, Smith, Deborah L, Di, Li, Kerns, Edward H, Schechter, Lee E, Robichaud, Albert J
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
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Journal Article
A regiospecific synthesis of a series of 1-sulfonyl azepinoindoles as potent 5-HT 6 ligands
Liu, Kevin G., Lo, Jennifer R., Comery, Thomas A., Zhang, Guo Ming, Zhang, Jean Y., Kowal, Dianne M., Smith, Deborah L., Di, Li, Kerns, Edward H., Schechter, Lee E., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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Journal Article
Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT(6) antagonists
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Published in Bioorganic & medicinal chemistry (01.01.2011)
Published in Bioorganic & medicinal chemistry (01.01.2011)
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Year of Publication 29.08.2024
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CRYSTALLINE SUCCINATE SALT OF 6-(6-AMINOPYRAZIN-2-YL)-N-(4-(4-(OXETAN-3-YL)PIPERAZIN-1-YL)PHENYL)IMIDAZO[1,2-a]PYRAZIN-8-AMINE
Lo, Jennifer R, Blomgren, Peter A, Mitchell, Scott A, Lee, Seung H, Xu, Jianjun, Schmitt, Aaron C, Xiong, Jin-Ming, Zhao, Zhongdong, Kropf, Jeffrey E, Currie, Kevin S, Swaminathan, Sundaramoorthi
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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