Macrocyclic biphenyl tetraoxazoles: Synthesis, evaluation as G-quadruplex stabilizers and cytotoxic activity
Blankson, Gifty A., Pilch, Daniel S., Liu, Angela A., Liu, Leroy F., Rice, Joseph E., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry (01.08.2013)
Published in Bioorganic & medicinal chemistry (01.08.2013)
Get full text
Journal Article
Hydrogen Peroxide Induces Topoisomerase I-mediated DNA Damage and Cell Death
Daroui, Parima, Desai, Shyamal D., Li, Tsai-Kun, Liu, Angela A., Liu, Leroy F.
Published in The Journal of biological chemistry (09.04.2004)
Published in The Journal of biological chemistry (09.04.2004)
Get full text
Journal Article
Macrocyclic hexaoxazoles: Influence of aminoalkyl substituents on RNA and DNA G-quadruplex stabilization and cytotoxicity
Satyanarayana, Mavurapu, Kim, Young-Ah, Rzuczek, Suzanne G., Pilch, Daniel S., Liu, Angela A., Liu, Leroy F., Rice, Joseph E., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Get full text
Journal Article
G-quadruplexes induce apoptosis in tumor cells
HAIYAN QI, LIN, Chao-Po, XUAN FU, WOOD, Laurence M, LIU, Angela A, TSAI, Yuan-Chin, YONGJIE CHEN, BARBIERI, Christopher M, PITCH, Daniel S, LIU, Leroy F
Published in Cancer research (Chicago, Ill.) (15.12.2006)
Published in Cancer research (Chicago, Ill.) (15.12.2006)
Get full text
Journal Article
Esters and amides of 2,3-dimethoxy-8,9-methylenedioxy-benzo[ i]phenanthridine-12-carboxylic acid: Potent cytotoxic and topoisomerase I-targeting agents
Zhu, Shejin, Ruchelman, Alexander L., Zhou, Nai, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry (15.12.2005)
Published in Bioorganic & medicinal chemistry (15.12.2005)
Get full text
Journal Article
Novel topoisomerase I-targeting antitumor agents synthesized from the N,N,N-trimethylammonium derivative of ARC-111, 5H-2,3-dimethoxy-8,9-methylenedioxy-5-[(2-N,N,N-trimethylammonium)ethyl]dibenzo[c,h][1,6]naphthyridin-6-one iodide
Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in European journal of medicinal chemistry (01.09.2009)
Published in European journal of medicinal chemistry (01.09.2009)
Get full text
Journal Article
Characterization of ARC-111 as a novel topoisomerase I-targeting anticancer drug
LI, Tsai-Kun, HOUGHTON, Peter J, DESAI, Shyamal D, DAROUI, Parima, LIU, Angela A, HARS, Eszter S, RUCHELMAN, Alexander L, LAVOIE, Edmond J, LIU, Leroy F
Published in Cancer research (Chicago, Ill.) (01.12.2003)
Get full text
Published in Cancer research (Chicago, Ill.) (01.12.2003)
Journal Article
12-Substituted 2,3-dimethoxy-8,9-methylenedioxybenzo[ i]phenanthridines as novel topoisomerase I-targeting antitumor agents
Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry (01.04.2009)
Published in Bioorganic & medicinal chemistry (01.04.2009)
Get full text
Journal Article
Cytotoxicity and TOP1-targeting activity of 8- and 9-amino derivatives of 5-butyl- and 5-(2-N,N-dimethylamino)ethyl-5H-dibenzo[c,h][1,6]naphthyridin-6-ones
Sharma, Lisa, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in European journal of medicinal chemistry (01.04.2009)
Published in European journal of medicinal chemistry (01.04.2009)
Get full text
Journal Article
Syntheses and biological evaluation of topoisomerase I-targeting agents related to 11 -[2-(N,N-dimethylamino)ethyl]-2,3-dimethoxy-8,9-methylenedioxy-11H-isoquino[4,3-c]cinnolin-12-one (ARC-31)
SATYANARAYANA, Mavurapu, WEI FENG, LIANG CHENG, LIU, Angela A, TSAI, Yuan-Chin, LIU, Leroy F, LAVOIE, Edmond J
Published in Bioorganic & medicinal chemistry (15.08.2008)
Published in Bioorganic & medicinal chemistry (15.08.2008)
Get full text
Journal Article
Facile formation of hydrophilic derivatives of 5H-8,9-dimethoxy-5-[2-(N,N-dimethylamino)ethyl]-2,3-methylenedioxydibenzo[c,h] [1,6]naphthyridin-6-one (ARC-111) and its 12-aza analog via quaternary ammonium intermediates
Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry letters (15.06.2008)
Published in Bioorganic & medicinal chemistry letters (15.06.2008)
Get full text
Journal Article
11-Substituted 2,3-dimethoxy-8,9-methylenedioxybenzo[ i]phenanthridine derivatives as novel topoisomerase I-targeting agents
Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry (15.09.2008)
Published in Bioorganic & medicinal chemistry (15.09.2008)
Get full text
Journal Article
Mutations of Human Topoisomerase IIα Affecting Multidrug Resistance and Sensitivity
Mao, Yong, Yu, Chiang, Hsieh, Tao-Shih, Nitiss, John L, Liu, Angela A, Wang, Huimin, Liu, Leroy F
Published in Biochemistry (Easton) (17.08.1999)
Published in Biochemistry (Easton) (17.08.1999)
Get full text
Journal Article
11-Substituted 2,3-dimethoxy-8,9-methylenedioxybenzo[i]phenanthridine derivatives as novel topoisomerase I-targeting agents
Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry (15.09.2008)
Published in Bioorganic & medicinal chemistry (15.09.2008)
Get full text
Journal Article
Differential Poisoning of Topoisomerases by Menogaril and Nogalamycin Dictated by the Minor Groove-Binding Nogalose Sugar
Sim, Sai-Peng, Gatto, Barbara, Yu, Chiang, Liu, Angela A, Li, Tsai-Kun, Pilch, Daniel S, LaVoie, Edmond J, Liu, Leroy F
Published in Biochemistry (Easton) (28.10.1997)
Published in Biochemistry (Easton) (28.10.1997)
Get full text
Journal Article
Cytotoxicity and TOPI-targeting activity of 8-and 9-amino derivatives of 5-butyl-and 5-(2-N,N-dimethylamino)ethyl-5H-dibenzo[c,h][1,6]naphthyridin-6-ones
SHARMA, Lisa, TSAI, Yuan-Chin, LIU, Angela A, LIU, Leroy F, LAVOIE, Edmond J
Published in European journal of medicinal chemistry (2009)
Get full text
Published in European journal of medicinal chemistry (2009)
Journal Article
Novel topoisomerase I-targeting antitumor agents synthesized from the N, N, N-trimethylammonium derivative of ARC-111, 5 H-2,3-dimethoxy-8,9-methylenedioxy-5-[(2- N, N, N-trimethylammonium)ethyl]dibenzo[ c, h][1,6]naphthyridin-6-one iodide
Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in European journal of medicinal chemistry (2009)
Published in European journal of medicinal chemistry (2009)
Get full text
Journal Article
Cytotoxicity and TOP1-targeting activity of 8- and 9-amino derivatives of 5-butyl- and 5-(2- N, N-dimethylamino)ethyl-5 H-dibenzo[ c, h][1,6]naphthyridin-6-ones
Sharma, Lisa, Tsai, Yuan-Chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in European journal of medicinal chemistry (2009)
Published in European journal of medicinal chemistry (2009)
Get full text
Journal Article
Facile formation of hydrophilic derivatives of 5H-8,9-dimethoxy-5-[2-(N,N-dimethylamino)ethyl]-2,3-methylene-dioxydibenzo[c,h] [1,6]naphthyridin-6-one (ARC-111) and its 12-aza analog via quaternary ammonium intermediates
WEI FENG, SATYANARAYANA, Mavurapu, TSAI, Yuan-Chin, LIU, Angela A, LIU, Leroy F, LAVOIE, Edmond J
Published in Bioorganic & medicinal chemistry letters (2008)
Get full text
Published in Bioorganic & medicinal chemistry letters (2008)
Journal Article
Facile formation of hydrophilic derivatives of 5 H-8,9-dimethoxy-5-[2-( N, N-dimethylamino)ethyl]-2,3-methylenedioxydibenzo[ c, h] [1,6]naphthyridin-6-one (ARC-111) and its 12-aza analog via quaternary ammonium intermediates
Feng, Wei, Satyanarayana, Mavurapu, Tsai, Yuan-chin, Liu, Angela A., Liu, Leroy F., LaVoie, Edmond J.
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
Get full text
Journal Article