Master Transcription Factors and Mediator Establish Super-Enhancers at Key Cell Identity Genes
Whyte, Warren A., Orlando, David A., Hnisz, Denes, Abraham, Brian J., Lin, Charles Y., Kagey, Michael H., Rahl, Peter B., Lee, Tong Ihn, Young, Richard A.
Published in Cell (11.04.2013)
Published in Cell (11.04.2013)
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Selective Inhibition of Tumor Oncogenes by Disruption of Super-Enhancers
Lovén, Jakob, Hoke, Heather A., Lin, Charles Y., Lau, Ashley, Orlando, David A., Vakoc, Christopher R., Bradner, James E., Lee, Tong Ihn, Young, Richard A.
Published in Cell (11.04.2013)
Published in Cell (11.04.2013)
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Transcriptional Amplification in Tumor Cells with Elevated c-Myc
Lin, Charles Y., Lovén, Jakob, Rahl, Peter B., Paranal, Ronald M., Burge, Christopher B., Bradner, James E., Lee, Tong Ihn, Young, Richard A.
Published in Cell (28.09.2012)
Published in Cell (28.09.2012)
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Convergence of Developmental and Oncogenic Signaling Pathways at Transcriptional Super-Enhancers
Hnisz, Denes, Schuijers, Jurian, Lin, Charles Y., Weintraub, Abraham S., Abraham, Brian J., Lee, Tong Ihn, Bradner, James E., Young, Richard A.
Published in Molecular cell (16.04.2015)
Published in Molecular cell (16.04.2015)
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Discovery and Characterization of Super-Enhancer-Associated Dependencies in Diffuse Large B Cell Lymphoma
Chapuy, Bjoern, McKeown, Michael R., Lin, Charles Y., Monti, Stefano, Roemer, Margaretha G.M., Qi, Jun, Rahl, Peter B., Sun, Heather H., Yeda, Kelly T., Doench, John G., Reichert, Elaine, Kung, Andrew L., Rodig, Scott J., Young, Richard A., Shipp, Margaret A., Bradner, James E.
Published in Cancer cell (09.12.2013)
Published in Cancer cell (09.12.2013)
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Revisiting Global Gene Expression Analysis
Lovén, Jakob, Orlando, David A., Sigova, Alla A., Lin, Charles Y., Rahl, Peter B., Burge, Christopher B., Levens, David L., Lee, Tong Ihn, Young, Richard A.
Published in Cell (26.10.2012)
Published in Cell (26.10.2012)
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BET Bromodomains Mediate Transcriptional Pause Release in Heart Failure
Anand, Priti, Brown, Jonathan D., Lin, Charles Y., Qi, Jun, Zhang, Rongli, Artero, Pedro Calderon, Alaiti, M. Amer, Bullard, Jace, Alazem, Kareem, Margulies, Kenneth B., Cappola, Thomas P., Lemieux, Madeleine, Plutzky, Jorge, Bradner, James E., Haldar, Saptarsi M.
Published in Cell (01.08.2013)
Published in Cell (01.08.2013)
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NF-κB Directs Dynamic Super Enhancer Formation in Inflammation and Atherogenesis
Brown, Jonathan D., Lin, Charles Y., Duan, Qiong, Griffin, Gabriel, Federation, Alexander J., Paranal, Ronald M., Bair, Steven, Newton, Gail, Lichtman, Andrew H., Kung, Andrew L., Yang, Tianlun, Wang, Hong, Luscinskas, Francis W., Croce, Kevin J., Bradner, James E., Plutzky, Jorge
Published in Molecular cell (23.10.2014)
Published in Molecular cell (23.10.2014)
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Taming of the beast: shaping Myc-dependent amplification
Wolf, Elmar, Lin, Charles Y, Eilers, Martin, Levens, David L
Published in Trends in cell biology (01.04.2015)
Published in Trends in cell biology (01.04.2015)
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Mutant NPM1 Maintains the Leukemic State through HOX Expression
Brunetti, Lorenzo, Gundry, Michael C., Sorcini, Daniele, Guzman, Anna G., Huang, Yung-Hsin, Ramabadran, Raghav, Gionfriddo, Ilaria, Mezzasoma, Federica, Milano, Francesca, Nabet, Behnam, Buckley, Dennis L., Kornblau, Steven M., Lin, Charles Y., Sportoletti, Paolo, Martelli, Maria Paola, Falini, Brunangelo, Goodell, Margaret A.
Published in Cancer cell (10.09.2018)
Published in Cancer cell (10.09.2018)
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BET Bromodomain Proteins Function as Master Transcription Elongation Factors Independent of CDK9 Recruitment
Winter, Georg E., Mayer, Andreas, Buckley, Dennis L., Erb, Michael A., Roderick, Justine E., Vittori, Sarah, Reyes, Jaime M., di Iulio, Julia, Souza, Amanda, Ott, Christopher J., Roberts, Justin M., Zeid, Rhamy, Scott, Thomas G., Paulk, Joshiawa, Lachance, Kate, Olson, Calla M., Dastjerdi, Shiva, Bauer, Sophie, Lin, Charles Y., Gray, Nathanael S., Kelliher, Michelle A., Churchman, L. Stirling, Bradner, James E.
Published in Molecular cell (06.07.2017)
Published in Molecular cell (06.07.2017)
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Models of human core transcriptional regulatory circuitries
Saint-André, Violaine, Federation, Alexander J, Lin, Charles Y, Abraham, Brian J, Reddy, Jessica, Lee, Tong Ihn, Bradner, James E, Young, Richard A
Published in Genome research (01.03.2016)
Published in Genome research (01.03.2016)
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Development of a Selective CDK7 Covalent Inhibitor Reveals Predominant Cell-Cycle Phenotype
Olson, Calla M, Liang, Yanke, Leggett, Alan, Park, Woojun D, Li, Lianbo, Mills, Caitlin E, Elsarrag, Selma Z, Ficarro, Scott B, Zhang, Tinghu, Düster, Robert, Geyer, Matthias, Sim, Taebo, Marto, Jarrod A, Sorger, Peter K, Westover, Ken D, Lin, Charles Y, Kwiatkowski, Nicholas, Gray, Nathanael S
Published in Cell chemical biology (20.06.2019)
Published in Cell chemical biology (20.06.2019)
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HDAC Inhibition Reverses Preexisting Diastolic Dysfunction and Blocks Covert Extracellular Matrix Remodeling
Travers, Joshua G, Wennersten, Sara A, Peña, Brisa, Bagchi, Rushita A, Smith, Harrison E, Hirsch, Rachel A, Vanderlinden, Lauren A, Lin, Ying-Hsi, Dobrinskikh, Evgenia, Demos-Davies, Kimberly M, Cavasin, Maria A, Mestroni, Luisa, Steinkühler, Christian, Lin, Charles Y, Houser, Steven R, Woulfe, Kathleen C, Lam, Maggie P Y, McKinsey, Timothy A
Published in Circulation (New York, N.Y.) (11.05.2021)
Published in Circulation (New York, N.Y.) (11.05.2021)
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Epigenomic analysis detects aberrant super-enhancer DNA methylation in human cancer
Heyn, Holger, Vidal, Enrique, Ferreira, Humberto J, Vizoso, Miguel, Sayols, Sergi, Gomez, Antonio, Moran, Sebastian, Boque-Sastre, Raquel, Guil, Sonia, Martinez-Cardus, Anna, Lin, Charles Y, Royo, Romina, Sanchez-Mut, Jose V, Martinez, Ramon, Gut, Marta, Torrents, David, Orozco, Modesto, Gut, Ivo, Young, Richard A, Esteller, Manel
Published in Genome Biology (26.01.2016)
Published in Genome Biology (26.01.2016)
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Discovery of a selective inhibitor of doublecortin like kinase 1
Ferguson, Fleur M, Nabet, Behnam, Raghavan, Srivatsan, Liu, Yan, Leggett, Alan L, Kuljanin, Miljan, Kalekar, Radha L, Yang, Annan, He, Shuning, Wang, Jinhua, Ng, Raymond W S, Sulahian, Rita, Li, Lianbo, Poulin, Emily J, Huang, Ling, Koren, Jost, Dieguez-Martinez, Nora, Espinosa, Sergio, Zeng, Zhiyang, Corona, Cesear R, Vasta, James D, Ohi, Ryoma, Sim, Taebo, Kim, Nam Doo, Harshbarger, Wayne, Lizcano, Jose M, Robers, Matthew B, Muthaswamy, Senthil, Lin, Charles Y, Look, A Thomas, Haigis, Kevin M, Mancias, Joseph D, Wolpin, Brian M, Aguirre, Andrew J, Hahn, William C, Westover, Kenneth D, Gray, Nathanael S
Published in Nature chemical biology (01.06.2020)
Published in Nature chemical biology (01.06.2020)
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PI3K/AKT Signaling Regulates H3K4 Methylation in Breast Cancer
Spangle, Jennifer M., Dreijerink, Koen M., Groner, Anna C., Cheng, Hailing, Ohlson, Carolynn E., Reyes, Jaime, Lin, Charles Y., Bradner, James, Zhao, Jean J., Roberts, Thomas M., Brown, Myles
Published in Cell reports (Cambridge) (21.06.2016)
Published in Cell reports (Cambridge) (21.06.2016)
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Targeting MYC dependency in ovarian cancer through inhibition of CDK7 and CDK12/13
Zeng, Mei, Kwiatkowski, Nicholas P, Zhang, Tinghu, Nabet, Behnam, Xu, Mousheng, Liang, Yanke, Quan, Chunshan, Wang, Jinhua, Hao, Mingfeng, Palakurthi, Sangeetha, Zhou, Shan, Zeng, Qing, Kirschmeier, Paul T, Meghani, Khyati, Leggett, Alan L, Qi, Jun, Shapiro, Geoffrey I, Liu, Joyce F, Matulonis, Ursula A, Lin, Charles Y, Konstantinopoulos, Panagiotis A, Gray, Nathanael S
Published in eLife (13.11.2018)
Published in eLife (13.11.2018)
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PAX8 activates metabolic genes via enhancer elements in Renal Cell Carcinoma
Bleu, Melusine, Gaulis, Swann, Lopes, Rui, Sprouffske, Kathleen, Apfel, Verena, Holwerda, Sjoerd, Pregnolato, Marco, Yildiz, Umut, Cordoʹ, Valentina, Dost, Antonella F M, Knehr, Judith, Carbone, Walter, Lohmann, Felix, Lin, Charles Y, Bradner, James E, Kauffmann, Audrey, Tordella, Luca, Roma, Guglielmo, Galli, Giorgio G
Published in Nature communications (20.08.2019)
Published in Nature communications (20.08.2019)
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BET bromodomain proteins regulate enhancer function during adipogenesis
Brown, Jonathan D., Feldman, Zachary B., Doherty, Sean P., Reyes, Jaime M., Rahl, Peter B., Lin, Charles Y., Sheng, Quanhu, Duan, Qiong, Federation, Alexander J., Kung, Andrew L., Haldar, Saptarsi M., Young, Richard A., Plutzky, Jorge, Bradner, James E.
Published in Proceedings of the National Academy of Sciences - PNAS (27.02.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (27.02.2018)
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