Discovery of STAT3 Inhibitors: Recent Advances and Future Perspectives
Song, Jiatao, Wang, Jiawei, Tian, Sheng, Li, Huanqiu
Published in Current medicinal chemistry (01.01.2023)
Published in Current medicinal chemistry (01.01.2023)
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Reaction-Based “Off–On” Fluorescent Probe Enabling Detection of Endogenous Labile Fe2+ and Imaging of Zn2+-induced Fe2+ Flux in Living Cells and Elevated Fe2+ in Ischemic Stroke
Xuan, Weimin, Pan, Rong, Wei, Yongyi, Cao, Yanting, Li, Huanqiu, Liang, Fu-Sen, Liu, Ke-Jian, Wang, Wei
Published in Bioconjugate chemistry (17.02.2016)
Published in Bioconjugate chemistry (17.02.2016)
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γ-AApeptides as a New Class of Peptidomimetics: Design, Synthesis, and Applications
Su, Ma, Zhu, Yifan, Wang, Wei, Liu, Feng, Li, Huanqiu
Published in Current topics in medicinal chemistry (01.01.2021)
Published in Current topics in medicinal chemistry (01.01.2021)
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Targeting P2Y14R protects against necroptosis of intestinal epithelial cells through PKA/CREB/RIPK1 axis in ulcerative colitis
Liu, Chunxiao, Wang, Hui, Han, Lu, Zhu, Yifan, Ni, Shurui, Zhi, Jingke, Yang, Xiping, Zhi, Jiayi, Sheng, Tian, Li, Huanqiu, Hu, Qinghua
Published in Nature communications (07.03.2024)
Published in Nature communications (07.03.2024)
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GPR105-Targeted Therapy Promotes Gout Resolution as a Switch Between NETosis and Apoptosis of Neutrophils
Liu, Chunxiao, Zhou, Mengze, Jiang, Wenjiao, Ye, Shumin, Tian, Sheng, Jiang, Cheng, Hao, Kun, Li, Huanqiu, Hu, Qinghua
Published in Frontiers in immunology (30.03.2022)
Published in Frontiers in immunology (30.03.2022)
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FDW028, a novel FUT8 inhibitor, impels lysosomal proteolysis of B7-H3 via chaperone-mediated autophagy pathway and exhibits potent efficacy against metastatic colorectal cancer
Wang, Mengmeng, Zhang, Zhoudong, Chen, Mengxi, Lv, Yixin, Tian, Sheng, Meng, Fanyi, Zhang, Yawen, Guo, Xuqin, Chen, Yinshuang, Yang, Man, Li, Jiawei, Qiu, Tian, Xu, Fang, Li, Zhi, Zhang, Qi, Yang, Jie, Sun, Jing, Zhang, Hongjian, Zhang, Haiyang, Li, Huanqiu, Wang, Weipeng
Published in Cell death & disease (03.08.2023)
Published in Cell death & disease (03.08.2023)
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A novel SRSF3 inhibitor, SFI003, exerts anticancer activity against colorectal cancer by modulating the SRSF3/DHCR24/ROS axis
Zhang, Yawen, Wang, Mengmeng, Meng, Fanyi, Yang, Man, Chen, Yinshuang, Guo, Xuqin, Wang, Weiwei, Zhu, Yifan, Guo, Yundi, Feng, Chunlai, Tian, Shen, Zhang, Hongjian, Li, Huanqiu, Sun, Jing, Wang, Weipeng
Published in Cell death discovery (02.05.2022)
Published in Cell death discovery (02.05.2022)
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Discovery of novel and potent P2Y14R antagonists via structure-based virtual screening for the treatment of acute gouty arthritis
Wang, Weiwei, Liu, Chunxiao, Li, Hanwen, Tian, Sheng, Liu, Yingxian, Wang, Nanxi, Yan, Duanyang, Li, Huanqiu, Hu, Qinghua
Published in Journal of advanced research (01.05.2020)
Published in Journal of advanced research (01.05.2020)
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Journal Article
Continued exploration of biphenylsulfonamide scaffold as a platform for aggrecanase-1 inhibition
Hu, Yonghan, Xing, Li, Thomason, Jennifer R., Xiang, Jason, Ipek, Manus, Guler, Satenig, Li, Huanqiu, Sabatini, Joshua, Chockalingam, Priya, Reifenberg, Erica, Sheldon, Richard, Morris, Elisabeth A., Georgiadis, Katy E., Tam, Steve
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
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Therapeutic potential of fucosyltransferases in cancer and recent development of targeted inhibitors
Lv, Yixin, Zhang, Zhoudong, Tian, Sheng, Wang, Weipeng, Li, Huanqiu
Published in Drug discovery today (01.01.2023)
Published in Drug discovery today (01.01.2023)
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Discovery of Janus Kinase 2 (JAK2) and Histone Deacetylase (HDAC) Dual Inhibitors as a Novel Strategy for the Combinational Treatment of Leukemia and Invasive Fungal Infections
Huang, Yahui, Dong, Guoqiang, Li, Huanqiu, Liu, Na, Zhang, Wannian, Sheng, Chunquan
Published in Journal of medicinal chemistry (26.07.2018)
Published in Journal of medicinal chemistry (26.07.2018)
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Corrigendum to “Therapeutic potential of fucosyltransferases in cancer and recent development of targeted inhibitors” [Drug Discov. Today 28(1) (2023) 103394]
Lv, Yixin, Zhang, Zhoudong, Tian, Sheng, Wang, Weipeng, Li, Huanqiu
Published in Drug discovery today (01.03.2023)
Published in Drug discovery today (01.03.2023)
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Journal Article
Sodium tanshinone IIA sulfonate ameliorates ischemia-induced myocardial inflammation and lipid accumulation in Beagle dogs through NLRP3 inflammasome
Hu, Qinghua, Wei, Bo, Wei, Linlin, Hua, Kai, Yu, Xing, Li, Huanqiu, Ji, Hui
Published in International journal of cardiology (01.10.2015)
Published in International journal of cardiology (01.10.2015)
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Journal Article
Prediction of Drug‐Induced Liver Injury: From Molecular Physicochemical Properties and Scaffold Architectures to Machine Learning Approaches
Zhao, Yulong, Zhang, Zhoudong, Kong, Xiaotian, Wang, Kai, Wang, Yaxuan, Jia, Jie, Li, Huanqiu, Tian, Sheng
Published in Chemical biology & drug design (01.08.2024)
Published in Chemical biology & drug design (01.08.2024)
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Macrophage P2Y6 receptor deletion attenuates atherosclerosis by limiting foam cell formation through phospholipase Cβ/store-operated calcium entry/calreticulin/scavenger receptor A pathways
Li, Yehong, Zhou, Mengze, Li, Huanqiu, Dai, Chen, Yin, Li, Liu, Chunxiao, Li, Yuxin, Zhang, Enming, Dong, Xinli, Ji, Hui, Hu, Qinghua
Published in European heart journal (27.01.2024)
Published in European heart journal (27.01.2024)
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HJ22, a Novel derivative of piperine, Attenuates ibotenic acid-induced cognitive impairment, oxidativestress, apoptosis and inflammation via inhibiting the protein-protein interaction of Keap1-Nrf2
Yang, Xiping, Ji, Jing, Liu, Chunxiao, Zhou, Mengze, Li, Huanqiu, Ye, Shumin, Hu, Qinghua
Published in International immunopharmacology (01.06.2020)
Published in International immunopharmacology (01.06.2020)
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Discovery and computational studies of 2-phenyl-benzoxazole acetamide derivatives as promising P2Y(14)R antagonists with anti-gout potential
Zhou, Mengze, Wang, Weiwei, Wang, Zhongkui, Wang, Yilin, Zhu, Yifan, Lin, Zhiqian, Tian, Sheng, Huang, Yuan, Hu, Qinghua, Li, Huanqiu
Published in European journal of medicinal chemistry (05.01.2022)
Published in European journal of medicinal chemistry (05.01.2022)
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