Bifunctional [2‘,6‘-Dimethyl-l-tyrosine]endomorphin-2 Analogues Substituted at Position 3 with Alkylated Phenylalanine Derivatives Yield Potent Mixed μ-Agonist/δ-Antagonist and Dual μ-Agonist/δ-Agonist Opioid Ligands
Li, Tingyou, Shiotani, Kimitaka, Miyazaki, Anna, Tsuda, Yuko, Ambo, Akihiro, Sasaki, Yusuke, Jinsmaa, Yunden, Marczak, Ewa, Bryant, Sharon D, Lazarus, Lawrence H, Okada, Yoshio
Published in Journal of medicinal chemistry (14.06.2007)
Published in Journal of medicinal chemistry (14.06.2007)
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Differentiation of opioid receptor preference by [Dmt 1]endomorphin-2-mediated antinociception in the mouse
Jinsmaa, Yunden, Fujita, Yoshio, Shiotani, Kimitaka, Miyazaki, Anna, Li, Tingyou, Tsuda, Yuko, Okada, Yoshio, Ambo, Akihiro, Sasaki, Yusuke, Bryant, Sharon D., Lazarus, Lawrence H.
Published in European journal of pharmacology (10.02.2005)
Published in European journal of pharmacology (10.02.2005)
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Oral Bioavailability of a New Class of μ-Opioid Receptor Agonists Containing 3,6-Bis[Dmt-NH(CH2) n ]-2(1H)-pyrazinone with Central-Mediated Analgesia
Jinsmaa, Yunden, Miyazaki, Anna, Fujita, Yoshio, Li, Tingyou, Fujisawa, Yutaka, Shiotani, Kimitaka, Tsuda, Yuko, Yokoi, Toshio, Ambo, Akihiro, Sasaki, Yusuke, Bryant, Sharon D, Lazarus, Lawrence H, Okada, Yoshio
Published in Journal of medicinal chemistry (06.05.2004)
Published in Journal of medicinal chemistry (06.05.2004)
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Potent in vivo antinociception and opioid receptor preference of the novel analogue [Dmt 1]endomorphin-1
Jinsmaa, Yunden, Marczak, Ewa, Fujita, Yoshio, Shiotani, Kimitaka, Miyazaki, Anna, Li, Tingyou, Tsuda, Yuko, Ambo, Akihiro, Sasaki, Yusuke, Bryant, Sharon D., Okada, Yoshio, Lazarus, Lawrence H.
Published in Pharmacology, biochemistry and behavior (01.06.2006)
Published in Pharmacology, biochemistry and behavior (01.06.2006)
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Transformation of μ-opioid receptor agonists into biologically potent μ-opioid receptor antagonists
Li, Tingyou, Jinsmaa, Yunden, Nedachi, Masahiro, Miyazaki, Anna, Tsuda, Yuko, Ambo, Akihiro, Sasaki, Yusuke, Bryant, Sharon D., Marczak, Ewa, Li, Qiang, Swartzwelder, H. Scott, Lazarus, Lawrence H., Okada, Yoshio
Published in Bioorganic & medicinal chemistry (01.02.2007)
Published in Bioorganic & medicinal chemistry (01.02.2007)
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Nonlinear relationship of vegetation greening with nature and human factors and its forecast – A case study of Southwest China
Liu, Huiyu, Jiao, Fusheng, Yin, Jingqiu, Li, Tingyou, Gong, Haibo, Wang, Zhaoyue, Lin, Zhenshan
Published in Ecological indicators (01.04.2020)
Published in Ecological indicators (01.04.2020)
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Design and synthesis of opioidmimetics containing 2′,6′-dimethyl- l-tyrosine and a pyrazinone-ring platform
Shiotani, Kimitaka, Li, Tingyou, Miyazaki, Anna, Tsuda, Yuko, Yokoi, Toshio, Ambo, Akihiro, Sasaki, Yusuke, Bryant, Sharon D., Lazarus, Lawrence H., Okada, Yoshio
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Enantioselective Synthesis of a Phenylalanine Library Containing Alkyl Groups on the Aromatic Moiety: Confirmation of Stereostructure by X-Ray Analysis
Li, Tingyou, Tsuda, Yuko, Minoura, Katsuhiko, In, Yasuko, Ishida, Toshimasa, Lazarus, Lawrence H., Okada, Yoshio
Published in Chemical & Pharmaceutical Bulletin (2006)
Published in Chemical & Pharmaceutical Bulletin (2006)
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Synthesis of 3,6-bis[H-Tyr/H-Dmt-NH(CH 2) m, n ]-2(1 H)pyrazinone derivatives: Function of alkyl chain length on opioid activity
Shiotani, Kimitaka, Li, Tingyou, Miyazaki, Anna, Tsuda, Yuko, Bryant, Sharon D., Ambo, Akihiro, Sasaki, Yusuke, Lazarus, Lawrence H., Okada, Yoshio
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
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A highly dl-stereoselective pinacolization of aromatic aldehydes mediated by TiCl4-Zn
Li, TY, Cui, W, Liu, JG, Zhao, JZ, Wang, ZM
Published in Chemical communications (Cambridge, England) (01.01.2000)
Published in Chemical communications (Cambridge, England) (01.01.2000)
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Nitric oxide-donating and reactive oxygen species-responsive prochelators based on 8-hydroxyquinoline as anticancer agents
Zhang, Yuxia, Yang, Jiaxin, Meng, Tingting, Qin, Yajuan, Li, Tingyou, Fu, Junjie, Yin, Jian
Published in European journal of medicinal chemistry (15.02.2021)
Published in European journal of medicinal chemistry (15.02.2021)
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Orthogonal Lithography for Halide Perovskite Optoelectronic Nanodevices
Lin, Chun-Ho, Cheng, Bin, Li, Ting-You, Retamal, José Ramón Durán, Wei, Tzu-Chiao, Fu, Hui-Chun, Fang, Xiaosheng, He, Jr-Hau
Published in ACS nano (26.02.2019)
Published in ACS nano (26.02.2019)
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Application of liquid chromatography–tandem mass spectrometry for the determination of opioidmimetics in the brain dialysates from rats treated with opioidmimetics intraperitoneally
Igarashi, Kazuo, Murabayashi, Yuki, Hotta, Koichiro, Kitamura, Youji, Kasuya, Fumiyo, Shiotani, Kimitaka, Tingyou, Li, Miyazaki, Anna, Tsuda, Yuko, Okada, Yoshio, Fukushima, Shoji
Published in Journal of chromatography. B (25.06.2004)
Published in Journal of chromatography. B (25.06.2004)
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Conference Proceeding
Suitability of three seaweeds as feed in culturing strawberry conch Strombus luhuanus
Li, Changlin, Liu, Ertian, Li, Tingyou, Wang, Aimin, Liu, Chunsheng, Gu, Zhifeng
Published in Aquaculture (30.03.2020)
Published in Aquaculture (30.03.2020)
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Intracerebroventricular administration of CYX-6, a potent μ-opioid receptor agonist, a δ- and κ-opioid receptor antagonist and a biased ligand at μ, δ & κ-opioid receptors, evokes antinociception with minimal constipation and respiratory depression in rats in contrast to morphine
Imam, Mohammad Zafar, Kuo, Andy, Ghassabian, Sussan, Cai, Yunxin, Qin, Yajuan, Li, Tingyou, Smith, Maree T.
Published in European journal of pharmacology (15.03.2020)
Published in European journal of pharmacology (15.03.2020)
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CYX-5, a G-protein biassed MOP receptor agonist, DOP receptor antagonist and KOP receptor agonist, evokes constipation but not respiratory depression relative to morphine in rats
Imam, Mohammad Zafar, Kuo, Andy, Ghassabian, Sussan, Cai, Yunxin, Qin, Yajuan, Li, Tingyou, Smith, Maree T.
Published in Pharmacological reports (01.06.2023)
Published in Pharmacological reports (01.06.2023)
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