Computational modeling studies reveal the origin of the binding preference of 3‐(3,4‐di hydroisoquinolin‐2(1H)‐ylsulfonyl)benzoic acids for AKR1C3 over its isoforms
Kong, Xiaotian, Xing, Enming, Wu, Sijin, Zhuang, Tony, Li, Pui‐Kai, Li, Chunhua, Cheng, Xiaolin
Published in Protein science (01.12.2022)
Published in Protein science (01.12.2022)
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Journal Article
Multi-targeted therapy of cancer by niclosamide: A new application for an old drug
Li, Yonghe, Li, Pui-Kai, Roberts, Michael J, Arend, Rebecca C, Samant, Rajeev S, Buchsbaum, Donald J
Published in Cancer letters (10.07.2014)
Published in Cancer letters (10.07.2014)
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Journal Article
STAT3 Is Necessary for Proliferation and Survival in Colon Cancer―Initiating Cells
LI LIN, AIGUO LIU, ZHENGANG PENG, LIN, Huey-Jen, LI, Pui-Kai, CHENGLONG LI, JIAYUH LIN
Published in Cancer research (Chicago, Ill.) (01.12.2011)
Published in Cancer research (Chicago, Ill.) (01.12.2011)
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Journal Article
Protective effect of suppressing STAT3 activity in LPS-induced acute lung injury
Zhao, Jiping, Yu, Hao, Liu, Yudong, Gibson, Sara A, Yan, Zhaoqi, Xu, Xin, Gaggar, Amit, Li, Pui-Kai, Li, Chenglong, Wei, Shi, Benveniste, Etty N, Qin, Hongwei
Published in American journal of physiology. Lung cellular and molecular physiology (01.11.2016)
Published in American journal of physiology. Lung cellular and molecular physiology (01.11.2016)
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Journal Article
BET Bromodomain Inhibitors: Novel Design Strategies and Therapeutic Applications
To, Kenneth K W, Xing, Enming, Larue, Ross C, Li, Pui-Kai
Published in Molecules (Basel, Switzerland) (29.03.2023)
Published in Molecules (Basel, Switzerland) (29.03.2023)
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Journal Article
Inhibition of STAT3 Signaling Blocks the Anti-apoptotic Activity of IL-6 in Human Liver Cancer Cells
Liu, Yan, Li, Pui-Kai, Li, Chenglong, Lin, Jiayuh
Published in The Journal of biological chemistry (27.08.2010)
Published in The Journal of biological chemistry (27.08.2010)
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Journal Article
JAK-STAT Blockade Inhibits Tumor Initiation and Clonogenic Recovery of Prostate Cancer Stem-like Cells
KROON, Paula, BERRY, Paul A, MAITLAND, Norman J, COLLINS, Anne T, STOWER, Michael J, RODRIGUES, Greta, MANN, Vincent M, SIMMS, Matthew, BHASIN, Deepak, CHETTIAR, Somsundaram, CHENGLONG LI, LI, Pui-Kai
Published in Cancer research (Chicago, Ill.) (15.08.2013)
Published in Cancer research (Chicago, Ill.) (15.08.2013)
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Journal Article
Novel STAT3 Phosphorylation Inhibitors Exhibit Potent Growth-Suppressive Activity in Pancreatic and Breast Cancer Cells
LI LIN, HUTZEN, Brian, LI, Pui-Kai, CHENGLONG LI, FUCHS, James, LIN, Jiayuh, MINGXIN ZUO, BALL, Sarah, DEANGELIS, Stephanie, FOUST, Elizabeth, PANDIT, Bulbul, IHNAT, Michael A, SHENOY, Satyendra S, KULP, Samuel
Published in Cancer research (Chicago, Ill.) (15.03.2010)
Published in Cancer research (Chicago, Ill.) (15.03.2010)
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Journal Article
Curcumin is a potent DNA hypomethylation agent
Liu, Zhongfa, Xie, Zhiliang, Jones, William, Pavlovicz, Ryan E., Liu, Shujun, Yu, Jianhua, Li, Pui-kai, Lin, Jiayuh, Fuchs, Jame R., Marcucci, Guido, Li, Chenglong, Chan, Kenneth K.
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Journal Article
Sorafenib Overcomes TRAIL Resistance of Hepatocellular Carcinoma Cells through the Inhibition of STAT3
CHEN, Kuen-Feng, TAI, Wei-Tien, LIU, Tsung-Hao, HUANG, Hsiang-Po, LIN, Yu-Chin, SHIAU, Chung-Wai, LI, Pui-Kai, CHEN, Pei-Jer, CHENG, Ann-Lii
Published in Clinical cancer research (01.11.2010)
Published in Clinical cancer research (01.11.2010)
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Journal Article
A small molecule, LLL12 inhibits constitutive STAT3 and IL-6-induced STAT3 signaling and exhibits potent growth suppressive activity in human multiple myeloma cells
Lin, Li, Benson Jr, Don M., DeAngelis, Stephanie, Bakan, Courtney E., Li, Pui-Kai, Li, Chenglong, Lin, Jiayuh
Published in International journal of cancer (15.03.2012)
Published in International journal of cancer (15.03.2012)
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Journal Article
A Novel Small Molecule, LLL12, Inhibits STAT3 Phosphorylation and Activities and Exhibits Potent Growth-Suppressive Activity in Human Cancer Cells
Lin, Li, Hutzen, Brian, Li, Pui-Kai, Ball, Sarah, Zuo, Mingxin, DeAngelis, Stephanie, Foust, Elizabeth, Sobo, Matthew, Friedman, Lauren, Bhasin, Deepak, Cen, Ling, Li, Chenglong, Lin, Jiayuh
Published in Neoplasia (New York, N.Y.) (01.01.2010)
Published in Neoplasia (New York, N.Y.) (01.01.2010)
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Journal Article
First-in-human trial of a STAT3 decoy oligonucleotide in head and neck tumors: implications for cancer therapy
Sen, Malabika, Thomas, Sufi M, Kim, Seungwon, Yeh, Joanne I, Ferris, Robert L, Johnson, Jonas T, Duvvuri, Umamaheswar, Lee, Jessica, Sahu, Nivedita, Joyce, Sonali, Freilino, Maria L, Shi, Haibin, Li, Changyou, Ly, Danith, Rapireddy, Srinivas, Etter, Jonathan P, Li, Pui-Kai, Wang, Lin, Chiosea, Simion, Seethala, Raja R, Gooding, William E, Chen, Xiaomin, Kaminski, Naftali, Pandit, Kusum, Johnson, Daniel E, Grandis, Jennifer R
Published in Cancer discovery (01.08.2012)
Published in Cancer discovery (01.08.2012)
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Journal Article
Evaluation of STAT3 signaling in ALDH+ and ALDH+/CD44+/CD24- subpopulations of breast cancer cells
Lin, Li, Hutzen, Brian, Lee, Hsiu-Fang, Peng, Zhengang, Wang, Wenlong, Zhao, Chongqiang, Lin, Huey-Jen, Sun, Duxin, Li, Pui-Kai, Li, Chenglong, Korkaya, Hasan, Wicha, Max S, Lin, Jiayuh
Published in PloS one (23.12.2013)
Published in PloS one (23.12.2013)
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Journal Article
Phosphoproteomic analysis of anaplastic lymphoma kinase (ALK) downstream signaling pathways identifies signal transducer and activator of transcription 3 as a functional target of activated ALK in neuroblastoma cells
Sattu, Kamaraj, Hochgräfe, Falko, Wu, Jianmin, Umapathy, Ganesh, Schönherr, Christina, Ruuth, Kristina, Chand, Damini, Witek, Barbara, Fuchs, James, Li, Pui‐Kai, Hugosson, Fredrik, Daly, Roger J., Palmer, Ruth H., Hallberg, Bengt
Published in The FEBS journal (01.11.2013)
Published in The FEBS journal (01.11.2013)
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Journal Article
Structurally modified curcumin analogs inhibit STAT3 phosphorylation and promote apoptosis of human renal cell carcinoma and melanoma cell lines
Bill, Matthew A, Nicholas, Courtney, Mace, Thomas A, Etter, Jonathan P, Li, Chenglong, Schwartz, Eric B, Fuchs, James R, Young, Gregory S, Lin, Li, Lin, Jiayuh, He, Lei, Phelps, Mitch, Li, Pui-Kai, Lesinski, Gregory B
Published in PloS one (10.08.2012)
Published in PloS one (10.08.2012)
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Journal Article
Glioma Cell Migration on Three-dimensional Nanofiber Scaffolds Is Regulated by Substrate Topography and Abolished by Inhibition of STAT3 Signaling
Agudelo-Garcia, Paula A, De Jesus, Jessica K, Williams, Shante P, Nowicki, Michal O, Chiocca, Ennio Antonio, Liyanarachchi, Sandya, Li, Pui-Kai, Lannutti, John J, Johnson, Jed K, Lawler, Sean E, Viapiano, Mariano S
Published in Neoplasia (New York, N.Y.) (01.09.2011)
Published in Neoplasia (New York, N.Y.) (01.09.2011)
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Journal Article
New curcumin analogues exhibit enhanced growth‐suppressive activity and inhibit AKT and signal transducer and activator of transcription 3 phosphorylation in breast and prostate cancer cells
Lin, Li, Hutzen, Brian, Ball, Sarah, Foust, Elizabeth, Sobo, Matthew, Deangelis, Stephanie, Pandit, Bulbul, Friedman, Lauren, Li, Chenglong, Li, Pui‐Kai, Fuchs, James, Lin, Jiayuh
Published in Cancer science (01.09.2009)
Published in Cancer science (01.09.2009)
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