A redox-neutral catechol synthesis
Wu, Qian, Yan, Dingyuan, Chen, Ying, Wang, Ting, Xiong, Feng, Wei, Wei, Lu, Yi, Sun, Wei-Yin, Li, Jie Jack, Zhao, Jing
Published in Nature communications (27.01.2017)
Published in Nature communications (27.01.2017)
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Journal Article
A bioinspired and biocompatible ortho-sulfiliminyl phenol synthesis
Xiong, Feng, Lu, Liang, Sun, Tian-Yu, Wu, Qian, Yan, Dingyuan, Chen, Ying, Zhang, Xinhao, Wei, Wei, Lu, Yi, Sun, Wei-Yin, Li, Jie Jack, Zhao, Jing
Published in Nature communications (19.06.2017)
Published in Nature communications (19.06.2017)
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Journal Article
Rational Design and Synthesis of 4-((1R,2R)-2-Hydroxycyclohexyl)-2(trifluoromethyl)benzonitrile (PF-998425), a Novel, Nonsteroidal Androgen Receptor Antagonist Devoid of Phototoxicity for Dermatological Indications
Li, Jie Jack, Iula, Donna M, Nguyen, Maria N, Hu, Lain-Yen, Dettling, Danielle, Johnson, Theodore R, Du, Daniel Y, Shanmugasundaram, Veerabahu, Van Camp, Jennifer A, Wang, Zhi, Harter, William G, Yue, Wen-Song, Boys, Mark L, Wade, Kimberly J, Drummond, Elena M, Samas, Brian M, Lefker, Bruce A, Hoge, Garrett S, Lovdahl, Mark J, Asbill, Jeffrey, Carroll, Matthew, Meade, Mary Ann, Ciotti, Susan M, Krieger-Burke, Theresa
Published in Journal of medicinal chemistry (13.11.2008)
Published in Journal of medicinal chemistry (13.11.2008)
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Journal Article
AlMe3-Promoted Formation of Amides from Acids and Amines
Li, Jianqing, Subramaniam, Krishnananthan, Smith, Daniel, Qiao, Jennifer X, Li, Jie Jack, Qian-Cutrone, Jingfang, Kadow, John F, Vite, Gregory D, Chen, Bang-Chi
Published in Organic letters (06.01.2012)
Published in Organic letters (06.01.2012)
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Journal Article
Sulfonimidation via ring-opening of 2-oxazolines with acidic sulfonimide nucleophiles
Gutierrez, David A., Dean, Dayton R., Laxamana, Candace M., Migliozzi-Smith, Madyson, O’Brien, Connor J., O’Neill, Claire L., Li, Jie Jack
Published in ARKIVOC (15.06.2016)
Published in ARKIVOC (15.06.2016)
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Quinazolinones and Pyrido[3,4-d]pyrimidin-4-ones as Orally Active and Specific Matrix Metalloproteinase-13 Inhibitors for the Treatment of Osteoarthritis
Li, Jie Jack, Nahra, Joe, Johnson, Adam R, Bunker, Amy, O’Brien, Patrick, Yue, Wen-Song, Ortwine, Daniel F, Man, Chiu-Fai, Baragi, Vijay, Kilgore, Kenneth, Dyer, Richard D, Han, Hyo-Kyung
Published in Journal of medicinal chemistry (28.02.2008)
Published in Journal of medicinal chemistry (28.02.2008)
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Journal Article
Synthesis and structure–Activity relationship of 2-amino-3-heteroaryl-quinoxalines as non-peptide, small-Molecule antagonists for interleukin-8 receptor
Li, Jie Jack, Carson, Kenneth G, Trivedi, Bharat K, Yue, Wen Song, Ye, Qing, Glynn, Roberta A, Miller, Steven R, Connor, David T, Roth, Bruce D, Luly, Jay R, Low, Joseph E, Heilig, David J, Yang, Weixing, Qin, Shixin, Hunt, Stephen
Published in Bioorganic & medicinal chemistry (15.08.2003)
Published in Bioorganic & medicinal chemistry (15.08.2003)
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Journal Article
An update on the discovery and development of reversible covalent inhibitors
Faridoon, Ng, Raymond, Zhang, Guiping, Li, Jie Jack
Published in Medicinal chemistry research (2023)
Published in Medicinal chemistry research (2023)
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Journal Article
Medicinal chemistry insights into non-hydroxamate HDAC6 selective inhibitors
Faridoon, Zha, Yuqi Lavender, Zhang, Guiping, Li, Jie Jack
Published in Medicinal chemistry research (2023)
Published in Medicinal chemistry research (2023)
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