An Angle on MK2 Inhibition—Optimization and Evaluation of Prevention of Activation Inhibitors
Hedström, Ulf, Norberg, Monica, Evertsson, Emma, Lever, Sarah R., Munck af Rosenschöld, Magnus, Lönn, Hans, Bold, Peter, Käck, Helena, Berntsson, Pia, Vinblad, Johanna, Liu, Jianming, Welinder, Anette, Karlsson, Johan, Snijder, Arjan, Pardali, Katerina, Andersson, Ulf, Davis, Andrew M., Mogemark, Mickael
Published in ChemMedChem (04.10.2019)
Published in ChemMedChem (04.10.2019)
Get full text
Journal Article
Effects of heating rate, temperature and iron catalysis on the thermal behaviour and decompostion of 2-nitrobenzoyl chloride
Get full text
Journal Article
Conference Proceeding
Discovery of AZD8154, a Dual PI3K gamma delta Inhibitor for the Treatment of Asthma
Perry, Matthew W. D., Bjorhall, Karin, Bold, Peter, Brulls, Mikael, Borjesson, Ulf, Carlsson, Johan, Chang, Hui-Fang Amy, Chen, Yunhua, Eriksson, Anders, Fihn, Britt-Marie, Fransson, Rebecca, Fredlund, Linda, Ge, Hongbin, Huang, Haijuan, Karabelas, Kostas, Bergstrom, Eva Lamm, Lever, Sarah, Lindmark, Helena, Mogemark, Mickael, Nikitidis, Antonios, Palmgren, Anna-Pia, Pemberton, Nils, Petersen, Jens, Blomqvist, Mio Rodrigo, Smith, Reed W., Thomas, Matthew J., Ullah, Victoria, Tyrchan, Christian, Wennberg, Tiiu, Eriksson, Annika Westin, Yang, Wenzhen, Zhao, Shuchun, Oster, Linda
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
Get full text
Journal Article
Discovery of Highly Isoform Selective Orally Bioavailable Phosphoinositide 3‑Kinase (PI3K)‑γ Inhibitors
Pemberton, Nils, Mogemark, Mickael, Arlbrandt, Susanne, Bold, Peter, Cox, Rhona J, Gardelli, Cristina, Holden, Neil S, Karabelas, Kostas, Karlsson, Johan, Lever, Sarah, Li, Xueshan, Lindmark, Helena, Norberg, Monica, Perry, Matthew W. D, Petersen, Jens, Rodrigo Blomqvist, Sandra, Thomas, Matthew, Tyrchan, Christian, Westin Eriksson, Annika, Zlatoidsky, Pavol, Öster, Linda
Published in Journal of medicinal chemistry (28.06.2018)
Published in Journal of medicinal chemistry (28.06.2018)
Get full text
Journal Article
AZD0284, a Potent, Selective, and Orally Bioavailable Inverse Agonist of Retinoic Acid Receptor-Related Orphan Receptor C2
Narjes, Frank, Llinas, Antonio, von Berg, Stefan, Jirholt, Johan, Lever, Sarah, Pehrson, Rikard, Collins, Mia, Malmberg, Anna, Svanberg, Petter, Xue, Yafeng, Olsson, Roine I, Malmberg, Jesper, Hughes, Glyn, Hossain, Nafizal, Grindebacke, Hanna, Leffler, Agnes, Krutrök, Nina, Bäck, Elisabeth, Ramnegård, Marie, Lepistö, Matti, Thunberg, Linda, Aagaard, Anna, McPheat, Jane, Hansson, Eva L, Chen, Rongfeng, Xiong, Yao, Hansson, Thomas G
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
Get full text
Journal Article
Discovery of AZD8154, a Dual PI3Kγδ Inhibitor for the Treatment of Asthma
Perry, Matthew W. D, Björhall, Karin, Bold, Peter, Brűlls, Mikael, Börjesson, Ulf, Carlsson, Johan, Chang, Hui-Fang Amy, Chen, Yunhua, Eriksson, Anders, Fihn, Britt-Marie, Fransson, Rebecca, Fredlund, Linda, Ge, Hongbin, Huang, Haijuan, Karabelas, Kostas, Lamm Bergström, Eva, Lever, Sarah, Lindmark, Helena, Mogemark, Mickael, Nikitidis, Antonios, Palmgren, Anna-Pia, Pemberton, Nils, Petersen, Jens, Rodrigo Blomqvist, Mio, Smith, Reed W, Thomas, Matthew J, Ullah, Victoria, Tyrchan, Christian, Wennberg, Tiiu, Westin Eriksson, Annika, Yang, Wenzhen, Zhao, Shuchun, Öster, Linda
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
Get full text
Journal Article
Fertility-sparing Surgery for Presumed Early-stage Invasive Cervical Cancer: A Survey of Practice in the United Kingdom
Tzafetas, Menelaos, Mitra, Anita, Kalliala, Ilkka, Lever, Sarah, Fotopoulou, Christina, Farthing, Alan, Smith, John Richard, Martin-Hirsch, Pierre, Paraskevaidis, Evangelos, Kyrgiou, Maria
Published in Anticancer research (01.06.2018)
Published in Anticancer research (01.06.2018)
Get full text
Journal Article
Front Cover: An Angle on MK2 Inhibition—Optimization and Evaluation of Prevention of Activation Inhibitors (ChemMedChem 19/2019)
Hedström, Ulf, Norberg, Monica, Evertsson, Emma, Lever, Sarah R., Munck af Rosenschöld, Magnus, Lönn, Hans, Bold, Peter, Käck, Helena, Berntsson, Pia, Vinblad, Johanna, Liu, Jianming, Welinder, Anette, Karlsson, Johan, Snijder, Arjan, Pardali, Katerina, Andersson, Ulf, Davis, Andrew M., Mogemark, Mickael
Published in ChemMedChem (04.10.2019)
Published in ChemMedChem (04.10.2019)
Get full text
Journal Article
Lead optimisation of pyrazoles as novel FPR1 antagonists
Morley, Andrew D., King, Sarah, Roberts, Bryan, Lever, Sarah, Teobald, Barry, Fisher, Adrian, Cook, Tony, Parker, Beth, Wenlock, Mark, Phillips, Caroline, Grime, Ken
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Get full text
Journal Article
Discovery of pyrazoles as novel FPR1 antagonists
Morley, Andrew D., Cook, Andrew, King, Sarah, Roberts, Bryan, Lever, Sarah, Weaver, Richard, MacDonald, Cathy, Unitt, John, Fagura, Malbinder, Phillips, Tim, Lewis, Richard, Wenlock, Mark
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
Published in Bioorganic & medicinal chemistry letters (01.11.2011)
Get full text
Journal Article
Study of condition-dependent decomposition reactions. Part I. The thermal behaviour and decomposition of 2-nitrobenzoyl chloride
Get full text
Conference Proceeding
Journal Article
ISOINDOLE COMPOUNDS
LEVER, SARAH, OLSSON, ROINE, INGEMAR, VON BERG, STEFAN, NARJES, FRANK
Year of Publication 24.03.2023
Get full text
Year of Publication 24.03.2023
Patent
ISOINDOLE COMPOUNDS
OLSSON, Roine, Ingemar, NARJES, Frank, VON BERG, Stefan, LEVER, Sarah
Year of Publication 06.07.2022
Get full text
Year of Publication 06.07.2022
Patent