Novel naphthyridines are histamine H sub(3) antagonists and serotonin reuptake transporter inhibitors
Letavic, Michael A, Keith, John M, Ly, Kiev S, Barbier, Ann J, Boggs, Jamin D, Wilson, Sandy J, Lord, Brian, Lovenberg, Timothy W, Carruthers, Nicholas I
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
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Journal Article
Synthesis and biological activity of piperazine and diazepane amides that are histamine H sub(3) antagonists and serotonin reuptake inhibitors
Ly, Kiev S, Letavic, Michael A, Keith, John M, Miller, Jennifer M, Stocking, Emily M, Barbier, Ann J, Bonaventure, Pascal, Lord, Brian, Jiang, Xiaohui, Boggs, Jamin D, Dvorak, Lisa, Miller, Kirsten L, Nepomuceno, Diane, Wilson, Sandy J, Carruthers, Nicholas I
Published in Bioorganic & medicinal chemistry (01.01.2008)
Published in Bioorganic & medicinal chemistry (01.01.2008)
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Journal Article
2-Aryloxymethylmorpholine histamine H 3 antagonists
Letavic, Michael A., Keith, John M., Ly, Kiev S., Bonaventure, Pascal, Feinstein, Mark A., Lord, Brian, Miller, Kirsten L., Motley, S. Timothy, Nepomuceno, Diane, Sutton, Steven W., Carruthers, Nicholas I.
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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Journal Article
Dual serotonin transporter/histamine H sub(3) ligands: Optimization of the H sub(3) pharmacophore
Keith, John M, Gomez, Leslie A, Letavic, Michael A, Ly, Kiev S, Jablonowski, Jill A, Seierstad, Mark, Barbier, Ann J, Wilson, Sandy J, Boggs, Jamin D, Fraser, Ian C, Mazur, Curt, Lovenberg, Timothy W, Carruthers, Nicholas I
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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Journal Article
SUBSTITUTED 4-AZAINDOLES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
RECH, JASON C, WALL, JESSICA L, LETAVIC, MICHAEL A, CHROVIAN, CHRISTA C, SOYODE-JOHNSON, AKINOLA
Year of Publication 03.10.2023
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Year of Publication 03.10.2023
Patent
P2X7 MODULATING N-ACYL-TRIAZOLOPYRAZINES
RECH, JASON C, ANDRES GIL, JOSE IGNACIO, LETAVIC, MICHAEL A, RUDOLPH, DALE A, SOYODE-JOHNSON, AKINOLA, CHROVIAN, CHRISTA C
Year of Publication 03.10.2023
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Year of Publication 03.10.2023
Patent
Novel tetrahydroisoquinolines are histamine H@@d3@ antagonists and serotonin reuptake inhibitors
Letavic, Michael A, Keith, John M, Jablonowski, Jill A, Stocking, Emily M, Gomez, Leslie A, Ly, Kiev S, Miller, Jennifer M, Barbier, Ann J, Bonaventure, Pascal, Boggs, Jamin D, Wilson, Sandy J, Miller, Kirsten L, Lord, Brian, McAllister, Heather M, Tognarelli, D J, Wu, Jiejun, Abad, Marta C, Schubert, Carsten, Lovenberg, Timothy W, Carruthers, Nicholas I
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
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Journal Article
Synthesis of a histamine H(3) receptor antagonist-manipulation of hydroxyproline stereochemistry, desymmetrization of homopiperazine, and nonextractive sodium triacetoxyborohydride reaction workup
Pippel, Daniel J, Young, Lana K, Letavic, Michael A, Ly, Kiev S, Naderi, Bita, Soyode-Johnson, Aki, Stocking, Emily M, Carruthers, Nicholas I, Mani, Neelakandha S
Published in Journal of organic chemistry (02.07.2010)
Published in Journal of organic chemistry (02.07.2010)
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Journal Article
SUBSTITUTED PYRAZOLO[4,3-b]PYRIDINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
LETAVIC, Michael A, SAMANT, Andrew, DVORAK, Curt, WALL, Jessica, HISCOX, Afton, GELIN, Christine, STENNE, Brice
Year of Publication 13.10.2022
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Year of Publication 13.10.2022
Patent
SUBSTITUTED PYRAZOLO-PYRIDINE AMIDES AND THEIR USE AS GLUN2B RECEPTOR
LETAVIC, Michael A, SAMANT, Andrew, DVORAK, Curt, HISCOX, Afton, CHROVIAN, Christa, SOYODE-JOHNSON, Akinola, GELIN, Christine, STENNE, Brice
Year of Publication 18.05.2023
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Year of Publication 18.05.2023
Patent
SUBSTITUTED PYRAZOLO[4,3-B]PYRIDINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
LETAVIC, Michael A, SAMANT, Andrew, DVORAK, Curt, WALL, Jessica, HISCOX, Afton, GELIN, Christine, STENNE, Brice
Year of Publication 20.04.2022
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Year of Publication 20.04.2022
Patent