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Published in Bioorganic & medicinal chemistry letters (15.02.2007)
Published in Bioorganic & medicinal chemistry letters (15.02.2007)
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Novel substituted pyrrolidines are high affinity histamine H3 receptor antagonists
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Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Novel naphthyridines are histamine H3 antagonists and serotonin reuptake transporter inhibitors
LETAVIC, Michael A, KEITH, John M, LY, Kiev S, BARBIER, Ann J, BOGGS, Jamin D, WILSON, Sandy J, LORD, Brian, LOVENBERG, Timothy W, CARRUTHERS, Nicholas I
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
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2-Aryloxymethylmorpholine histamine H(3) antagonists
Letavic, Michael A, Keith, John M, Ly, Kiev S, Bonaventure, Pascal, Feinstein, Mark A, Lord, Brian, Miller, Kirsten L, Motley, S Timothy, Nepomuceno, Diane, Sutton, Steven W, Carruthers, Nicholas I
Published in Bioorganic & medicinal chemistry letters (01.11.2008)
Published in Bioorganic & medicinal chemistry letters (01.11.2008)
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2-Aryloxymethylmorpholine histamine H3 antagonists
LETAVIC, Michael A, KEITH, John M, CARRUTHERS, Nicholas I, LY, Kiev S, BONAVENTURE, Pascal, FEINSTEIN, Mark A, LORD, Brian, MILLER, Kirsten L, MOTLEY, S. Timothy, NEPOMUCENO, Diane, SUTTON, Steven W
Published in Bioorganic & medicinal chemistry letters (01.11.2008)
Published in Bioorganic & medicinal chemistry letters (01.11.2008)
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Benzylamine histamine H3 antagonists and serotonin reuptake inhibitors
LETAVIC, Michael A, STOCKING, Emily M, BARBIER, Ann J, BONAVENTURE, Pascal, BOGGS, Jamin D, LORD, Brian, MILLER, Kirsten L, WILSON, Sandy J, CARRUTHERS, Nicholas I
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
Published in Bioorganic & medicinal chemistry letters (01.09.2007)
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Pre-clinical characterization of aryloxypyridine amides as histamine H3 receptor antagonists: Identification of candidates for clinical development
Letavic, Michael A., Aluisio, Leah, Atack, John R., Bonaventure, Pascal, Carruthers, Nicholas I., Dugovic, Christine, Everson, Anita, Feinstein, Mark A., Fraser, Ian C., Hoey, Kenway, Jiang, Xiaohui, Keith, John M., Koudriakova, Tatiana, Leung, Perry, Lord, Brian, Lovenberg, Timothy W., Ly, Kiev S., Morton, Kirsten L., Timothy Motley, S., Nepomuceno, Diane, Rizzolio, Michele, Rynberg, Raymond, Sepassi, Kia, Shelton, Jonathan
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
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Synthesis and biological activity of selective pipecolic acid-based TNF-α converting enzyme (TACE) inhibitors
Letavic, Michael A., Axt, Matt Z., Barberia, John T., Carty, Thomas J., Danley, Dennis E., Geoghegan, Kieran F., Halim, Nadia S., Hoth, Lise R., Kamath, Ajith V., Laird, Ellen R., Lopresti-Morrow, Lori L., McClure, Kim F., Mitchell, Peter G., Natarajan, Vijayalakshmi, Noe, Mark C., Pandit, Jayvardhan, Reeves, Lisa, Schulte, Gayle K., Snow, Sheri L., Sweeney, Francis J., Tan, Douglas H., Yu, Chul H.
Published in Bioorganic & medicinal chemistry letters (20.05.2002)
Published in Bioorganic & medicinal chemistry letters (20.05.2002)
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Structure–activity relationships of triazolopyridine oxazole p38 inhibitors: Identification of candidates for clinical development
McClure, Kim F., Letavic, Michael A., Kalgutkar, Amit S., Gabel, Christopher A., Audoly, Laurent, Barberia, John T., Braganza, John F., Carter, Demetrius, Carty, Thomas J., Cortina, Santo R., Dombroski, Mark A., Donahue, Kathleen M., Elliott, Nancy C., Gibbons, Colleen P., Jordan, Crystal K., Kuperman, Alexander V., Labasi, Jeff M., LaLiberte, Ronald E., McCoy, Jennifer M., Naiman, Brian M., Nelson, Kendra L., Nguyen, Hang T., Peese, Kevin M., Sweeney, Francis J., Taylor, Timothy J., Trebino, Catherine E., Abramov, Yuriy A., Laird, Ellen R., Volberg, Walter A., Zhou, Jun, Bach, Justin, Lombardo, Franco
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Year of Publication 13.04.2023
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Year of Publication 13.04.2023
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Benzimidazolone p38 inhibitors
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Published in Bioorganic & medicinal chemistry letters (23.02.2004)
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
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Year of Publication 07.04.2022
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Year of Publication 07.04.2022
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Asymmetric Reactions of 2-Methoxy-1,4-benzoquinones with Styrenyl Systems: Enantioselective Syntheses of 8-Aryl-3-methoxybicyclo[4.2.0]oct-3-en-2,5-diones, 7-Aryl-3-hydroxybicyclo[3.2.1]oct-3-en-2,8-diones, 2-Aryl-6-methoxy-2,3-dihydrobenzofuran-5-ols, and Pterocarpans
Engler, Thomas A, Letavic, Michael A, Iyengar, Rajesh, LaTessa, Kenneth O, Reddy, Jayachandra P
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Year of Publication 13.03.2018
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Year of Publication 13.03.2018
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Synthesis and Activity of a Novel Class of Tribasic Macrocyclic Antibiotics: The Triamilides
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LETAVIC MICHAEL A, STENNE BRICE M, CHROVIAN CHRISTA C, JOHNSON AKINOLA SOYODE, RUDOLPH DALE A, RECH JASON C, WALL JESSICA L
Year of Publication 24.05.2019
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Year of Publication 24.05.2019
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Synthesis and biological activity of piperazine-Based dual MMP-13 and TNF-α converting enzyme inhibitors
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Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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NR2B-선택적 NMDA 조절제로서 치환된 1,2,3-트라이아졸
CHEN GANG, LETAVIC MICHAEL A, HISCOX AFTON, CHROVIAN CHRISTA C, GELIN CHRISTINE F, STENNE BRICE, DVORAK CURT A, COATE HEATHER R, RECH JASON C, SOYODE JOHNSON AKINOLA, WALL JESSICA L, ZHANG WEI
Year of Publication 04.10.2018
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Year of Publication 04.10.2018
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34- DISUBSTITUTED OCTAHYDROPYRROLO[34-c]PYRROLES AS OREXIN RECEPTOR MODULATORS
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Year of Publication 11.12.2017
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Year of Publication 11.12.2017
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