Increased Potency and Selectivity for Group III Metabotropic Glutamate Receptor Agonists Binding at Dual sites
Selvam, Chelliah, Lemasson, Isabelle A, Brabet, Isabelle, Oueslati, Nadia, Karaman, Berin, Cabaye, Alexandre, Tora, Amélie S, Commare, Bruno, Courtiol, Tiphanie, Cesarini, Sara, McCort-Tranchepain, Isabelle, Rigault, Delphine, Mony, Laetitia, Bessiron, Thomas, McLean, Heather, Leroux, Frédéric R, Colobert, Françoise, Daniel, Hervé, Goupil-Lamy, Anne, Bertrand, Hugues-Olivier, Goudet, Cyril, Pin, Jean-Philippe, Acher, Francine C
Published in Journal of medicinal chemistry (08.03.2018)
Published in Journal of medicinal chemistry (08.03.2018)
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Stereoselective Synthesis of o-Bromo (or Iodo)aryl P-Chirogenic Phosphines Based on Aryne Chemistry
Bayardon, Jérôme, Laureano, Hugo, Diemer, Vincent, Dutartre, Mathieu, Das, Utpal, Rousselin, Yoann, Henry, Jean-Christophe, Colobert, Françoise, Leroux, Frédéric R, Jugé, Sylvain
Published in Journal of organic chemistry (06.07.2012)
Published in Journal of organic chemistry (06.07.2012)
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A fluorine scan of a tubulin polymerization inhibitor isocombretastatin A-4: Design, synthesis, molecular modelling, and biological evaluation
Naret, Timothée, Bignon, Jérôme, Bernadat, Guillaume, Benchekroun, Mohamed, Levaique, Helene, Lenoir, Christine, Dubois, Joelle, Pruvost, Alain, Saller, François, Borgel, Delphine, Manoury, Boris, Leblais, Veronique, Darrigrand, Romain, Apcher, Sébastien, Brion, Jean-Daniel, Schmitt, Etienne, Leroux, Frédéric R., Alami, Mouad, Hamze, Abdallah
Published in European journal of medicinal chemistry (01.01.2018)
Published in European journal of medicinal chemistry (01.01.2018)
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Triazolopyridines. Part 28. The ring–chain isomerization strategy: triazolopyridine- and triazoloquinoline–pyridine based fluorescence ligands
Ballesteros-Garrido, Rafael, Delgado-Pinar, Estefanía, Abarca, Belén, Ballesteros, Rafael, Leroux, Frédéric R., Colobert, Françoise, Zaragozá, Ramón J., García-España, Enrique
Published in Tetrahedron (13.05.2012)
Published in Tetrahedron (13.05.2012)
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Synthesis and structural properties of hexaaza[5]helicene containing two [1,2,3]triazolo[1,5-a]pyridine moieties
Adam, Rosa, Ballesteros-Garrido, Rafael, Vallcorba, Oriol, Abarca, Belén, Ballesteros, Rafael, Leroux, Frédéric R., Colobert, Françoise, Amigó, José M., Rius, Jordi
Published in Tetrahedron letters (07.08.2013)
Published in Tetrahedron letters (07.08.2013)
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Recent advances in transition metal-catalyzed Csp(2)-monofluoro-, difluoro-, perfluoromethylation and trifluoromethylthiolation
Landelle, Grégory, Panossian, Armen, Pazenok, Sergiy, Vors, Jean-Pierre, Leroux, Frédéric R
Published in Beilstein journal of organic chemistry (15.11.2013)
Published in Beilstein journal of organic chemistry (15.11.2013)
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Palladium‐Catalyzed Silylcyanation of Ynamides: Regio‐ and Stereoselective Access to Tetrasubstituted 3‐Silyl‐2‐Aminoacrylonitriles
Hansjacob, Pierre, Leroux, Frédéric R., Gandon, Vincent, Donnard, Morgan
Published in Angewandte Chemie International Edition (28.03.2022)
Published in Angewandte Chemie International Edition (28.03.2022)
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Ketenimines as Intermediates To Access Difluoromethoxylated Scaffolds
Loison, Anaïs, Hanquet, Gilles, Toulgoat, Fabien, Billard, Thierry, Panossian, Armen, Leroux, Frédéric R.
Published in Organic letters (18.11.2022)
Published in Organic letters (18.11.2022)
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Recent advances in transition metal-catalyzed Csp2-monofluoro-, difluoro-, perfluoromethylation and trifluoromethylthiolation
Landelle, Grégory, Panossian, Armen, Pazenok, Sergiy, Vors, Jean-Pierre, Leroux, Frédéric R
Published in Beilstein journal of organic chemistry (15.11.2013)
Published in Beilstein journal of organic chemistry (15.11.2013)
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Deprotonative Functionalization of the Difluoromethyl Group
Santos, Laura, Panossian, Armen, Donnard, Morgan, Vors, Jean-Pierre, Pazenok, Sergii, Bernier, David, Leroux, Frédéric R
Published in Organic letters (06.11.2020)
Published in Organic letters (06.11.2020)
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Study of a Stable “Trifluoromethoxide Anion Solution” Arising from 2,4‐Dinitro‐Trifluoromethoxybenzene
Bonnefoy, Clémence, Chefdeville, Emmanuel, Panosian, Armen, Hanquet, Gilles, Leroux, Frédéric R., Toulgoat, Fabien, Billard, Thierry
Published in Chemistry : a European journal (17.11.2021)
Published in Chemistry : a European journal (17.11.2021)
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