Discovery of ANA975: An Oral Prodrug of the TLR-7 Agonist Isatoribine
Xiang, Alan X., Webber, Stephen E., Kerr, Bradley M., Rueden, Erik J., Lennox, Joseph R., Haley, Gregory J., Wang, Tingmin, Ng, John S., Herbert, Mark R., Clark, David L., Banh, Virginia N., Li, Wei, Fletcher, Simon P., Steffy, Kevin R., Bartkowski, Darian M., Kirkovsky, Leonid I., Bauman, Lisa A., Averett, Devron R.
Published in Nucleosides, nucleotides & nucleic acids (26.11.2007)
Published in Nucleosides, nucleotides & nucleic acids (26.11.2007)
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Synthesis and bladder smooth muscle relaxing properties of substituted 3-amino-4-aryl-(and aralkyl-)cyclobut-3-ene-1,2-diones
Butera, John A., Jenkins, Douglas J., Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N. Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
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Journal Article
Synthesis and potassium channel opening activity of substituted 10H-benzo[4,5]furo[3,2-b]indole- and 5,10-dihydro-indeno[1,2-b]indole-1-carboxylic acids
BUTERA, John A, ANTANE, Schuyler A, HIRTH, Bradford, LENNOX, Joseph R, SHELDON, Jeffrey H, NORTON, N. Wesley, WARGA, Dawn, ARGENTIERI, Thomas M
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 1. N-Cyanoguanidine Bioisosteres Possessing in Vivo Bladder Selectivity
Butera, John A, Antane, Madelene M, Antane, Schuyler A, Argentieri, Thomas M, Freeden, Chris, Graceffa, Russell F, Hirth, Bradford H, Jenkins, Douglas, Lennox, Joseph R, Matelan, Edward, Norton, N. Wesley, Quagliato, Dominick, Sheldon, Jeffrey H, Spinelli, Walter, Warga, Dawn, Wojdan, Alexandra, Woods, Morgan
Published in Journal of medicinal chemistry (23.03.2000)
Published in Journal of medicinal chemistry (23.03.2000)
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Journal Article
Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 2. Selective and Potent Benzylamino Cyclobutenediones
Gilbert, Adam M, Antane, Madelene M, Argentieri, Thomas M, Butera, John A, Francisco, Gerardo D, Freeden, Chris, Gundersen, Eric G, Graceffa, Russell F, Herbst, David, Hirth, Bradford H, Lennox, Joseph R, McFarlane, Geraldine, Norton, N. Wesley, Quagliato, Dominick, Sheldon, Jeffrey H, Warga, Dawn, Wojdan, Alexandra, Woods, Morgan
Published in Journal of medicinal chemistry (23.03.2000)
Published in Journal of medicinal chemistry (23.03.2000)
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Synthesis and potassium channel opening activity of substituted 10H-Benzofuro[3,2-b]indole- and 5,10-Dihydro-indeno[1,2-b]indole-1-carboxylic acids
Butera, John A., Antane, Schuyler A., Hirth, Bradford, Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N.Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (01.08.2001)
Published in Bioorganic & medicinal chemistry letters (01.08.2001)
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Journal Article
Synthesis and potassium channel opening activity of substituted 10 H-Benzo [4,5]furo[3,2- b]indole- and 5,10-Dihydro-indeno[1,2- b]indole-1-carboxylic acids
Butera, John A., Antane, Schuyler A., Hirth, Bradford, Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N.Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (2001)
Published in Bioorganic & medicinal chemistry letters (2001)
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compostos, sais ou hidratos farmaceuticamente aceitos, composição farmacêutica e uso de quantidade terapeutica ou profilaticamente eficaz de composto ou de composição farmacêutica
Stephen E. Webber, Erik J. Rueden, Joseph R. Lennox, Alan X. Xiang, Gregory J. Haley
Year of Publication 25.05.2021
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Year of Publication 25.05.2021
Patent
compostos, sais ou hidratos farmaceuticamente aceitos, composição farmacêutica e uso de quantidade terapeutica ou profilaticamente eficaz de composto ou de composição farmacêutica
Stephen E. Webber, Erik J. Rueden, Joseph R. Lennox, Alan X. Xiang, Gregory J. Haley
Year of Publication 09.03.2021
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Year of Publication 09.03.2021
Patent
PRODRUGS OF 5-AMINO-3-(3'-DEOXY-.BETA.-D-RIBOFURANOSYL)-THIAZOLO[4,5-D]PYRIMIDIN-2,7-DIONE
HALEY, GREGORY J, LENNOX, JOSEPH R, XIANG, ALAN XIN, WEBBER, STEPHEN E
Year of Publication 18.11.2014
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Year of Publication 18.11.2014
Patent